KR102057491B1 - 시스-알콕시-치환된 스피로시클릭 페닐아세틸아미노산 에스테르 및 시스-알콕시-치환된 스피로시클릭 1h-피롤리딘-2,4-디온 유도체의 제조 방법 - Google Patents
시스-알콕시-치환된 스피로시클릭 페닐아세틸아미노산 에스테르 및 시스-알콕시-치환된 스피로시클릭 1h-피롤리딘-2,4-디온 유도체의 제조 방법 Download PDFInfo
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- KR102057491B1 KR102057491B1 KR1020147026703A KR20147026703A KR102057491B1 KR 102057491 B1 KR102057491 B1 KR 102057491B1 KR 1020147026703 A KR1020147026703 A KR 1020147026703A KR 20147026703 A KR20147026703 A KR 20147026703A KR 102057491 B1 KR102057491 B1 KR 102057491B1
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- 0 *c1cc(CC(O2)=N[C@](CC3)(CC[C@]3O*)C2=O)c(*)cc1 Chemical compound *c1cc(CC(O2)=N[C@](CC3)(CC[C@]3O*)C2=O)c(*)cc1 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
- C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C07C233/51—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
- C07C233/52—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a ring other than a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/54—Spiro-condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
- Pyrrole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12161837 | 2012-03-28 | ||
| EP12161837.5 | 2012-03-28 | ||
| PCT/EP2013/056318 WO2013144101A1 (de) | 2012-03-28 | 2013-03-25 | Verfahren zur herstellung von cis-alkoxysubstituierten spirocyclischen phenylacetylaminosäureestern und cis-alkoxysubstituierten spirocyclischen 1-h-pyrrolidin-2,4-dion-derivaten |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20140140045A KR20140140045A (ko) | 2014-12-08 |
| KR102057491B1 true KR102057491B1 (ko) | 2019-12-19 |
Family
ID=47997506
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020147026703A Active KR102057491B1 (ko) | 2012-03-28 | 2013-03-25 | 시스-알콕시-치환된 스피로시클릭 페닐아세틸아미노산 에스테르 및 시스-알콕시-치환된 스피로시클릭 1h-피롤리딘-2,4-디온 유도체의 제조 방법 |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US9376374B2 (enExample) |
| EP (1) | EP2831038B1 (enExample) |
| JP (1) | JP6158293B2 (enExample) |
| KR (1) | KR102057491B1 (enExample) |
| CN (2) | CN104245664B (enExample) |
| BR (1) | BR112014023999B8 (enExample) |
| DK (1) | DK2831038T3 (enExample) |
| ES (1) | ES2644126T3 (enExample) |
| IL (1) | IL234626A (enExample) |
| IN (1) | IN2014DN07407A (enExample) |
| MX (1) | MX349985B (enExample) |
| TW (1) | TWI579260B (enExample) |
| WO (1) | WO2013144101A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10577320B2 (en) * | 2016-05-04 | 2020-03-03 | Bayer Cropscience Aktiengesellschaft | Method for preparing cis-alkoxy-substituted spirocyclic 1-H-pyrrolidine-2,4-dione derivatives |
| EP3301092A3 (de) | 2018-01-26 | 2018-09-12 | Bayer CropScience Aktiengesellschaft | Verfahren zur herstellung von spiroketal-substituierten phenylacetylaminosäureestern und spiroketal-substituierten cyclischen ketoenolen |
| CN115448869B (zh) * | 2021-06-09 | 2024-08-09 | 顺毅南通化工有限公司 | 一种螺虫乙酯合成用中间体的制备方法 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007080882A1 (ja) | 2006-01-11 | 2007-07-19 | Seikagaku Corporation | オキサゾロン誘導体 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2733233A (en) * | 1956-01-31 | Vinyl esters of n-carbacyl-alpha-mono- | ||
| DE4431730A1 (de) * | 1994-02-09 | 1995-08-10 | Bayer Ag | Substituierte 1H-3-Aryl-pyrrolidin-2,4-dion-Derivate |
| CN1075060C (zh) * | 1994-04-05 | 2001-11-21 | 拜尔公司 | 用作除草剂和农药的烷氧基－烷基取代的1－h－3－芳基－吡咯烷－2,4－二酮 |
| JP4036470B2 (ja) * | 1995-02-13 | 2008-01-23 | バイエル・アクチエンゲゼルシヤフト | 除草剤および有害生物防除剤としての２−フェニル置換複素環式１，３−ケトエノール |
| BR9608229A (pt) * | 1995-05-09 | 1998-12-29 | Bayer Ag | Cetoenóis alquil-dihalogenofenil-substituídos |
| RU2195449C2 (ru) * | 1995-06-28 | 2002-12-27 | Байер Акциенгезельшафт | 2,4,5-тризамещенные фенилкетоенолы, промежуточные соединения для их получения, способ и средство для борьбы с насекомыми и паукообразными на их основе |
| DK1277734T3 (da) * | 1996-08-05 | 2007-06-04 | Bayer Cropscience Ag | 2- og 2,5-substituerede phenylketoenoler |
| DE10016544A1 (de) * | 2000-04-03 | 2001-10-11 | Bayer Ag | C2-phenylsubstituierte Ketoenole |
| DE10032587A1 (de) * | 2000-07-05 | 2002-01-17 | Bayer Ag | 4-Alkoxy-cyclohexan-1-amino-carbonsäureester und Verfahren zu ihrer Herstellung |
| DE10231333A1 (de) * | 2002-07-11 | 2004-01-22 | Bayer Cropscience Ag | Cis-Alkoxysubstituierte spirocyclische 1-H-Pyrrolidin-2,4-dion-Derivate |
| DE10239479A1 (de) * | 2002-08-28 | 2004-03-04 | Bayer Cropscience Ag | Substituierte spirocyclische Ketoenole |
| DE102004030753A1 (de) * | 2004-06-25 | 2006-01-19 | Bayer Cropscience Ag | 3'-Alkoxy spirocyclische Tetram- und Tretronsäuren |
| DE102004044827A1 (de) * | 2004-09-16 | 2006-03-23 | Bayer Cropscience Ag | Jod-phenylsubstituierte cyclische Ketoenole |
| JP3975226B2 (ja) * | 2006-01-11 | 2007-09-12 | 生化学工業株式会社 | シクロアルキルカルボニルアミノ酸誘導体及びその製造方法 |
| CN102241590B (zh) * | 2011-05-17 | 2013-06-19 | 永农生物科学有限公司 | 一种螺环季酮酸类化合物关键中间体的合成方法 |
| DE102011080406A1 (de) * | 2011-08-04 | 2013-02-07 | Bayer Pharma AG | Substituierte 3-(Biphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro8[4.5]dec-3-en-2-one |
-
2013
- 2013-03-15 TW TW102109182A patent/TWI579260B/zh active
- 2013-03-25 MX MX2014011577A patent/MX349985B/es active IP Right Grant
- 2013-03-25 IN IN7407DEN2014 patent/IN2014DN07407A/en unknown
- 2013-03-25 BR BR112014023999A patent/BR112014023999B8/pt active IP Right Grant
- 2013-03-25 CN CN201380017552.7A patent/CN104245664B/zh active Active
- 2013-03-25 KR KR1020147026703A patent/KR102057491B1/ko active Active
- 2013-03-25 CN CN201611037398.1A patent/CN106748861B/zh active Active
- 2013-03-25 EP EP13712251.1A patent/EP2831038B1/de active Active
- 2013-03-25 ES ES13712251.1T patent/ES2644126T3/es active Active
- 2013-03-25 DK DK13712251.1T patent/DK2831038T3/en active
- 2013-03-25 WO PCT/EP2013/056318 patent/WO2013144101A1/de not_active Ceased
- 2013-03-25 JP JP2015502287A patent/JP6158293B2/ja active Active
- 2013-03-25 US US14/387,249 patent/US9376374B2/en active Active
-
2014
- 2014-09-14 IL IL234626A patent/IL234626A/en active IP Right Grant
-
2016
- 2016-05-23 US US15/161,978 patent/US9840459B2/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007080882A1 (ja) | 2006-01-11 | 2007-07-19 | Seikagaku Corporation | オキサゾロン誘導体 |
Non-Patent Citations (1)
| Title |
|---|
| 논문 Chemistry and Industry, Vol. 75, pp. 1568 (1968) |
Also Published As
| Publication number | Publication date |
|---|---|
| BR112014023999B8 (pt) | 2020-05-12 |
| CN106748861B (zh) | 2018-10-19 |
| KR20140140045A (ko) | 2014-12-08 |
| IN2014DN07407A (enExample) | 2015-04-24 |
| US9376374B2 (en) | 2016-06-28 |
| TWI579260B (zh) | 2017-04-21 |
| MX349985B (es) | 2017-08-22 |
| JP2015516380A (ja) | 2015-06-11 |
| IL234626A (en) | 2017-07-31 |
| CN104245664B (zh) | 2016-12-07 |
| CN106748861A (zh) | 2017-05-31 |
| EP2831038B1 (de) | 2017-07-19 |
| US20150051407A1 (en) | 2015-02-19 |
| TW201400440A (zh) | 2014-01-01 |
| JP6158293B2 (ja) | 2017-07-05 |
| EP2831038A1 (de) | 2015-02-04 |
| CN104245664A (zh) | 2014-12-24 |
| DK2831038T3 (en) | 2017-10-30 |
| ES2644126T3 (es) | 2017-11-27 |
| MX2014011577A (es) | 2014-11-21 |
| US20160264516A1 (en) | 2016-09-15 |
| US9840459B2 (en) | 2017-12-12 |
| WO2013144101A1 (de) | 2013-10-03 |
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