KR20020000636A - 티오-옥신돌 유도체 - Google Patents

티오-옥신돌 유도체 Download PDF

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Publication number
KR20020000636A
KR20020000636A KR1020017014076A KR20017014076A KR20020000636A KR 20020000636 A KR20020000636 A KR 20020000636A KR 1020017014076 A KR1020017014076 A KR 1020017014076A KR 20017014076 A KR20017014076 A KR 20017014076A KR 20020000636 A KR20020000636 A KR 20020000636A
Authority
KR
South Korea
Prior art keywords
alkyl
substituted
aryl
csnh
conh
Prior art date
Application number
KR1020017014076A
Other languages
English (en)
Korean (ko)
Inventor
펜섬앤드류
장푸웬
코코마르시씨.
지린
존즈토드케이.
테글리크리스토퍼엠.
로벨제이이.
에드워즈제임즈피.
멜렌스키에드워드지.
Original Assignee
이곤 이 버그
아메리칸 홈 푸로닥츠 코포레이션
윌리암 엘. 레스페스
리간드 파마슈티칼스 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/552,033 external-priority patent/US6355648B1/en
Application filed by 이곤 이 버그, 아메리칸 홈 푸로닥츠 코포레이션, 윌리암 엘. 레스페스, 리간드 파마슈티칼스 인코포레이티드 filed Critical 이곤 이 버그
Publication of KR20020000636A publication Critical patent/KR20020000636A/ko

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/40—Nitrogen atoms, not forming part of a nitro radical, e.g. isatin semicarbazone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
KR1020017014076A 1999-05-04 2000-05-01 티오-옥신돌 유도체 KR20020000636A (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US17225999P 1999-05-04 1999-05-04
US60/172,259 1999-05-04
US09/552,033 US6355648B1 (en) 1999-05-04 2000-04-19 Thio-oxindole derivatives
US09/552,033 2000-04-19
PCT/US2000/011630 WO2000066555A1 (en) 1999-05-04 2000-05-01 Thio-oxindole derivatives

Publications (1)

Publication Number Publication Date
KR20020000636A true KR20020000636A (ko) 2002-01-05

Family

ID=26867898

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017014076A KR20020000636A (ko) 1999-05-04 2000-05-01 티오-옥신돌 유도체

Country Status (18)

Country Link
EP (1) EP1181275A1 (zh)
JP (1) JP2002543182A (zh)
KR (1) KR20020000636A (zh)
CN (1) CN1143847C (zh)
AU (1) AU767762B2 (zh)
BG (1) BG106078A (zh)
BR (1) BR0010216A (zh)
CA (1) CA2371633A1 (zh)
CZ (1) CZ20013950A3 (zh)
EA (1) EA005034B1 (zh)
GE (1) GEP20043266B (zh)
HU (1) HUP0200993A3 (zh)
MX (1) MXPA01011285A (zh)
NO (1) NO320912B1 (zh)
NZ (1) NZ515351A (zh)
PL (1) PL351407A1 (zh)
SK (1) SK15902001A3 (zh)
TR (1) TR200103288T2 (zh)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11724982B2 (en) 2014-10-10 2023-08-15 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA06011695A (es) * 2004-04-08 2006-12-14 Wyeth Corp Metodos para minimizar las impurezas de tioamida.
DK1732921T3 (da) * 2004-04-08 2009-02-23 Wyeth Corp Thiomidderivater som progesteronreceptormodulatorer
GB201113538D0 (en) * 2011-08-04 2011-09-21 Karobio Ab Novel estrogen receptor ligands
CN104995194B (zh) * 2012-10-12 2017-08-29 学校法人冲绳科学技术大学院大学学园 螺环吲哚衍生物及其制备方法
WO2018064557A1 (en) * 2016-09-30 2018-04-05 Epizyme, Inc. Substituted fused bi- or tri- heterocyclic compounds as ehmt2 inhibitors

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11724982B2 (en) 2014-10-10 2023-08-15 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration

Also Published As

Publication number Publication date
NO20015380L (no) 2002-01-03
AU767762B2 (en) 2003-11-20
SK15902001A3 (sk) 2002-11-06
CN1349499A (zh) 2002-05-15
CN1143847C (zh) 2004-03-31
NO320912B1 (no) 2006-02-13
MXPA01011285A (es) 2003-09-04
NZ515351A (en) 2004-01-30
EA200101180A1 (ru) 2002-04-25
JP2002543182A (ja) 2002-12-17
GEP20043266B (en) 2004-06-25
TR200103288T2 (tr) 2002-04-22
EP1181275A1 (en) 2002-02-27
CZ20013950A3 (cs) 2002-06-12
BR0010216A (pt) 2002-03-19
PL351407A1 (en) 2003-04-22
AU4681400A (en) 2000-11-17
EA005034B1 (ru) 2004-10-28
CA2371633A1 (en) 2000-11-09
BG106078A (en) 2002-05-31
HUP0200993A2 (hu) 2002-07-29
NO20015380D0 (no) 2001-11-02
HUP0200993A3 (en) 2003-05-28

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Legal Events

Date Code Title Description
A201 Request for examination
E902 Notification of reason for refusal
N231 Notification of change of applicant
E601 Decision to refuse application