KR102052983B1 - 펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도 - Google Patents

펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도 Download PDF

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KR102052983B1
KR102052983B1 KR1020177016079A KR20177016079A KR102052983B1 KR 102052983 B1 KR102052983 B1 KR 102052983B1 KR 1020177016079 A KR1020177016079 A KR 1020177016079A KR 20177016079 A KR20177016079 A KR 20177016079A KR 102052983 B1 KR102052983 B1 KR 102052983B1
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KR20170071613A (ko
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크리스토퍼 제이. 소레스
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크리스토퍼 제이. 소레스
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/57527—Calcitonin gene related peptide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/225—Calcitonin gene related peptide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/23—Calcitonins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
    • A61P5/22—Drugs for disorders of the endocrine system of the parathyroid hormones for decreasing, blocking or antagonising the activity of calcitonin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/585—Calcitonins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
KR1020177016079A 2012-01-26 2013-01-25 펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도 Active KR102052983B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261591236P 2012-01-26 2012-01-26
US61/591,236 2012-01-26
PCT/US2013/023260 WO2013112912A1 (en) 2012-01-26 2013-01-25 Peptide antagonists of the calcitonin cgrp family of peptide hormones and their use

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020147023782A Division KR101855242B1 (ko) 2012-01-26 2013-01-25 펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도

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Publication Number Publication Date
KR20170071613A KR20170071613A (ko) 2017-06-23
KR102052983B1 true KR102052983B1 (ko) 2019-12-06

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KR1020177016079A Active KR102052983B1 (ko) 2012-01-26 2013-01-25 펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도
KR1020147023782A Active KR101855242B1 (ko) 2012-01-26 2013-01-25 펩타이드 호르몬의 칼시토닌 cgrp 패밀리의 펩타이드 길항제 및 그의 용도

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US (3) US9193776B2 (enExample)
EP (2) EP3272769B1 (enExample)
JP (3) JP6025871B2 (enExample)
KR (2) KR102052983B1 (enExample)
CN (2) CN108997490A (enExample)
AU (2) AU2013211929B2 (enExample)
CA (1) CA2861392C (enExample)
DK (1) DK2807187T3 (enExample)
ES (2) ES2819825T3 (enExample)
IL (2) IL233655A (enExample)
MX (1) MX347229B (enExample)
NO (1) NO2864579T3 (enExample)
RU (2) RU2624016C2 (enExample)
WO (1) WO2013112912A1 (enExample)

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AU2013211929B2 (en) * 2012-01-26 2016-05-26 Christopher J. Soares Peptide antagonists of the calcitonin CGRP family of peptide hormones and their use
WO2015017455A1 (en) * 2013-07-30 2015-02-05 Soares Christopher J Cgrp agonist peptides
JO3669B1 (ar) * 2015-01-06 2020-08-27 Ferring Bv بيبتيدات مضَادَّة لببتيد المرتبط بجين الكالسيتونين
CN109311959A (zh) * 2016-01-04 2019-02-05 艾得佩索拉公司 肽类似物
CA3035561A1 (en) 2016-09-02 2018-03-08 Christopher J. Soares Use of cgrp receptor antagonists in neuroprotection and neurological disorders
CA2967616A1 (en) * 2016-09-19 2018-03-19 The Governors Of The University Of Alberta Brain penetrant amylin receptor based peptides for alzheimer's disease
JP2021501784A (ja) * 2017-11-06 2021-01-21 オークランド ユニサービシーズ リミティド ペプチド複合体ｃｇｒｐ受容体アンタゴニストおよびその調製方法および使用方法
JP7214100B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
JP7214104B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
JP7214102B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
CN116456981A (zh) * 2020-11-19 2023-07-18 辉瑞爱尔兰制药公司 用于改善的grp抑制剂递送的组合物

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Also Published As

Publication number Publication date
RU2624016C2 (ru) 2017-06-30
CN108997490A (zh) 2018-12-14
HK1249915A1 (en) 2018-11-16
MX2014008960A (es) 2015-01-16
AU2016205801A1 (en) 2016-08-04
KR20170071613A (ko) 2017-06-23
WO2013112912A1 (en) 2013-08-01
AU2013211929A1 (en) 2014-09-11
ES2641325T3 (es) 2017-11-08
EP3272769A1 (en) 2018-01-24
US20140329752A1 (en) 2014-11-06
JP2017036308A (ja) 2017-02-16
JP6025871B2 (ja) 2016-11-16
JP6411425B2 (ja) 2018-10-24
CN104271596B (zh) 2018-09-18
CA2861392C (en) 2021-08-17
US9193776B2 (en) 2015-11-24
ES2819825T3 (es) 2021-04-19
US20170204155A1 (en) 2017-07-20
KR101855242B1 (ko) 2018-05-09
US20160145315A1 (en) 2016-05-26
EP2807187A1 (en) 2014-12-03
RU2742826C2 (ru) 2021-02-11
BR112014018284A2 (pt) 2017-07-04
NO2864579T3 (enExample) 2018-01-20
US10370425B2 (en) 2019-08-06
MX347229B (es) 2017-04-19
IL252555B (en) 2020-06-30
AU2013211929B2 (en) 2016-05-26
JP2019006821A (ja) 2019-01-17
RU2014131605A (ru) 2016-03-20
KR20140132342A (ko) 2014-11-17
IL233655A0 (en) 2014-08-31
RU2017119773A3 (enExample) 2020-11-18
EP3272769B1 (en) 2020-06-17
CA2861392A1 (en) 2013-08-01
HK1201068A1 (en) 2015-08-21
RU2017119773A (ru) 2018-12-06
JP2015513318A (ja) 2015-05-07
IL252555A0 (en) 2017-07-31
EP2807187B1 (en) 2017-07-26
DK2807187T3 (en) 2017-09-11
CN104271596A (zh) 2015-01-07
IL233655A (en) 2017-06-29

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