KR100940054B1 - 호르몬 효과를 갖는 17알파-히드록시-14베타-스테로이드 - Google Patents

호르몬 효과를 갖는 17알파-히드록시-14베타-스테로이드 Download PDF

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Publication number
KR100940054B1
KR100940054B1 KR1020047003609A KR20047003609A KR100940054B1 KR 100940054 B1 KR100940054 B1 KR 100940054B1 KR 1020047003609 A KR1020047003609 A KR 1020047003609A KR 20047003609 A KR20047003609 A KR 20047003609A KR 100940054 B1 KR100940054 B1 KR 100940054B1
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KR
South Korea
Prior art keywords
hydroxy
androgen
compound
compounds
product
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Expired - Fee Related
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KR1020047003609A
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English (en)
Korean (ko)
Other versions
KR20040039346A (ko
Inventor
반더루얍
레이젠디르크
드구이저마르셀에베르
Original Assignee
엔.브이.오가논
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0062—Estrane derivatives substituted in position 17 alfa not substituted in position 17 beta
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020047003609A 2001-09-12 2002-09-06 호르몬 효과를 갖는 17알파-히드록시-14베타-스테로이드 Expired - Fee Related KR100940054B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP01203455 2001-09-12
EP01203455.9 2001-09-12
PCT/EP2002/010041 WO2003022864A1 (en) 2001-09-12 2002-09-06 17alpha-hydroxy-14beta-steroids with hormonal effect

Publications (2)

Publication Number Publication Date
KR20040039346A KR20040039346A (ko) 2004-05-10
KR100940054B1 true KR100940054B1 (ko) 2010-02-04

Family

ID=8180920

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020047003609A Expired - Fee Related KR100940054B1 (ko) 2001-09-12 2002-09-06 호르몬 효과를 갖는 17알파-히드록시-14베타-스테로이드

Country Status (28)

Country Link
US (1) US7169769B2 (enExample)
EP (1) EP1427748B1 (enExample)
JP (1) JP4471653B2 (enExample)
KR (1) KR100940054B1 (enExample)
CN (1) CN1257913C (enExample)
AR (1) AR036462A1 (enExample)
AT (1) ATE395352T1 (enExample)
AU (1) AU2002339536B2 (enExample)
BR (1) BR0212409A (enExample)
CA (1) CA2505575C (enExample)
CY (1) CY1108152T1 (enExample)
DE (1) DE60226623D1 (enExample)
DK (1) DK1427748T3 (enExample)
EC (1) ECSP045012A (enExample)
ES (1) ES2305306T3 (enExample)
HR (1) HRP20040193A2 (enExample)
HU (1) HUP0402139A3 (enExample)
IL (2) IL160451A0 (enExample)
IS (1) IS2555B (enExample)
MX (1) MXPA04002418A (enExample)
NO (1) NO326624B1 (enExample)
NZ (1) NZ531487A (enExample)
PL (1) PL207493B1 (enExample)
PT (1) PT1427748E (enExample)
RU (1) RU2294332C2 (enExample)
TW (1) TWI221154B (enExample)
WO (1) WO2003022864A1 (enExample)
ZA (1) ZA200401992B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI221154B (en) 2001-09-12 2004-09-21 Akzo Nobel Nv 17alpha-hydroxy-14beta-steroids with hormonal effect

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000053619A1 (en) * 1999-03-08 2000-09-14 Akzo Nobel N.V. 14.beta., 17-alpha-hydroxymethylandrostane derivatives as androgens

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3338925A (en) * 1965-10-25 1967-08-29 Syntex Corp 17-substituted 14beta-estr-4-enes
AU4299301A (en) * 2000-02-29 2001-09-12 National University Of Singapore, The A method for modulating steroidogenic activity
US6391868B2 (en) * 2000-05-10 2002-05-21 Lpt Research, Inc. Use of 5-alpha-androst-1-en-3,17-dione to increase the level of the anabolic/androgenic hormone 17-beta-hydroxy-5-alpha-androst-1-en-3-one in humans
TWI221154B (en) 2001-09-12 2004-09-21 Akzo Nobel Nv 17alpha-hydroxy-14beta-steroids with hormonal effect

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000053619A1 (en) * 1999-03-08 2000-09-14 Akzo Nobel N.V. 14.beta., 17-alpha-hydroxymethylandrostane derivatives as androgens

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
Chem. Pharm. Bull., Vol.25(6), 1977, 1295-301
Pharmacol. Res., Vol.32(4), 1995, 217-21
Steroids. Vol.59(10), 1994, 568-71.

Also Published As

Publication number Publication date
RU2294332C2 (ru) 2007-02-27
WO2003022864A1 (en) 2003-03-20
ATE395352T1 (de) 2008-05-15
PL207493B1 (pl) 2010-12-31
CA2505575C (en) 2010-01-26
US20040259849A1 (en) 2004-12-23
ECSP045012A (es) 2004-09-27
AR036462A1 (es) 2004-09-08
NO326624B1 (no) 2009-01-19
AU2002339536B2 (en) 2008-04-24
CA2505575A1 (en) 2003-03-20
HUP0402139A2 (hu) 2005-02-28
CN1553917A (zh) 2004-12-08
IS7165A (is) 2004-02-26
HK1063637A1 (en) 2005-01-07
JP4471653B2 (ja) 2010-06-02
IS2555B (is) 2009-10-15
RU2004110934A (ru) 2005-08-20
PL368727A1 (en) 2005-04-04
CN1257913C (zh) 2006-05-31
JP2005505566A (ja) 2005-02-24
MXPA04002418A (es) 2004-07-30
ZA200401992B (en) 2005-04-21
NZ531487A (en) 2005-08-26
NO20041010L (no) 2004-03-10
EP1427748B1 (en) 2008-05-14
BR0212409A (pt) 2004-08-03
IL160451A0 (en) 2004-07-25
DK1427748T3 (da) 2008-09-08
KR20040039346A (ko) 2004-05-10
ES2305306T3 (es) 2008-11-01
EP1427748A1 (en) 2004-06-16
HUP0402139A3 (en) 2012-12-28
HRP20040193A2 (en) 2004-08-31
DE60226623D1 (de) 2008-06-26
PT1427748E (pt) 2008-08-27
IL160451A (en) 2009-11-18
US7169769B2 (en) 2007-01-30
CY1108152T1 (el) 2014-02-12
TWI221154B (en) 2004-09-21

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