KR102630889B1 - 키나제를 조절하는 화합물의 고형 형태 - Google Patents

키나제를 조절하는 화합물의 고형 형태 Download PDF

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KR102630889B1
KR102630889B1 KR1020177034519A KR20177034519A KR102630889B1 KR 102630889 B1 KR102630889 B1 KR 102630889B1 KR 1020177034519 A KR1020177034519 A KR 1020177034519A KR 20177034519 A KR20177034519 A KR 20177034519A KR 102630889 B1 KR102630889 B1 KR 102630889B1
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KR20180002741A (ko
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프라바 엔. 이브라힘
개리 콘래드 바이저
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다이이치 산쿄 인코포레이티드
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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KR1020177034519A 2015-05-06 2016-05-05 키나제를 조절하는 화합물의 고형 형태 Active KR102630889B1 (ko)

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Application Number Priority Date Filing Date Title
US201562157902P 2015-05-06 2015-05-06
US62/157,902 2015-05-06
PCT/US2016/031027 WO2016179415A1 (en) 2015-05-06 2016-05-05 Solid forms of a compound modulating kinases

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KR20180002741A KR20180002741A (ko) 2018-01-08
KR102630889B1 true KR102630889B1 (ko) 2024-01-30

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US (4) US9802932B2 (enExample)
EP (2) EP3757104A1 (enExample)
JP (1) JP6946194B2 (enExample)
KR (1) KR102630889B1 (enExample)
CN (1) CN107548394B (enExample)
AU (1) AU2016258027B2 (enExample)
BR (1) BR112017023490B1 (enExample)
CA (1) CA2984910C (enExample)
CO (1) CO2017011534A2 (enExample)
CY (1) CY1123796T1 (enExample)
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SI (1) SI3292123T1 (enExample)
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