KR100522239B1 - 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 - Google Patents
아세트아미노펜을 함유하는 제어방출성의 경구용 제제 Download PDFInfo
- Publication number
- KR100522239B1 KR100522239B1 KR10-2002-0041469A KR20020041469A KR100522239B1 KR 100522239 B1 KR100522239 B1 KR 100522239B1 KR 20020041469 A KR20020041469 A KR 20020041469A KR 100522239 B1 KR100522239 B1 KR 100522239B1
- Authority
- KR
- South Korea
- Prior art keywords
- acetaminophen
- weight
- water
- drug
- parts
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR10-2002-0041469A KR100522239B1 (ko) | 2002-07-16 | 2002-07-16 | 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 |
AU2003232652A AU2003232652A1 (en) | 2002-07-16 | 2003-05-27 | Oral controlled-release dosage forms containing acetaminophen |
PCT/KR2003/001036 WO2004006904A1 (fr) | 2002-07-16 | 2003-05-27 | Formes posologiques a liberation controlee administrees par voie orale contenant de l'acetaminophene |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR10-2002-0041469A KR100522239B1 (ko) | 2002-07-16 | 2002-07-16 | 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR20040006887A KR20040006887A (ko) | 2004-01-24 |
KR100522239B1 true KR100522239B1 (ko) | 2005-10-18 |
Family
ID=30113186
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR10-2002-0041469A KR100522239B1 (ko) | 2002-07-16 | 2002-07-16 | 아세트아미노펜을 함유하는 제어방출성의 경구용 제제 |
Country Status (3)
Country | Link |
---|---|
KR (1) | KR100522239B1 (fr) |
AU (1) | AU2003232652A1 (fr) |
WO (1) | WO2004006904A1 (fr) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100676298B1 (ko) * | 2005-08-24 | 2007-01-30 | 씨제이 주식회사 | 고체분산체 및 그 제조방법 |
KR100704008B1 (ko) * | 2005-11-23 | 2007-04-04 | 파미래 주식회사 | 실니디핀을 함유하는 경구용 제제 및 그의 제조방법 |
EP1935411A1 (fr) | 2006-12-15 | 2008-06-25 | Campina Nederland Holding B.V. | Excipient à libération prolongée et son utilisation |
KR100944121B1 (ko) * | 2007-09-28 | 2010-02-24 | 대원제약주식회사 | 콩 다당체를 포함하는 속효성이 향상된 약제학적 조성물 |
JP5453280B2 (ja) | 2007-10-16 | 2014-03-26 | ラボファーム インコーポレイテッド | アセトアミノフェンおよびトラマドールを持続的に放出するための二層組成物 |
BRPI0821732A2 (pt) | 2007-12-17 | 2015-06-16 | Labopharm Inc | Formulações de liberação controlada , forma de dosagem sólida, e, uso da formulação de liberação controlada |
JP2011511782A (ja) | 2008-02-12 | 2011-04-14 | アボット・ラボラトリーズ | 長期放出性ヒドロコドンアセトアミノフェンならびにその関連方法および用途 |
EP2367541B1 (fr) | 2008-12-16 | 2014-07-16 | Paladin Labs Inc. | Composition à libération contrôlée prévenant un mésusage |
CZ302789B6 (cs) * | 2009-11-25 | 2011-11-09 | Zentiva, K. S. | Zpusob zvýšení rozpustnosti farmaceuticky aktivních látek a cílený (kontrolovaný) transport do streva |
KR20180025993A (ko) * | 2012-01-04 | 2018-03-09 | 웰즐리 파마슈티컬스 엘엘씨 | 배뇨 빈도를 감소시키기 위한 연장-방출형 제제 및 이의 사용 방법 |
KR102237799B1 (ko) | 2012-11-14 | 2021-04-08 | 더블유.알. 그레이스 앤드 캄파니-콘. | 생물학적 활성 물질 및 비-정렬된 무기 산화물을 함유하는 조성물 |
PL3069733T3 (pl) * | 2013-11-13 | 2023-02-13 | National Defense Education And Research Foundation | Nowa kompozycja związku stanowiącego acetaminofen niepowodująca w wątrobie działań niepożądanych |
WO2016042570A1 (fr) * | 2014-09-16 | 2016-03-24 | Suresh Pareek | Formulation à libération prolongée d'acétaminophène |
JP7458317B2 (ja) * | 2017-10-31 | 2024-03-29 | サムヤン、ホールディングス、コーポレーション | 崩壊が改善された経口用固形製剤組成物及びその製造方法 |
JP6858729B2 (ja) * | 2018-05-25 | 2021-04-14 | ▲財▼▲団▼法人国防教育研究基金会National Defense Education And Research Foundation | 肝臓に対する副作用がない、新しいアセトアミノフェン複合組成 |
KR102168395B1 (ko) * | 2018-10-30 | 2020-10-22 | 한양대학교 에리카산학협력단 | 용해도가 개선된 실데나필 유리염기 고체분산체 및 이의 제조방법 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4820522A (en) * | 1987-07-27 | 1989-04-11 | Mcneilab, Inc. | Oral sustained release acetaminophen formulation and process |
US6149953A (en) * | 1993-11-08 | 2000-11-21 | Delta Food Group, Inc. | Seeded microcapsules |
US5948438A (en) * | 1995-01-09 | 1999-09-07 | Edward Mendell Co., Inc. | Pharmaceutical formulations having improved disintegration and/or absorptivity |
US5733578A (en) * | 1995-11-15 | 1998-03-31 | Edward Mendell Co., Inc. | Directly compressible high load acetaminophen formulations |
US6254891B1 (en) * | 1998-09-03 | 2001-07-03 | Ascent Pediatrics, Inc. | Extended release acetaminophen |
-
2002
- 2002-07-16 KR KR10-2002-0041469A patent/KR100522239B1/ko not_active IP Right Cessation
-
2003
- 2003-05-27 AU AU2003232652A patent/AU2003232652A1/en not_active Abandoned
- 2003-05-27 WO PCT/KR2003/001036 patent/WO2004006904A1/fr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
KR20040006887A (ko) | 2004-01-24 |
AU2003232652A1 (en) | 2004-02-02 |
WO2004006904A1 (fr) | 2004-01-22 |
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