KR100236246B1 - 디리트로마이신의 일단계 제조방법 - Google Patents

디리트로마이신의 일단계 제조방법 Download PDF

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Publication number
KR100236246B1
KR100236246B1 KR1019920017679A KR920017679A KR100236246B1 KR 100236246 B1 KR100236246 B1 KR 100236246B1 KR 1019920017679 A KR1019920017679 A KR 1019920017679A KR 920017679 A KR920017679 A KR 920017679A KR 100236246 B1 KR100236246 B1 KR 100236246B1
Authority
KR
South Korea
Prior art keywords
acetal
reaction
hydrolysis
amount
dilitthromycin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1019920017679A
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English (en)
Korean (ko)
Other versions
KR930006044A (ko
Inventor
맥닐 맥길 존
Original Assignee
피터 지. 스트링거
일라이 릴리 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 피터 지. 스트링거, 일라이 릴리 앤드 캄파니 filed Critical 피터 지. 스트링거
Publication of KR930006044A publication Critical patent/KR930006044A/ko
Application granted granted Critical
Publication of KR100236246B1 publication Critical patent/KR100236246B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1019920017679A 1991-09-30 1992-09-28 디리트로마이신의 일단계 제조방법 Expired - Fee Related KR100236246B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76880391A 1991-09-30 1991-09-30
US768,803 1991-09-30

Publications (2)

Publication Number Publication Date
KR930006044A KR930006044A (ko) 1993-04-20
KR100236246B1 true KR100236246B1 (ko) 1999-12-15

Family

ID=25083529

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019920017679A Expired - Fee Related KR100236246B1 (ko) 1991-09-30 1992-09-28 디리트로마이신의 일단계 제조방법

Country Status (28)

Country Link
US (1) US5578713A (enExample)
EP (1) EP0535900B1 (enExample)
JP (1) JP3197957B2 (enExample)
KR (1) KR100236246B1 (enExample)
CN (1) CN1030455C (enExample)
AR (1) AR248282A1 (enExample)
AT (1) ATE133178T1 (enExample)
BR (1) BR9203799A (enExample)
CA (1) CA2079430A1 (enExample)
CZ (1) CZ281664B6 (enExample)
DE (1) DE69207696T2 (enExample)
DK (1) DK0535900T3 (enExample)
ES (1) ES2083103T3 (enExample)
FI (1) FI104969B (enExample)
GR (1) GR3018726T3 (enExample)
HK (1) HK1006842A1 (enExample)
HU (1) HU213620B (enExample)
IL (1) IL103276A (enExample)
MX (1) MX9205455A (enExample)
MY (1) MY113261A (enExample)
NO (1) NO178150C (enExample)
NZ (1) NZ244495A (enExample)
PH (1) PH30959A (enExample)
RU (1) RU2045534C1 (enExample)
SK (1) SK279270B6 (enExample)
TW (1) TW287165B (enExample)
YU (1) YU48748B (enExample)
ZA (1) ZA927328B (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA966601B (en) * 1995-08-03 1997-02-19 Chugai Pharmaceutical Co Ltd Process for producing erythromycin derivatives.
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
WO2005009364A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
EP1648415A4 (en) 2003-07-21 2011-11-16 Middlebrook Pharmaceuticals Inc ANTIBIOTIC PRODUCT, ITS USE AND FORMULATION
WO2005009368A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
CA2535177A1 (en) 2003-08-11 2005-02-24 Advancis Pharmaceutical Corporation Robust pellet
JP2007502294A (ja) 2003-08-12 2007-02-08 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
AU2004270170B2 (en) * 2003-08-29 2011-01-27 Shionogi, Inc. Antibiotic product, use and formulation thereof
WO2005027877A1 (en) 2003-09-15 2005-03-31 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
CA2572292A1 (en) 2004-07-02 2006-02-09 Advancis Pharmaceutical Corporation Tablet for pulsed delivery
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8299052B2 (en) 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
US4438109A (en) * 1980-07-25 1984-03-20 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Tylosin derivatives
JPS62103098A (ja) * 1985-05-13 1987-05-13 Microbial Chem Res Found タイロシン誘導体

Also Published As

Publication number Publication date
FI924360A0 (fi) 1992-09-29
KR930006044A (ko) 1993-04-20
IL103276A0 (en) 1993-02-21
FI104969B (fi) 2000-05-15
EP0535900B1 (en) 1996-01-17
CZ293592A3 (en) 1993-04-14
TW287165B (enExample) 1996-10-01
HUT62308A (en) 1993-04-28
AU645443B2 (en) 1994-01-13
DE69207696T2 (de) 1996-06-05
RU2045534C1 (ru) 1995-10-10
CN1070914A (zh) 1993-04-14
HU9203101D0 (en) 1992-12-28
DK0535900T3 (da) 1996-02-12
ATE133178T1 (de) 1996-02-15
CN1030455C (zh) 1995-12-06
MY113261A (en) 2002-01-31
BR9203799A (pt) 1993-04-20
CA2079430A1 (en) 1993-03-31
IL103276A (en) 1997-06-10
DE69207696D1 (de) 1996-02-29
YU87792A (sh) 1995-03-27
NZ244495A (en) 1995-04-27
NO178150C (no) 1996-01-31
HU213620B (en) 1997-08-28
EP0535900A1 (en) 1993-04-07
NO923765L (no) 1993-03-31
AR248282A1 (es) 1995-07-12
HK1006842A1 (en) 1999-03-19
MX9205455A (es) 1993-05-01
YU48748B (sh) 1999-09-27
ES2083103T3 (es) 1996-04-01
US5578713A (en) 1996-11-26
GR3018726T3 (en) 1996-04-30
JPH05213983A (ja) 1993-08-24
SK293592A3 (en) 1998-08-05
JP3197957B2 (ja) 2001-08-13
PH30959A (en) 1997-12-23
ZA927328B (en) 1994-03-24
NO178150B (no) 1995-10-23
NO923765D0 (no) 1992-09-28
AU2536592A (en) 1993-04-01
CZ281664B6 (cs) 1996-12-11
FI924360L (fi) 1993-03-31
SK279270B6 (sk) 1998-08-05

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