KR101567969B1 - 벤질페닐 시클로헥산 유도체 및 이의 사용 방법 - Google Patents

벤질페닐 시클로헥산 유도체 및 이의 사용 방법 Download PDF

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Publication number
KR101567969B1
KR101567969B1 KR1020107015420A KR20107015420A KR101567969B1 KR 101567969 B1 KR101567969 B1 KR 101567969B1 KR 1020107015420 A KR1020107015420 A KR 1020107015420A KR 20107015420 A KR20107015420 A KR 20107015420A KR 101567969 B1 KR101567969 B1 KR 101567969B1
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South Korea
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phenyl
diabetes
chloro
rti
compound
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Expired - Fee Related
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English (en)
Korean (ko)
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KR20100098690A (ko
Inventor
위안웨이 첸
쿤 펭
릴리 장
빈후아 엘브이
바이후아 쉬
지아지아 동
지얀 두
얀 펭
게 수
바산타쿠말 라자판
브라이언 시드
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테라코스, 인코포레이티드
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Publication of KR20100098690A publication Critical patent/KR20100098690A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
KR1020107015420A 2007-12-13 2008-12-11 벤질페닐 시클로헥산 유도체 및 이의 사용 방법 Expired - Fee Related KR101567969B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1351707P 2007-12-13 2007-12-13
US61/013,517 2007-12-13

Publications (2)

Publication Number Publication Date
KR20100098690A KR20100098690A (ko) 2010-09-08
KR101567969B1 true KR101567969B1 (ko) 2015-11-10

Family

ID=40754059

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020107015420A Expired - Fee Related KR101567969B1 (ko) 2007-12-13 2008-12-11 벤질페닐 시클로헥산 유도체 및 이의 사용 방법

Country Status (16)

Country Link
US (1) US8129434B2 (enExample)
EP (1) EP2230907B1 (enExample)
JP (1) JP5507464B2 (enExample)
KR (1) KR101567969B1 (enExample)
CN (1) CN101938902B (enExample)
AR (2) AR071268A1 (enExample)
AU (1) AU2008335080B2 (enExample)
BR (1) BRPI0819930A2 (enExample)
CA (1) CA2707909C (enExample)
IL (1) IL206234A0 (enExample)
NZ (1) NZ586639A (enExample)
RU (1) RU2505521C2 (enExample)
TW (1) TWI426081B (enExample)
UA (1) UA101004C2 (enExample)
WO (1) WO2009076550A1 (enExample)
ZA (1) ZA201004400B (enExample)

Families Citing this family (14)

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CN102149280B (zh) * 2008-07-15 2017-05-24 泰拉科斯有限公司 氘化苄基苯衍生物及其使用方法
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
BR112013030163A2 (pt) * 2011-05-26 2017-03-01 Tfchem composto, uso cosmético de pelo menos um composto, composição farmacêutica ou cosmética e processo para preparar um composto.
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN103570671B (zh) * 2012-09-26 2016-03-30 上海天慈生物谷生物工程有限公司 一种降糖化合物及其制法和应用
WO2015051484A1 (en) 2013-10-12 2015-04-16 Theracos, Inc. Preparation of hydroxy-benzylbenzene derivatives
CN105828815B (zh) 2013-12-17 2020-03-27 勃林格殷格翰动物保健有限公司 猫科动物中代谢紊乱的治疗
US10759729B2 (en) * 2016-11-07 2020-09-01 The Chinese University Of Hong Kong Compounds for treating diabetes
CN116785268A (zh) * 2022-03-14 2023-09-22 江苏万邦生化医药集团有限责任公司 一种sglt-2抑制剂的药物组合物

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Also Published As

Publication number Publication date
JP5507464B2 (ja) 2014-05-28
JP2011506469A (ja) 2011-03-03
NZ586639A (en) 2011-06-30
TW200932755A (en) 2009-08-01
EP2230907A4 (en) 2015-04-08
TWI426081B (zh) 2014-02-11
CA2707909A1 (en) 2009-06-18
CN101938902B (zh) 2014-07-02
AR071268A1 (es) 2010-06-09
AU2008335080B2 (en) 2014-06-05
IL206234A0 (en) 2010-12-30
WO2009076550A1 (en) 2009-06-18
RU2505521C2 (ru) 2014-01-27
CA2707909C (en) 2016-10-18
UA101004C2 (en) 2013-02-25
ZA201004400B (en) 2014-10-29
US20090156516A1 (en) 2009-06-18
AU2008335080A1 (en) 2009-06-18
US8129434B2 (en) 2012-03-06
AR113211A2 (es) 2020-02-19
RU2010128940A (ru) 2012-01-20
BRPI0819930A2 (pt) 2016-05-17
CN101938902A (zh) 2011-01-05
KR20100098690A (ko) 2010-09-08
EP2230907A1 (en) 2010-09-29
EP2230907B1 (en) 2018-05-09

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