AR071268A1 - Derivados de bencilfenilciclohexano, metodos de uso y una composicion farmaceutica - Google Patents

Derivados de bencilfenilciclohexano, metodos de uso y una composicion farmaceutica

Info

Publication number
AR071268A1
AR071268A1 ARP080105417A ARP080105417A AR071268A1 AR 071268 A1 AR071268 A1 AR 071268A1 AR P080105417 A ARP080105417 A AR P080105417A AR P080105417 A ARP080105417 A AR P080105417A AR 071268 A1 AR071268 A1 AR 071268A1
Authority
AR
Argentina
Prior art keywords
alkyl
cycloalkyl
optionally
alkyloxy
cycloalkenyl
Prior art date
Application number
ARP080105417A
Other languages
English (en)
Spanish (es)
Original Assignee
Theracos Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theracos Inc filed Critical Theracos Inc
Publication of AR071268A1 publication Critical patent/AR071268A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
ARP080105417A 2007-12-13 2008-12-12 Derivados de bencilfenilciclohexano, metodos de uso y una composicion farmaceutica AR071268A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1351707P 2007-12-13 2007-12-13

Publications (1)

Publication Number Publication Date
AR071268A1 true AR071268A1 (es) 2010-06-09

Family

ID=40754059

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP080105417A AR071268A1 (es) 2007-12-13 2008-12-12 Derivados de bencilfenilciclohexano, metodos de uso y una composicion farmaceutica
ARP180100403A AR113211A2 (es) 2007-12-13 2018-02-21 Derivados de bencilfenilciclohexano y métodos de uso

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP180100403A AR113211A2 (es) 2007-12-13 2018-02-21 Derivados de bencilfenilciclohexano y métodos de uso

Country Status (16)

Country Link
US (1) US8129434B2 (enExample)
EP (1) EP2230907B1 (enExample)
JP (1) JP5507464B2 (enExample)
KR (1) KR101567969B1 (enExample)
CN (1) CN101938902B (enExample)
AR (2) AR071268A1 (enExample)
AU (1) AU2008335080B2 (enExample)
BR (1) BRPI0819930A2 (enExample)
CA (1) CA2707909C (enExample)
IL (1) IL206234A0 (enExample)
NZ (1) NZ586639A (enExample)
RU (1) RU2505521C2 (enExample)
TW (1) TWI426081B (enExample)
UA (1) UA101004C2 (enExample)
WO (1) WO2009076550A1 (enExample)
ZA (1) ZA201004400B (enExample)

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US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
CN103649033B (zh) * 2011-05-26 2016-02-24 Tf化学公司 芳基、杂芳基、o-芳基和o-杂芳基碳环糖家族
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN103570671B (zh) * 2012-09-26 2016-03-30 上海天慈生物谷生物工程有限公司 一种降糖化合物及其制法和应用
WO2015051484A1 (en) 2013-10-12 2015-04-16 Theracos, Inc. Preparation of hydroxy-benzylbenzene derivatives
EP3082829B1 (en) 2013-12-17 2021-02-17 Boehringer Ingelheim Vetmedica GmbH Sglt2 inhibitors for the treatment of metabolic disorders in feline animals
US10759729B2 (en) * 2016-11-07 2020-09-01 The Chinese University Of Hong Kong Compounds for treating diabetes
CN116785268A (zh) * 2022-03-14 2023-09-22 江苏万邦生化医药集团有限责任公司 一种sglt-2抑制剂的药物组合物

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Also Published As

Publication number Publication date
ZA201004400B (en) 2014-10-29
JP2011506469A (ja) 2011-03-03
US8129434B2 (en) 2012-03-06
TW200932755A (en) 2009-08-01
CA2707909A1 (en) 2009-06-18
KR20100098690A (ko) 2010-09-08
CA2707909C (en) 2016-10-18
AU2008335080B2 (en) 2014-06-05
UA101004C2 (en) 2013-02-25
RU2505521C2 (ru) 2014-01-27
AU2008335080A1 (en) 2009-06-18
EP2230907B1 (en) 2018-05-09
JP5507464B2 (ja) 2014-05-28
NZ586639A (en) 2011-06-30
AR113211A2 (es) 2020-02-19
US20090156516A1 (en) 2009-06-18
CN101938902A (zh) 2011-01-05
RU2010128940A (ru) 2012-01-20
BRPI0819930A2 (pt) 2016-05-17
TWI426081B (zh) 2014-02-11
WO2009076550A1 (en) 2009-06-18
EP2230907A1 (en) 2010-09-29
CN101938902B (zh) 2014-07-02
KR101567969B1 (ko) 2015-11-10
IL206234A0 (en) 2010-12-30
EP2230907A4 (en) 2015-04-08

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