KR100248537B1 - 유기물질에 대한 안정화제로서 유용한 테트라메틸피페리딘 화합물 - Google Patents

유기물질에 대한 안정화제로서 유용한 테트라메틸피페리딘 화합물 Download PDF

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KR100248537B1
KR100248537B1 KR1019920024858A KR920024858A KR100248537B1 KR 100248537 B1 KR100248537 B1 KR 100248537B1 KR 1019920024858 A KR1019920024858 A KR 1019920024858A KR 920024858 A KR920024858 A KR 920024858A KR 100248537 B1 KR100248537 B1 KR 100248537B1
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alkyl
alkylene
formula
group
different
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Korean (ko)
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보르자타 발레리오
비그날리 그라지아노
Original Assignee
에프. 아. 프라저
시바 스페셜티 케미칼스 홀딩 인크.
에른스트 알테르 (에. 알테르)
한스 페터 비틀린 (하. 페. 비틀린)
피. 랍 보프
브이. 스펜글러
페. 아에글러
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08KUse of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00Use of organic ingredients
    • C08K5/16Nitrogen-containing compounds
    • C08K5/34Heterocyclic compounds having nitrogen in the ring
    • C08K5/3442Heterocyclic compounds having nitrogen in the ring having two nitrogen atoms in the ring
    • C08K5/3445Five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Materials For Photolithography (AREA)
  • Detergent Compositions (AREA)
KR1019920024858A 1991-12-17 1992-12-16 유기물질에 대한 안정화제로서 유용한 테트라메틸피페리딘 화합물 Expired - Fee Related KR100248537B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI913374A IT1252227B (it) 1991-12-17 1991-12-17 Composti tetrametilpiperidinici atti all'impiego come stabilizzanti per materiali organici
ITMI91A003374 1991-12-17

Publications (1)

Publication Number Publication Date
KR100248537B1 true KR100248537B1 (ko) 2000-04-01

Family

ID=11361349

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019920024858A Expired - Fee Related KR100248537B1 (ko) 1991-12-17 1992-12-16 유기물질에 대한 안정화제로서 유용한 테트라메틸피페리딘 화합물

Country Status (10)

Country Link
US (1) US5310767A (enExample)
EP (1) EP0548015B1 (enExample)
JP (1) JPH05255312A (enExample)
KR (1) KR100248537B1 (enExample)
BR (1) BR9205032A (enExample)
CA (1) CA2085379A1 (enExample)
DE (1) DE69207370T2 (enExample)
ES (1) ES2082434T3 (enExample)
IT (1) IT1252227B (enExample)
TW (1) TW242156B (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1263892B (it) * 1993-02-11 1996-09-05 Graziano Vignali Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici
US5721250A (en) * 1993-12-23 1998-02-24 Merck & Co. Inc. Di-and tri-substituted piperidines, pyrrolidines and hexahydro-1H-azepines promote release of growth hormone
AU780006B2 (en) 2000-03-06 2005-02-24 Acadia Pharmaceuticals, Inc. Azacyclic compounds for use in the treatment of serotonin related diseases
NZ571695A (en) 2001-12-28 2010-02-26 Acadia Pharm Inc Spiroazacyclic compounds as monoamine receptor for modulating 5-HT2A receptor-mediated events
US7253186B2 (en) 2002-06-24 2007-08-07 Carl-Magnus Andersson N-substituted piperidine derivatives as serotonin receptor agents
MXPA04012893A (es) 2002-06-24 2005-03-31 Acadia Pharm Inc Derivados de piperidina n-substituidos como agentes receptores de serotonina.
US7538222B2 (en) 2002-06-24 2009-05-26 Acadia Pharmaceuticals, Inc. N-substituted piperidine derivatives as serotonin receptor agents
PT1587789E (pt) 2003-01-16 2008-12-16 Acadia Pharm Inc Agonistas inversos selectivos para receptores 2a/2c da serotonina como agentes terapêuticos para doenças neurodegenerativas
US20050261278A1 (en) 2004-05-21 2005-11-24 Weiner David M Selective serotonin receptor inverse agonists as therapeutics for disease
US7820695B2 (en) 2004-05-21 2010-10-26 Acadia Pharmaceuticals, Inc. Selective serotonin receptor inverse agonists as therapeutics for disease
CA2580136C (en) 2004-09-27 2015-08-18 Acadia Pharmaceuticals Inc. Synthesis of n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and crystalline forms
US7790899B2 (en) 2004-09-27 2010-09-07 Acadia Pharmaceuticals, Inc. Synthesis of N-(4-fluorobenzyl)-N-(1-methylpiperidin-4-yl)-N′-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and crystalline forms
CA2681506C (en) 2007-03-19 2016-05-24 Perry Peters Combinations of 5-ht2a inverse agonists and antagonists with antipsychotics
TWI386451B (zh) * 2009-05-12 2013-02-21 Nanya Plastics Corp 一種pvc樹脂組成物及其製品
CA2992728A1 (en) 2015-07-20 2017-01-26 Acadia Pharmaceuticals Inc. Methods for preparing n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and polymorphic form c
WO2017165635A1 (en) 2016-03-25 2017-09-28 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome p450 modulators
US10953000B2 (en) 2016-03-25 2021-03-23 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome P450 modulators
EP3558311A1 (en) 2016-12-20 2019-10-30 Acadia Pharmaceuticals Inc. Pimavanserin alone or in combination for use in the treatment of alzheimer's disease psychosis
EP3615028A1 (en) 2017-04-28 2020-03-04 Acadia Pharmaceuticals Inc. Pimavanserin for treating impulse control disorder
US20210077479A1 (en) 2017-08-30 2021-03-18 Acadia Pharmaceuticals Inc. Formulations of pimavanserin

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3684765A (en) * 1970-01-08 1972-08-15 Sankyo Co Stabilization of synthetic polymers
GB1393551A (en) * 1972-04-21 1975-05-07 Ciba Geigy Ag Piperidine derivatives
JPS557861B2 (enExample) * 1972-10-04 1980-02-28
IT1060458B (it) * 1975-12-18 1982-08-20 Chimosa Chimica Organica Spa Composti piperidil triazinici adatti per la stabilizzazione di polimeri sintetici e procedimento per la loro preparazione
IT1097753B (it) * 1978-07-28 1985-08-31 Chimosa Chimica Organica Spa Compcsti piperidinici, processo per la loro preparazione e loro impiego come stabil izzanti per polimeri sintetici
IT7921841A0 (it) * 1979-04-13 1979-04-13 Chimosa Chimica Organica Spa Nuovi composti piperidinici, processo per la loro preparazione e loro impiego come stabilizzanti per polimeri sintetici.
DE2944729A1 (de) * 1979-11-06 1981-05-14 Hoechst Ag, 6000 Frankfurt Neue triazinstabilisatoren
DE3382687D1 (de) * 1982-09-30 1993-07-01 Ciba Geigy Ag Mit bis-(polyalkylpiperidinyl-amino)-1,3,5-triazinen stabilisierte polyolefine.
JPS59122487A (ja) * 1982-12-28 1984-07-14 Sankyo Co Ltd ピペリジル−トリアジン−トリアミン誘導体及び高分子材料用安定剤
IT1193659B (it) * 1983-02-04 1988-07-21 Chimosa Chimica Organica Spa Composti piperidinil-triazinici utili come stabilizzanti per polimeri sintetici
JPS6181441A (ja) * 1984-09-28 1986-04-25 Adeka Argus Chem Co Ltd 高分子材料組成物
JPS6218444A (ja) * 1985-07-16 1987-01-27 Adeka Argus Chem Co Ltd 安定化された高分子材料組成物
IT1227334B (it) * 1988-08-04 1991-04-08 Ciba Geigy Spa Composti piperidin triazinici atti all'impiego come stabilizzanti per materiali organici.
IT1231329B (it) * 1989-07-28 1991-11-28 Ciba Geigy Spa Composti piperazin piperidinici atti all'impiego come stabilizzanti per materiali organici
IT1237129B (it) * 1989-11-10 1993-05-18 Valerio Borzatta Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici.
IT1243374B (it) * 1990-07-27 1994-06-10 Ciba Geigy Spa Composti piperidin-triazinici contenenti gruppi tetraidrofuranici o tetraidropiranici atti all'impiego come stabilizzanti per materiali organici
IT1243433B (it) * 1990-10-03 1994-06-10 Ciba Geigy Spa Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici
IT1243409B (it) * 1990-12-17 1994-06-10 Ciba Geigy Spa Composti piperidinici contenenti gruppi silenici atti all'impiego come stabilizzanti per materiali organici

Also Published As

Publication number Publication date
DE69207370D1 (de) 1996-02-15
CA2085379A1 (en) 1993-06-18
TW242156B (enExample) 1995-03-01
US5310767A (en) 1994-05-10
IT1252227B (it) 1995-06-05
JPH05255312A (ja) 1993-10-05
EP0548015A1 (en) 1993-06-23
EP0548015B1 (en) 1996-01-03
ITMI913374A1 (it) 1993-06-17
ES2082434T3 (es) 1996-03-16
BR9205032A (pt) 1993-06-22
DE69207370T2 (de) 1996-11-14
ITMI913374A0 (it) 1991-12-17

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