KR101300831B1 - 이미다조[1,2-a]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 - Google Patents

이미다조[1,2-a]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 Download PDF

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KR101300831B1
KR101300831B1 KR1020077023609A KR20077023609A KR101300831B1 KR 101300831 B1 KR101300831 B1 KR 101300831B1 KR 1020077023609 A KR1020077023609 A KR 1020077023609A KR 20077023609 A KR20077023609 A KR 20077023609A KR 101300831 B1 KR101300831 B1 KR 101300831B1
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pyridin
imidazo
hydroxy
delete delete
acrylamide
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KR20080005207A (ko
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켄 치 릭 리
에릭 티 선
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에스*바이오 피티이 리미티드
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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KR1020077023609A 2005-03-21 2006-03-20 이미다조[1,2-a]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 Expired - Fee Related KR101300831B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US66326505P 2005-03-21 2005-03-21
US60/663,265 2005-03-21
US75954406P 2006-01-18 2006-01-18
US60/759,544 2006-01-18
PCT/SG2006/000064 WO2006101455A1 (en) 2005-03-21 2006-03-20 Imidazo[1,2-a]pyridine derivatives: preparation and pharmaceutical applications

Publications (2)

Publication Number Publication Date
KR20080005207A KR20080005207A (ko) 2008-01-10
KR101300831B1 true KR101300831B1 (ko) 2013-08-30

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Country Status (12)

Country Link
EP (1) EP1863811B1 (enExample)
JP (1) JP5206405B2 (enExample)
KR (1) KR101300831B1 (enExample)
CN (1) CN101218238B (enExample)
AR (1) AR056187A1 (enExample)
AU (1) AU2006225355B2 (enExample)
CA (1) CA2602328C (enExample)
ES (1) ES2470766T3 (enExample)
MX (1) MX2007011710A (enExample)
MY (1) MY147647A (enExample)
TW (1) TW200714600A (enExample)
WO (1) WO2006101455A1 (enExample)

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WO2008068392A1 (fr) * 2006-12-07 2008-06-12 Commissariat A L'energie Atomique Nouveaux derives fluorophores imidazo [1,2-a] pyridin-3-yl-amine et leur procede de preparation
EP2155744A1 (en) 2007-04-10 2010-02-24 Lundbeck, H., A/S Heteroaryl amide analogues as p2x7 antagonists
WO2008134553A1 (en) * 2007-04-26 2008-11-06 Xenon Pharmaceuticals Inc. Methods of using bicyclic compounds in treating sodium channel-mediated diseases
CN101855222A (zh) * 2007-05-10 2010-10-06 通用电气健康护理有限公司 对大麻素cb2受体具有活性的咪唑并(1,2-a)吡啶和相关化合物
EP2180893B1 (en) * 2007-08-09 2014-11-12 Urifer Ltd Pharmaceutical compositions and methods for the treatment of cancer
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JP2011502133A (ja) * 2007-11-02 2011-01-20 メシルジーン インコーポレイテッド ヒストンデアセチラーゼの阻害剤
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WO2010032195A1 (en) 2008-09-16 2010-03-25 Csir Imidazopyridines and imidazopyrimidines as hiv-i reverse transcriptase inhibitors
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AU2011285708B2 (en) * 2010-08-03 2014-07-24 The Regents Of The University Of California Compounds and compositions for mitigating tissue damage and lethality
US9000186B2 (en) 2011-02-01 2015-04-07 Kyowa Hakko Kirin Co., Ltd. Ring-fused heterocyclic derivative
US20140221354A1 (en) * 2011-03-31 2014-08-07 Emblem Technology Transfer Gmbh IMIDAZO [1,2-a]PYRIDINE COMPOUNDS FOR USE IN THERAPY
UY34305A (es) 2011-09-01 2013-04-30 Novartis Ag Derivados de heterociclos bicíclicos para el tratamiento de la hipertensión arterial pulmonar
CN104619707A (zh) * 2012-07-31 2015-05-13 协和发酵麒麟株式会社 稠环杂环化合物
US9073921B2 (en) 2013-03-01 2015-07-07 Novartis Ag Salt forms of bicyclic heterocyclic derivatives
SI2991984T1 (sl) * 2013-04-30 2017-05-31 F. Hoffmann-La Roche Ag Povezovanje pirazolovih amidov, katalizirano s paladijem
SG11201509650YA (en) * 2013-05-24 2015-12-30 Iomet Pharma Ltd Slc2a transporter inhibitors
CN105358151B (zh) 2013-06-25 2019-04-12 豪夫迈·罗氏有限公司 用于治疗脊髓性肌萎缩的化合物
WO2015058106A1 (en) 2013-10-18 2015-04-23 The General Hospital Corporation Imaging histone deacetylases with a radiotracer using positron emission tomography
US10723705B2 (en) 2015-08-14 2020-07-28 Incyte Corporation Heterocyclic compounds and uses thereof
WO2018048261A1 (ko) * 2016-09-08 2018-03-15 가천대학교 산학협력단 신규 스피로퀴논 유도체 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 신경계 질환의 예방 또는 치료용 약학적 조성물
EP4019607B1 (en) 2020-12-22 2024-05-15 Essilor International Electrochromic compounds and optical articles containing them
CN113321651B (zh) * 2021-06-22 2022-06-14 四川省医学科学院·四川省人民医院 吡唑并吡啶异羟肟酸类化合物、其制备方法及其应用

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US20050005471A1 (en) 2003-07-10 2005-01-13 Kung-Sheng Pan Flocked footwear

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EP1863811A4 (en) 2008-11-12
CN101218238B (zh) 2011-10-26
CA2602328A1 (en) 2006-09-28
EP1863811B1 (en) 2014-03-12
CA2602328C (en) 2014-07-29
EP1863811A1 (en) 2007-12-12
JP5206405B2 (ja) 2013-06-12
MY147647A (en) 2012-12-31
MX2007011710A (es) 2007-11-20
JP2008533198A (ja) 2008-08-21
ES2470766T3 (es) 2014-06-24
AU2006225355B2 (en) 2010-12-09
CN101218238A (zh) 2008-07-09
AU2006225355A1 (en) 2006-09-28
WO2006101455A1 (en) 2006-09-28
AR056187A1 (es) 2007-09-26
KR20080005207A (ko) 2008-01-10
TW200714600A (en) 2007-04-16

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