KR102087020B1 - 1-(5,6-다이클로로-1h-벤조[d]이미다졸-2-일)-1h-피라졸-4-카르복실산의 메글루민 염 제형 - Google Patents

1-(5,6-다이클로로-1h-벤조[d]이미다졸-2-일)-1h-피라졸-4-카르복실산의 메글루민 염 제형 Download PDF

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KR102087020B1
KR102087020B1 KR1020147013440A KR20147013440A KR102087020B1 KR 102087020 B1 KR102087020 B1 KR 102087020B1 KR 1020147013440 A KR1020147013440 A KR 1020147013440A KR 20147013440 A KR20147013440 A KR 20147013440A KR 102087020 B1 KR102087020 B1 KR 102087020B1
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compound
acid
hif
phd
salt
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KR20140094547A (ko
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키아 세파스시
미켈레 체. 리졸리오
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얀센 파마슈티카 엔.브이.
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • A61P19/00—Drugs for skeletal disorders
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A—HUMAN NECESSITIES
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
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    • A61P3/00—Drugs for disorders of the metabolism
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
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  • Child & Adolescent Psychology (AREA)
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  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Inorganic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
KR1020147013440A 2011-10-25 2012-10-25 1-(5,6-다이클로로-1h-벤조[d]이미다졸-2-일)-1h-피라졸-4-카르복실산의 메글루민 염 제형 Expired - Fee Related KR102087020B1 (ko)

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US201161551395P 2011-10-25 2011-10-25
US61/551,395 2011-10-25
PCT/US2012/061847 WO2013063221A1 (en) 2011-10-25 2012-10-25 Meglumine salt formulations of 1-(5,6-dichloro-1h-benzo[d]imidazol-2-yl)-1h-pyrazole-4-carboxylic acid

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KR20140094547A KR20140094547A (ko) 2014-07-30
KR102087020B1 true KR102087020B1 (ko) 2020-03-11

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US (4) US9273034B2 (enExample)
EP (3) EP2776023B1 (enExample)
JP (2) JP6122862B2 (enExample)
KR (1) KR102087020B1 (enExample)
CN (2) CN104053439B (enExample)
AU (2) AU2012328763A1 (enExample)
BR (1) BR112014009910B1 (enExample)
CA (1) CA2853455C (enExample)
CY (1) CY1123426T1 (enExample)
ES (3) ES2689481T3 (enExample)
HU (1) HUE052128T2 (enExample)
IN (1) IN2014DN03155A (enExample)
MX (2) MX368157B (enExample)
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CN104812389B (zh) 2012-09-24 2020-07-17 润新生物公司 某些化学实体、组合物及方法
EP2916838B1 (en) 2012-11-12 2019-03-13 Neupharma, Inc. Certain chemical entities, compositions, and methods
CN104610153B (zh) * 2015-01-19 2017-02-22 沈阳中海生物技术开发有限公司 奥扎格雷葡甲胺盐及其组合物、制备方法和用途
AU2019319448B2 (en) 2018-08-07 2022-06-02 Metagone Biotech Inc. Ammonium salts of 3-(3,5-dibromo-4-hydroxybenzyliden)-5-indo-1,3-dihydroindol-2-one and uses thereof
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AU2017204598A1 (en) 2017-07-27
CN104053439B (zh) 2016-08-24
BR112014009910A2 (pt) 2017-04-25
JP2014530915A (ja) 2014-11-20
MX2014005075A (es) 2014-08-08
MX344109B (es) 2016-12-05
MX368157B (es) 2019-09-20
WO2013063221A1 (en) 2013-05-02
EP3461820B1 (en) 2020-07-29
EP2776023A1 (en) 2014-09-17
US20180201605A1 (en) 2018-07-19
AU2012328763A1 (en) 2014-05-01
CN106038556A (zh) 2016-10-26
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CA2853455A1 (en) 2013-05-02
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