KR101245062B1 - 칼슘이온-방출-활성화-칼슘이온 채널을 조절하는 방법 - Google Patents
칼슘이온-방출-활성화-칼슘이온 채널을 조절하는 방법 Download PDFInfo
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- KR101245062B1 KR101245062B1 KR1020067001589A KR20067001589A KR101245062B1 KR 101245062 B1 KR101245062 B1 KR 101245062B1 KR 1020067001589 A KR1020067001589 A KR 1020067001589A KR 20067001589 A KR20067001589 A KR 20067001589A KR 101245062 B1 KR101245062 B1 KR 101245062B1
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- biphenyl
- trifluoromethyl
- carboxylic acid
- amide
- methyl
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- 0 Cc1cc(-c(cc2)ccc2NC(c2ccncc2*)=O)c(C)cc1 Chemical compound Cc1cc(-c(cc2)ccc2NC(c2ccncc2*)=O)c(C)cc1 0.000 description 3
- GFEIWXNLDKUWIK-UHFFFAOYSA-N COc(cc1-c(cc2)ccc2NC(c2ccncc2F)=O)ccc1OC Chemical compound COc(cc1-c(cc2)ccc2NC(c2ccncc2F)=O)ccc1OC GFEIWXNLDKUWIK-UHFFFAOYSA-N 0.000 description 1
- YAGRGSPLLIWGFE-UHFFFAOYSA-N COc1ccc[n]2c(-c(cc3)ccc3NC(c(c(F)ccc3)c3F)=O)c(C(F)(F)F)cc12 Chemical compound COc1ccc[n]2c(-c(cc3)ccc3NC(c(c(F)ccc3)c3F)=O)c(C(F)(F)F)cc12 YAGRGSPLLIWGFE-UHFFFAOYSA-N 0.000 description 1
- GWFQDZLHSGIQQR-UHFFFAOYSA-N C[n]1c(C(Nc(cc2)ccc2-c2cc(C(F)(F)F)ccc2C(F)(F)F)=O)cnc1 Chemical compound C[n]1c(C(Nc(cc2)ccc2-c2cc(C(F)(F)F)ccc2C(F)(F)F)=O)cnc1 GWFQDZLHSGIQQR-UHFFFAOYSA-N 0.000 description 1
- DIPKRDUMYXHGED-UHFFFAOYSA-N O=C(c(c(F)ccc1)c1F)Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F Chemical compound O=C(c(c(F)ccc1)c1F)Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F DIPKRDUMYXHGED-UHFFFAOYSA-N 0.000 description 1
- VRYAOEYBOOCTDR-UHFFFAOYSA-N O=C(c1c(C(F)(F)F)ccnc1)Nc(cc1)ccc1-c1c(C(F)(F)F)cccc1 Chemical compound O=C(c1c(C(F)(F)F)ccnc1)Nc(cc1)ccc1-c1c(C(F)(F)F)cccc1 VRYAOEYBOOCTDR-UHFFFAOYSA-N 0.000 description 1
- YIGKCCOEDOTGOC-UHFFFAOYSA-N O=C(c1ccncc1F)Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F Chemical compound O=C(c1ccncc1F)Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F YIGKCCOEDOTGOC-UHFFFAOYSA-N 0.000 description 1
- ITDRLFXSUNQUCT-UHFFFAOYSA-N Oc1ccccc1C(Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F)=O Chemical compound Oc1ccccc1C(Nc(cc1)ccc1-c1cc(C(F)(F)F)ccc1C(F)(F)F)=O ITDRLFXSUNQUCT-UHFFFAOYSA-N 0.000 description 1
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- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
-
- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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PCT/US2004/023797 WO2005009954A2 (en) | 2003-07-23 | 2004-07-22 | Method for modulating calcium ion-release-activated calcium ion channels |
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KR1020067001589A KR101245062B1 (ko) | 2003-07-23 | 2004-07-22 | 칼슘이온-방출-활성화-칼슘이온 채널을 조절하는 방법 |
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2004
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- 2004-07-22 NZ NZ545447A patent/NZ545447A/en not_active IP Right Cessation
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- 2006-10-27 HK HK06111889.5A patent/HK1089973A1/xx not_active IP Right Cessation
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