KR100369417B1 - 제약상활성인화합물을제조하기위한중간체 - Google Patents

제약상활성인화합물을제조하기위한중간체 Download PDF

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Publication number
KR100369417B1
KR100369417B1 KR1019960706579A KR19960706579A KR100369417B1 KR 100369417 B1 KR100369417 B1 KR 100369417B1 KR 1019960706579 A KR1019960706579 A KR 1019960706579A KR 19960706579 A KR19960706579 A KR 19960706579A KR 100369417 B1 KR100369417 B1 KR 100369417B1
Authority
KR
South Korea
Prior art keywords
formula
compound
methyl
intermediates
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1019960706579A
Other languages
English (en)
Korean (ko)
Inventor
레이몬드 이. 데거
Original Assignee
스미스클라인 비참 코포레이션
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 스미스클라인 비참 코포레이션 filed Critical 스미스클라인 비참 코포레이션
Application granted granted Critical
Publication of KR100369417B1 publication Critical patent/KR100369417B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Lining Or Joining Of Plastics Or The Like (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Lubricants (AREA)
  • Detergent Compositions (AREA)
KR1019960706579A 1994-05-20 1995-05-04 제약상활성인화합물을제조하기위한중간체 Expired - Fee Related KR100369417B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24643194A 1994-05-20 1994-05-20
US08246,431 1994-05-20

Publications (1)

Publication Number Publication Date
KR100369417B1 true KR100369417B1 (ko) 2003-04-23

Family

ID=22930661

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019960706579A Expired - Fee Related KR100369417B1 (ko) 1994-05-20 1995-05-04 제약상활성인화합물을제조하기위한중간체

Country Status (20)

Country Link
US (1) US5719293A (https=)
EP (1) EP0850225B1 (https=)
JP (1) JPH10500681A (https=)
KR (1) KR100369417B1 (https=)
CN (1) CN1067059C (https=)
AT (1) ATE247091T1 (https=)
AU (1) AU690270B2 (https=)
BR (1) BR9507668A (https=)
CZ (1) CZ289968B6 (https=)
DE (1) DE69531507T2 (https=)
DK (1) DK0850225T3 (https=)
ES (1) ES2204950T3 (https=)
HU (1) HU221905B1 (https=)
MX (1) MX9605794A (https=)
NO (1) NO306673B1 (https=)
NZ (1) NZ285588A (https=)
PL (1) PL185858B1 (https=)
PT (1) PT850225E (https=)
WO (1) WO1995032189A1 (https=)
ZA (1) ZA954053B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR011125A1 (es) * 1997-02-14 2000-08-02 Smithkline Beecham Corp Procedimiento para preparar eprosartano

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1214324A (fr) * 1957-11-16 1960-04-07 Merck Ag E Procédé de préparation du pyridoxal et de ses dérivés à groupe aldéhyde protégé
US3798172A (en) * 1969-05-26 1974-03-19 Dan River Inc Dyeing textile materials with vat and sulfur dyes and reducing agent stabilizers for same
JPS518934B2 (https=) * 1972-02-04 1976-03-22
US4024067A (en) * 1976-01-07 1977-05-17 The United States Of America As Represented By The Secretary Of The Navy Processes for the preparation of bis-benzoins and bis-benzils
JPS55104254A (en) * 1979-02-05 1980-08-09 Kuraray Co Ltd N-substituted-alpha-cyano-3-phenoxybenzylamine
JPS55167274A (en) * 1979-06-14 1980-12-26 Banyu Pharmaceut Co Ltd Forphenicine derivative and its preparation
JPS5671074A (en) * 1979-11-12 1981-06-13 Takeda Chem Ind Ltd 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative
US5185351A (en) * 1989-06-14 1993-02-09 Smithkline Beecham Corporation Imidazolyl-alkenoic acids useful as angiotensin II receptor antagonists
WO1991000281A2 (en) * 1989-06-30 1991-01-10 E.I. Du Pont De Nemours And Company Fused-ring aryl substituted imidazoles
JPH03112940A (ja) * 1989-09-26 1991-05-14 Nkk Corp （±）―４―ホルミル―α―アルキルベンジルアルコール類の製造方法

Also Published As

Publication number Publication date
HUT75714A (en) 1997-05-28
DE69531507T2 (de) 2004-06-17
EP0850225A1 (en) 1998-07-01
PL317538A1 (en) 1997-04-14
NO964921L (no) 1996-11-20
MX9605794A (es) 1997-12-31
DE69531507D1 (de) 2003-09-18
AU2473795A (en) 1995-12-18
US5719293A (en) 1998-02-17
NO306673B1 (no) 1999-12-06
PL185858B1 (pl) 2003-08-29
BR9507668A (pt) 1997-10-07
NO964921D0 (no) 1996-11-19
CZ289968B6 (cs) 2002-05-15
ES2204950T3 (es) 2004-05-01
CZ340396A3 (en) 1997-03-12
EP0850225A4 (https=) 1998-07-01
EP0850225B1 (en) 2003-08-13
AU690270B2 (en) 1998-04-23
NZ285588A (en) 1997-12-19
CN1151734A (zh) 1997-06-11
DK0850225T3 (da) 2003-12-01
HU221905B1 (hu) 2003-02-28
WO1995032189A1 (en) 1995-11-30
ATE247091T1 (de) 2003-08-15
JPH10500681A (ja) 1998-01-20
HK1014939A1 (en) 1999-10-08
ZA954053B (en) 1996-01-19
CN1067059C (zh) 2001-06-13
HU9603205D0 (en) 1997-01-28
PT850225E (pt) 2003-11-28

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