AU2006225355B2 - Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications - Google Patents
Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications Download PDFInfo
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- AU2006225355B2 AU2006225355B2 AU2006225355A AU2006225355A AU2006225355B2 AU 2006225355 B2 AU2006225355 B2 AU 2006225355B2 AU 2006225355 A AU2006225355 A AU 2006225355A AU 2006225355 A AU2006225355 A AU 2006225355A AU 2006225355 B2 AU2006225355 B2 AU 2006225355B2
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- hydroxy
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- acrylamide
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- 150000005234 imidazo[1,2-a]pyridines Chemical class 0.000 title description 2
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Landscapes
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Applications Claiming Priority (5)
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| US66326505P | 2005-03-21 | 2005-03-21 | |
| US60/663,265 | 2005-03-21 | ||
| US75954406P | 2006-01-18 | 2006-01-18 | |
| US60/759,544 | 2006-01-18 | ||
| PCT/SG2006/000064 WO2006101455A1 (en) | 2005-03-21 | 2006-03-20 | Imidazo[1,2-a]pyridine derivatives: preparation and pharmaceutical applications |
Publications (2)
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| AU2006225355A1 AU2006225355A1 (en) | 2006-09-28 |
| AU2006225355B2 true AU2006225355B2 (en) | 2010-12-09 |
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| AU2006225355A Ceased AU2006225355B2 (en) | 2005-03-21 | 2006-03-20 | Imidazo(1,2-a)pyridine derivatives: preparation and pharmaceutical applications |
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| JP (1) | JP5206405B2 (enExample) |
| KR (1) | KR101300831B1 (enExample) |
| CN (1) | CN101218238B (enExample) |
| AR (1) | AR056187A1 (enExample) |
| AU (1) | AU2006225355B2 (enExample) |
| CA (1) | CA2602328C (enExample) |
| ES (1) | ES2470766T3 (enExample) |
| MX (1) | MX2007011710A (enExample) |
| MY (1) | MY147647A (enExample) |
| TW (1) | TW200714600A (enExample) |
| WO (1) | WO2006101455A1 (enExample) |
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| US20080004311A1 (en) * | 2002-11-12 | 2008-01-03 | Alcon, Inc. | Histone deacetylase inhibitors for treating degenerative diseases of the eye |
| US7666880B2 (en) | 2005-03-21 | 2010-02-23 | S*Bio Pte Ltd. | Imidazo[1,2-A]pyridine derivatives: preparation and pharmaceutical applications |
| WO2008029152A2 (en) * | 2006-09-08 | 2008-03-13 | Summit Corporation Plc | Treatment of duchenne muscular dystrophy |
| EP2064211B1 (en) * | 2006-09-20 | 2015-11-11 | MEI Pharma, Inc. | Imidazo[1,2-a]pyridine hydroxymate compounds that are inhibitors of histone deacetylase |
| EA201300152A1 (ru) | 2006-11-27 | 2013-07-30 | Х. Лундбекк А/С | Гетероариламидные производные |
| WO2008068392A1 (fr) * | 2006-12-07 | 2008-06-12 | Commissariat A L'energie Atomique | Nouveaux derives fluorophores imidazo [1,2-a] pyridin-3-yl-amine et leur procede de preparation |
| EP2155744A1 (en) | 2007-04-10 | 2010-02-24 | Lundbeck, H., A/S | Heteroaryl amide analogues as p2x7 antagonists |
| WO2008134553A1 (en) * | 2007-04-26 | 2008-11-06 | Xenon Pharmaceuticals Inc. | Methods of using bicyclic compounds in treating sodium channel-mediated diseases |
| CN101855222A (zh) * | 2007-05-10 | 2010-10-06 | 通用电气健康护理有限公司 | 对大麻素cb2受体具有活性的咪唑并(1,2-a)吡啶和相关化合物 |
| EP2180893B1 (en) * | 2007-08-09 | 2014-11-12 | Urifer Ltd | Pharmaceutical compositions and methods for the treatment of cancer |
| DE102007040336A1 (de) | 2007-08-27 | 2009-03-05 | Johann Wolfgang Goethe-Universität Frankfurt am Main | Neue Inhibitoren der 5-Lipoxygenase und deren Verwendungen |
| JP2011502133A (ja) * | 2007-11-02 | 2011-01-20 | メシルジーン インコーポレイテッド | ヒストンデアセチラーゼの阻害剤 |
| WO2009143156A2 (en) * | 2008-05-19 | 2009-11-26 | Sepracor Inc. | IMIDAZO[1,2-a]PYRIDINE COMPOUNDS |
| WO2010032195A1 (en) | 2008-09-16 | 2010-03-25 | Csir | Imidazopyridines and imidazopyrimidines as hiv-i reverse transcriptase inhibitors |
| WO2010043953A2 (en) * | 2008-10-15 | 2010-04-22 | Orchid Research Laboratories Ltd. | Novel bridged cyclic compounds as histone deacetylase inhibitors |
| AU2011285708B2 (en) * | 2010-08-03 | 2014-07-24 | The Regents Of The University Of California | Compounds and compositions for mitigating tissue damage and lethality |
| US9000186B2 (en) | 2011-02-01 | 2015-04-07 | Kyowa Hakko Kirin Co., Ltd. | Ring-fused heterocyclic derivative |
| US20140221354A1 (en) * | 2011-03-31 | 2014-08-07 | Emblem Technology Transfer Gmbh | IMIDAZO [1,2-a]PYRIDINE COMPOUNDS FOR USE IN THERAPY |
| UY34305A (es) | 2011-09-01 | 2013-04-30 | Novartis Ag | Derivados de heterociclos bicíclicos para el tratamiento de la hipertensión arterial pulmonar |
| CN104619707A (zh) * | 2012-07-31 | 2015-05-13 | 协和发酵麒麟株式会社 | 稠环杂环化合物 |
| US9073921B2 (en) | 2013-03-01 | 2015-07-07 | Novartis Ag | Salt forms of bicyclic heterocyclic derivatives |
| SI2991984T1 (sl) * | 2013-04-30 | 2017-05-31 | F. Hoffmann-La Roche Ag | Povezovanje pirazolovih amidov, katalizirano s paladijem |
| SG11201509650YA (en) * | 2013-05-24 | 2015-12-30 | Iomet Pharma Ltd | Slc2a transporter inhibitors |
| CN105358151B (zh) | 2013-06-25 | 2019-04-12 | 豪夫迈·罗氏有限公司 | 用于治疗脊髓性肌萎缩的化合物 |
| WO2015058106A1 (en) | 2013-10-18 | 2015-04-23 | The General Hospital Corporation | Imaging histone deacetylases with a radiotracer using positron emission tomography |
| US10723705B2 (en) | 2015-08-14 | 2020-07-28 | Incyte Corporation | Heterocyclic compounds and uses thereof |
| WO2018048261A1 (ko) * | 2016-09-08 | 2018-03-15 | 가천대학교 산학협력단 | 신규 스피로퀴논 유도체 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 신경계 질환의 예방 또는 치료용 약학적 조성물 |
| EP4019607B1 (en) | 2020-12-22 | 2024-05-15 | Essilor International | Electrochromic compounds and optical articles containing them |
| CN113321651B (zh) * | 2021-06-22 | 2022-06-14 | 四川省医学科学院·四川省人民医院 | 吡唑并吡啶异羟肟酸类化合物、其制备方法及其应用 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0266890A1 (en) | 1986-10-07 | 1988-05-11 | Yamanouchi Pharmaceutical Co. Ltd. | Imidazopyridine derivatives, their production, and pharmaceutical compositions containing them |
| JPH11505524A (ja) * | 1995-05-01 | 1999-05-21 | 藤沢薬品工業株式会社 | イミダゾ１，２−ａピリジンおよびイミダゾ１，２−ａピリデジン誘導体、および骨吸収阻害剤としてのその用途 |
| SE9801526D0 (sv) * | 1998-04-29 | 1998-04-29 | Astra Ab | New compounds |
| JP2002515433A (ja) * | 1998-05-20 | 2002-05-28 | イーライ・リリー・アンド・カンパニー | 抗ウイルス化合物 |
| UA80296C2 (en) * | 2002-09-06 | 2007-09-10 | Biogen Inc | Imidazolopyridines and methods of making and using the same |
| US7381825B2 (en) * | 2003-03-17 | 2008-06-03 | Takeda San Diego, Inc. | Histone deacetylase inhibitors |
| TW200501897A (en) | 2003-07-10 | 2005-01-16 | Kung-Sheng Pan | Shoes electrostatically embedded with objects |
| US7144907B2 (en) * | 2003-09-03 | 2006-12-05 | Array Biopharma Inc. | Heterocyclic inhibitors of MEK and methods of use thereof |
| US7538120B2 (en) * | 2003-09-03 | 2009-05-26 | Array Biopharma Inc. | Method of treating inflammatory diseases |
| CN1934094A (zh) * | 2004-03-05 | 2007-03-21 | 万有制药株式会社 | 二芳基取代杂环5元环衍生物 |
| EP1735318A2 (en) * | 2004-03-17 | 2006-12-27 | Altana Pharma AG | 7h-8,9-dihydro-pyrano(2,3-c)imidazo(1,2a)pyridine derivatives and their use as gastric acid secretion inhibitors |
-
2006
- 2006-03-20 AU AU2006225355A patent/AU2006225355B2/en not_active Ceased
- 2006-03-20 TW TW095109517A patent/TW200714600A/zh unknown
- 2006-03-20 MX MX2007011710A patent/MX2007011710A/es active IP Right Grant
- 2006-03-20 CN CN2006800092539A patent/CN101218238B/zh not_active Expired - Fee Related
- 2006-03-20 KR KR1020077023609A patent/KR101300831B1/ko not_active Expired - Fee Related
- 2006-03-20 ES ES06717188.4T patent/ES2470766T3/es active Active
- 2006-03-20 MY MYPI20061225A patent/MY147647A/en unknown
- 2006-03-20 CA CA2602328A patent/CA2602328C/en not_active Expired - Fee Related
- 2006-03-20 JP JP2008502953A patent/JP5206405B2/ja not_active Expired - Fee Related
- 2006-03-20 AR ARP060101088A patent/AR056187A1/es unknown
- 2006-03-20 EP EP06717188.4A patent/EP1863811B1/en not_active Not-in-force
- 2006-03-20 WO PCT/SG2006/000064 patent/WO2006101455A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP1863811A4 (en) | 2008-11-12 |
| CN101218238B (zh) | 2011-10-26 |
| CA2602328A1 (en) | 2006-09-28 |
| EP1863811B1 (en) | 2014-03-12 |
| CA2602328C (en) | 2014-07-29 |
| EP1863811A1 (en) | 2007-12-12 |
| JP5206405B2 (ja) | 2013-06-12 |
| MY147647A (en) | 2012-12-31 |
| MX2007011710A (es) | 2007-11-20 |
| JP2008533198A (ja) | 2008-08-21 |
| ES2470766T3 (es) | 2014-06-24 |
| KR101300831B1 (ko) | 2013-08-30 |
| CN101218238A (zh) | 2008-07-09 |
| AU2006225355A1 (en) | 2006-09-28 |
| WO2006101455A1 (en) | 2006-09-28 |
| AR056187A1 (es) | 2007-09-26 |
| KR20080005207A (ko) | 2008-01-10 |
| TW200714600A (en) | 2007-04-16 |
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| FGA | Letters patent sealed or granted (standard patent) | ||
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Owner name: HELSINN HEALTHCARE SA Free format text: FORMER OWNER(S): S*BIO PTE LTD |
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| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |