HK1006842A1 - One step process for production of dirithromycin - Google Patents

One step process for production of dirithromycin Download PDF

Info

Publication number
HK1006842A1
HK1006842A1 HK98105921A HK98105921A HK1006842A1 HK 1006842 A1 HK1006842 A1 HK 1006842A1 HK 98105921 A HK98105921 A HK 98105921A HK 98105921 A HK98105921 A HK 98105921A HK 1006842 A1 HK1006842 A1 HK 1006842A1
Authority
HK
Hong Kong
Prior art keywords
acetal
erythromycylamine
dirithromycin
acid
amount
Prior art date
Application number
HK98105921A
Other languages
German (de)
English (en)
French (fr)
Chinese (zh)
Other versions
HK1006842B (en
Inventor
Mcneil Mcgill John
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of HK1006842B publication Critical patent/HK1006842B/en
Publication of HK1006842A1 publication Critical patent/HK1006842A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HK98105921A 1991-09-30 1998-06-22 One step process for production of dirithromycin HK1006842A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76880391A 1991-09-30 1991-09-30
US768803 1991-09-30

Publications (2)

Publication Number Publication Date
HK1006842B HK1006842B (en) 1999-03-19
HK1006842A1 true HK1006842A1 (en) 1999-03-19

Family

ID=25083529

Family Applications (1)

Application Number Title Priority Date Filing Date
HK98105921A HK1006842A1 (en) 1991-09-30 1998-06-22 One step process for production of dirithromycin

Country Status (28)

Country Link
US (1) US5578713A (enExample)
EP (1) EP0535900B1 (enExample)
JP (1) JP3197957B2 (enExample)
KR (1) KR100236246B1 (enExample)
CN (1) CN1030455C (enExample)
AR (1) AR248282A1 (enExample)
AT (1) ATE133178T1 (enExample)
BR (1) BR9203799A (enExample)
CA (1) CA2079430A1 (enExample)
CZ (1) CZ281664B6 (enExample)
DE (1) DE69207696T2 (enExample)
DK (1) DK0535900T3 (enExample)
ES (1) ES2083103T3 (enExample)
FI (1) FI104969B (enExample)
GR (1) GR3018726T3 (enExample)
HK (1) HK1006842A1 (enExample)
HU (1) HU213620B (enExample)
IL (1) IL103276A (enExample)
MX (1) MX9205455A (enExample)
MY (1) MY113261A (enExample)
NO (1) NO178150C (enExample)
NZ (1) NZ244495A (enExample)
PH (1) PH30959A (enExample)
RU (1) RU2045534C1 (enExample)
SK (1) SK279270B6 (enExample)
TW (1) TW287165B (enExample)
YU (1) YU48748B (enExample)
ZA (1) ZA927328B (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA966601B (en) * 1995-08-03 1997-02-19 Chugai Pharmaceutical Co Ltd Process for producing erythromycin derivatives.
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
WO2005009364A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
EP1648415A4 (en) 2003-07-21 2011-11-16 Middlebrook Pharmaceuticals Inc ANTIBIOTIC PRODUCT, ITS USE AND FORMULATION
WO2005009368A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
CA2535177A1 (en) 2003-08-11 2005-02-24 Advancis Pharmaceutical Corporation Robust pellet
JP2007502294A (ja) 2003-08-12 2007-02-08 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
AU2004270170B2 (en) * 2003-08-29 2011-01-27 Shionogi, Inc. Antibiotic product, use and formulation thereof
WO2005027877A1 (en) 2003-09-15 2005-03-31 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
CA2572292A1 (en) 2004-07-02 2006-02-09 Advancis Pharmaceutical Corporation Tablet for pulsed delivery
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8299052B2 (en) 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
US4438109A (en) * 1980-07-25 1984-03-20 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Tylosin derivatives
JPS62103098A (ja) * 1985-05-13 1987-05-13 Microbial Chem Res Found タイロシン誘導体

Also Published As

Publication number Publication date
FI924360A0 (fi) 1992-09-29
KR930006044A (ko) 1993-04-20
IL103276A0 (en) 1993-02-21
FI104969B (fi) 2000-05-15
EP0535900B1 (en) 1996-01-17
CZ293592A3 (en) 1993-04-14
TW287165B (enExample) 1996-10-01
HUT62308A (en) 1993-04-28
AU645443B2 (en) 1994-01-13
DE69207696T2 (de) 1996-06-05
RU2045534C1 (ru) 1995-10-10
CN1070914A (zh) 1993-04-14
HU9203101D0 (en) 1992-12-28
DK0535900T3 (da) 1996-02-12
ATE133178T1 (de) 1996-02-15
CN1030455C (zh) 1995-12-06
MY113261A (en) 2002-01-31
BR9203799A (pt) 1993-04-20
CA2079430A1 (en) 1993-03-31
IL103276A (en) 1997-06-10
DE69207696D1 (de) 1996-02-29
YU87792A (sh) 1995-03-27
NZ244495A (en) 1995-04-27
NO178150C (no) 1996-01-31
KR100236246B1 (ko) 1999-12-15
HU213620B (en) 1997-08-28
EP0535900A1 (en) 1993-04-07
NO923765L (no) 1993-03-31
AR248282A1 (es) 1995-07-12
MX9205455A (es) 1993-05-01
YU48748B (sh) 1999-09-27
ES2083103T3 (es) 1996-04-01
US5578713A (en) 1996-11-26
GR3018726T3 (en) 1996-04-30
JPH05213983A (ja) 1993-08-24
SK293592A3 (en) 1998-08-05
JP3197957B2 (ja) 2001-08-13
PH30959A (en) 1997-12-23
ZA927328B (en) 1994-03-24
NO178150B (no) 1995-10-23
NO923765D0 (no) 1992-09-28
AU2536592A (en) 1993-04-01
CZ281664B6 (cs) 1996-12-11
FI924360L (fi) 1993-03-31
SK279270B6 (sk) 1998-08-05

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Legal Events

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)