KR102854313B1 - 융합된 비시클릭 sGC 자극제 - Google Patents

융합된 비시클릭 sGC 자극제

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Publication number
KR102854313B1
KR102854313B1 KR1020237027632A KR20237027632A KR102854313B1 KR 102854313 B1 KR102854313 B1 KR 102854313B1 KR 1020237027632 A KR1020237027632 A KR 1020237027632A KR 20237027632 A KR20237027632 A KR 20237027632A KR 102854313 B1 KR102854313 B1 KR 102854313B1
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South Korea
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compound
pharmaceutically acceptable
acceptable salt
disease
alkyl
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KR20230124760A (ko
Inventor
글렌 로버트 레니
라예시 알. 이옌가르
토마스 와이-호 리
타카시 나카이
아라 메르메리안
레이 지아
지-윤 제이미 임
폴 알란 렌하우에
준 정
피터 게르마노
카르티크 이예르
티모시 클라우드 바르덴
킴 탕
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티센토 쎄라퓨틱스 인크.
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    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
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    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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KR1020237027632A 2016-09-02 2017-09-01 융합된 비시클릭 sGC 자극제 Active KR102854313B1 (ko)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US201662382942P 2016-09-02 2016-09-02
US62/382,942 2016-09-02
US201662423445P 2016-11-17 2016-11-17
US62/423,445 2016-11-17
US201762468598P 2017-03-08 2017-03-08
US62/468,598 2017-03-08
US201762482486P 2017-04-06 2017-04-06
US62/482,486 2017-04-06
PCT/US2017/049834 WO2018045276A1 (en) 2016-09-02 2017-09-01 Fused bicyclic sgc stimulators
KR1020197008522A KR102568384B1 (ko) 2016-09-02 2017-09-01 융합된 비시클릭 sGC 자극제

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KR20230124760A KR20230124760A (ko) 2023-08-25
KR102854313B1 true KR102854313B1 (ko) 2025-09-04

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