KR101396639B1 - 레보도파 프로드럭 메실레이트, 그것의 조성물 및 그것의용도 - Google Patents

레보도파 프로드럭 메실레이트, 그것의 조성물 및 그것의용도 Download PDF

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KR101396639B1
KR101396639B1 KR1020087016252A KR20087016252A KR101396639B1 KR 101396639 B1 KR101396639 B1 KR 101396639B1 KR 1020087016252 A KR1020087016252 A KR 1020087016252A KR 20087016252 A KR20087016252 A KR 20087016252A KR 101396639 B1 KR101396639 B1 KR 101396639B1
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amino
dihydroxyphenyl
phenylcarbonyloxypropyl
propanoate
propanoate mesylate
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KR20080073365A (ko
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자닝 샹
쉐동 다이
신디 엑스 저우
?화 리
마크 큐 구엔
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제노포트 인코포레이티드
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4458—Non condensed piperidines, e.g. piperocaine only substituted in position 2, e.g. methylphenidate
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/04—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing only one sulfo group
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    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
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KR1020087016252A 2005-12-05 2006-12-04 레보도파 프로드럭 메실레이트, 그것의 조성물 및 그것의용도 Expired - Fee Related KR101396639B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74187605P 2005-12-05 2005-12-05
US60/741,876 2005-12-05
PCT/US2006/046273 WO2007067495A2 (en) 2005-12-05 2006-12-04 Levodopa prodrug mesylate, compositions thereof, and uses thereof

Publications (2)

Publication Number Publication Date
KR20080073365A KR20080073365A (ko) 2008-08-08
KR101396639B1 true KR101396639B1 (ko) 2014-05-21

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US (5) US7563821B2 (enExample)
EP (1) EP1959948B1 (enExample)
JP (1) JP5153641B2 (enExample)
KR (1) KR101396639B1 (enExample)
CN (1) CN101365439B (enExample)
AU (1) AU2006322051B2 (enExample)
BR (1) BRPI0619425A2 (enExample)
CA (1) CA2631643C (enExample)
CY (1) CY1113108T1 (enExample)
DK (1) DK1959948T3 (enExample)
ES (1) ES2391575T3 (enExample)
IL (1) IL191937A (enExample)
NO (1) NO20082768L (enExample)
NZ (1) NZ569485A (enExample)
PL (1) PL1959948T3 (enExample)
PT (1) PT1959948E (enExample)
RU (1) RU2429223C2 (enExample)
TW (1) TWI403493B (enExample)
WO (1) WO2007067495A2 (enExample)
ZA (1) ZA200805511B (enExample)

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