KR100522239B1 - 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 - Google Patents

아세트아미노펜을 함유하는 제어방출성의 경구용 제제 Download PDF

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Publication number
KR100522239B1
KR100522239B1 KR10-2002-0041469A KR20020041469A KR100522239B1 KR 100522239 B1 KR100522239 B1 KR 100522239B1 KR 20020041469 A KR20020041469 A KR 20020041469A KR 100522239 B1 KR100522239 B1 KR 100522239B1
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KR
South Korea
Prior art keywords
acetaminophen
weight
water
drug
parts
Prior art date
Application number
KR10-2002-0041469A
Other languages
English (en)
Korean (ko)
Other versions
KR20040006887A (ko
Inventor
이범진
조청일
최연웅
Original Assignee
주식회사 서울제약
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 주식회사 서울제약 filed Critical 주식회사 서울제약
Priority to KR10-2002-0041469A priority Critical patent/KR100522239B1/ko
Priority to AU2003232652A priority patent/AU2003232652A1/en
Priority to PCT/KR2003/001036 priority patent/WO2004006904A1/fr
Publication of KR20040006887A publication Critical patent/KR20040006887A/ko
Application granted granted Critical
Publication of KR100522239B1 publication Critical patent/KR100522239B1/ko

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
KR10-2002-0041469A 2002-07-16 2002-07-16 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 KR100522239B1 (ko)

Priority Applications (3)

Application Number Priority Date Filing Date Title
KR10-2002-0041469A KR100522239B1 (ko) 2002-07-16 2002-07-16 아세트아미노펜을 함유하는 제어방출성의 경구용 제제
AU2003232652A AU2003232652A1 (en) 2002-07-16 2003-05-27 Oral controlled-release dosage forms containing acetaminophen
PCT/KR2003/001036 WO2004006904A1 (fr) 2002-07-16 2003-05-27 Formes posologiques a liberation controlee administrees par voie orale contenant de l'acetaminophene

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR10-2002-0041469A KR100522239B1 (ko) 2002-07-16 2002-07-16 아세트아미노펜을 함유하는 제어방출성의 경구용 제제

Publications (2)

Publication Number Publication Date
KR20040006887A KR20040006887A (ko) 2004-01-24
KR100522239B1 true KR100522239B1 (ko) 2005-10-18

Family

ID=30113186

Family Applications (1)

Application Number Title Priority Date Filing Date
KR10-2002-0041469A KR100522239B1 (ko) 2002-07-16 2002-07-16 아세트아미노펜을 함유하는 제어방출성의 경구용 제제

Country Status (3)

Country Link
KR (1) KR100522239B1 (fr)
AU (1) AU2003232652A1 (fr)
WO (1) WO2004006904A1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100676298B1 (ko) * 2005-08-24 2007-01-30 씨제이 주식회사 고체분산체 및 그 제조방법
KR100704008B1 (ko) * 2005-11-23 2007-04-04 파미래 주식회사 실니디핀을 함유하는 경구용 제제 및 그의 제조방법
EP1935411A1 (fr) 2006-12-15 2008-06-25 Campina Nederland Holding B.V. Excipient à libération prolongée et son utilisation
KR100944121B1 (ko) * 2007-09-28 2010-02-24 대원제약주식회사 콩 다당체를 포함하는 속효성이 향상된 약제학적 조성물
JP5453280B2 (ja) 2007-10-16 2014-03-26 ラボファーム インコーポレイテッド アセトアミノフェンおよびトラマドールを持続的に放出するための二層組成物
BRPI0821732A2 (pt) 2007-12-17 2015-06-16 Labopharm Inc Formulações de liberação controlada , forma de dosagem sólida, e, uso da formulação de liberação controlada
JP2011511782A (ja) 2008-02-12 2011-04-14 アボット・ラボラトリーズ 長期放出性ヒドロコドンアセトアミノフェンならびにその関連方法および用途
EP2367541B1 (fr) 2008-12-16 2014-07-16 Paladin Labs Inc. Composition à libération contrôlée prévenant un mésusage
CZ302789B6 (cs) * 2009-11-25 2011-11-09 Zentiva, K. S. Zpusob zvýšení rozpustnosti farmaceuticky aktivních látek a cílený (kontrolovaný) transport do streva
KR20180025993A (ko) * 2012-01-04 2018-03-09 웰즐리 파마슈티컬스 엘엘씨 배뇨 빈도를 감소시키기 위한 연장-방출형 제제 및 이의 사용 방법
KR102237799B1 (ko) 2012-11-14 2021-04-08 더블유.알. 그레이스 앤드 캄파니-콘. 생물학적 활성 물질 및 비-정렬된 무기 산화물을 함유하는 조성물
PL3069733T3 (pl) * 2013-11-13 2023-02-13 National Defense Education And Research Foundation Nowa kompozycja związku stanowiącego acetaminofen niepowodująca w wątrobie działań niepożądanych
WO2016042570A1 (fr) * 2014-09-16 2016-03-24 Suresh Pareek Formulation à libération prolongée d'acétaminophène
JP7458317B2 (ja) * 2017-10-31 2024-03-29 サムヤン、ホールディングス、コーポレーション 崩壊が改善された経口用固形製剤組成物及びその製造方法
JP6858729B2 (ja) * 2018-05-25 2021-04-14 ▲財▼▲団▼法人国防教育研究基金会National Defense Education And Research Foundation 肝臓に対する副作用がない、新しいアセトアミノフェン複合組成
KR102168395B1 (ko) * 2018-10-30 2020-10-22 한양대학교 에리카산학협력단 용해도가 개선된 실데나필 유리염기 고체분산체 및 이의 제조방법

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820522A (en) * 1987-07-27 1989-04-11 Mcneilab, Inc. Oral sustained release acetaminophen formulation and process
US6149953A (en) * 1993-11-08 2000-11-21 Delta Food Group, Inc. Seeded microcapsules
US5948438A (en) * 1995-01-09 1999-09-07 Edward Mendell Co., Inc. Pharmaceutical formulations having improved disintegration and/or absorptivity
US5733578A (en) * 1995-11-15 1998-03-31 Edward Mendell Co., Inc. Directly compressible high load acetaminophen formulations
US6254891B1 (en) * 1998-09-03 2001-07-03 Ascent Pediatrics, Inc. Extended release acetaminophen

Also Published As

Publication number Publication date
KR20040006887A (ko) 2004-01-24
AU2003232652A1 (en) 2004-02-02
WO2004006904A1 (fr) 2004-01-22

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