JPWO2022014680A5 - - Google Patents
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- Publication number
- JPWO2022014680A5 JPWO2022014680A5 JP2022536446A JP2022536446A JPWO2022014680A5 JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5 JP 2022536446 A JP2022536446 A JP 2022536446A JP 2022536446 A JP2022536446 A JP 2022536446A JP WO2022014680 A5 JPWO2022014680 A5 JP WO2022014680A5
- Authority
- JP
- Japan
- Prior art keywords
- octan
- azabicyclo
- represented
- formula
- fluoropyrimidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- DLFVBJFMPXGRIB-UHFFFAOYSA-N thioacetamide Natural products CC(N)=O DLFVBJFMPXGRIB-UHFFFAOYSA-N 0.000 claims 6
- 150000003839 salts Chemical class 0.000 claims 5
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020122864 | 2020-07-17 | ||
| JP2020122864 | 2020-07-17 | ||
| PCT/JP2021/026649 WO2022014680A1 (ja) | 2020-07-17 | 2021-07-15 | 置換ピペリジン化合物及びその用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2022014680A1 JPWO2022014680A1 (https=) | 2022-01-20 |
| JP7190612B2 JP7190612B2 (ja) | 2022-12-15 |
| JPWO2022014680A5 true JPWO2022014680A5 (https=) | 2022-12-16 |
Family
ID=79291962
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022536446A Active JP7190612B2 (ja) | 2020-07-17 | 2021-07-15 | 置換ピペリジン化合物及びその用途 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US11479552B2 (https=) |
| EP (1) | EP4151277B1 (https=) |
| JP (1) | JP7190612B2 (https=) |
| KR (1) | KR20230040953A (https=) |
| CN (3) | CN119235864A (https=) |
| AR (1) | AR122973A1 (https=) |
| AU (1) | AU2021308053A1 (https=) |
| BR (1) | BR112022026161A2 (https=) |
| CA (1) | CA3187835A1 (https=) |
| CL (1) | CL2022003666A1 (https=) |
| CO (1) | CO2022018446A2 (https=) |
| DK (1) | DK4151277T3 (https=) |
| FI (1) | FI4151277T3 (https=) |
| IL (1) | IL299125B2 (https=) |
| JO (1) | JOP20220345A1 (https=) |
| LT (1) | LT4151277T (https=) |
| MX (1) | MX2022016388A (https=) |
| PE (1) | PE20231103A1 (https=) |
| PH (1) | PH12022553488A1 (https=) |
| TW (1) | TWI888599B (https=) |
| UA (1) | UA129636C2 (https=) |
| WO (1) | WO2022014680A1 (https=) |
| ZA (1) | ZA202213562B (https=) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4065585B1 (en) | 2019-11-25 | 2025-08-20 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| US11760747B2 (en) | 2020-12-21 | 2023-09-19 | Alkermes, Inc. | Substituted piperidino compounds and related methods of treatment |
| US12006330B2 (en) | 2020-12-21 | 2024-06-11 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| JP7591592B2 (ja) * | 2022-01-14 | 2024-11-28 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 置換ピペリジン化合物を含有する医薬 |
| JPWO2023136279A1 (https=) * | 2022-01-14 | 2023-07-20 | ||
| WO2024075825A1 (ja) * | 2022-10-07 | 2024-04-11 | キッセイ薬品工業株式会社 | シクロペンタン化合物 |
| EP4611745A1 (en) * | 2022-10-31 | 2025-09-10 | Takeda Pharmaceutical Company Limited | Dosing of orexin type 2 receptor agonists |
| WO2024128305A1 (ja) | 2022-12-16 | 2024-06-20 | 第一三共株式会社 | ２－アザビシクロ［３．１．１］ヘプタン化合物 |
| EP4719397A1 (en) | 2023-06-02 | 2026-04-08 | Takeda Pharmaceutical Company Limited | Use of an orexin 2 receptor agonist for improving respiratory function during sleep |
| WO2025124698A1 (en) | 2023-12-12 | 2025-06-19 | Idorsia Pharmaceuticals Ltd | Aryl sulfone and sulfanone derivatives as orexin receptor modulators |
| TW202542165A (zh) | 2023-12-19 | 2025-11-01 | 瑞士商愛杜西亞製藥有限公司 | 大環食慾素激動劑 |
| WO2025137359A1 (en) | 2023-12-20 | 2025-06-26 | Eisai R&D Management Co., Ltd. | Assay methods to identify a disease |
| WO2025229493A1 (en) | 2024-04-29 | 2025-11-06 | Takeda Pharmaceutical Company Limited | Dosing of orexin type 2 receptor agonists |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG34208A1 (en) | 1995-03-01 | 1996-12-06 | Guy Andrew Vaz | Blast and fragment resistant polyurethane boot sole for safety footwear |
| EP0828751A4 (en) | 1995-05-05 | 1999-01-20 | Human Genome Sciences Inc | HUMAN NEUROPEPTIDE RECEPTOR |
| US6309854B1 (en) | 1996-12-17 | 2001-10-30 | Smithkline Beecham Corporation | Polynucleotides encoding ligands of the neuropeptide receptor HFGAN72 |
| US6159605A (en) | 1997-02-18 | 2000-12-12 | Dainichiseika Color & Chemicals Mfg. Co., Ltd. | Ink-jet recording sheet |
| US5935814A (en) | 1997-04-30 | 1999-08-10 | Smithkline Beecham Corporation | Polynucleotides encoding HFGAN72Y receptor |
| US6020157A (en) | 1997-04-30 | 2000-02-01 | Smithkline Beecham Corporation | Polynucleotides encoding HFGAN72X receptor |
| US6166193A (en) | 1997-07-25 | 2000-12-26 | Board Of Regents, University Of Texas System | Polynucleotides encoding MY1 receptor |
| KR100327888B1 (ko) | 1999-07-14 | 2002-03-09 | 정숭렬 | 도로포장 파손촉진 시험장치의 무선제어 시스템 |
| AU2004274309B2 (en) * | 2003-09-22 | 2010-04-08 | Msd K.K. | Novel piperidine derivative |
| EP1805183B1 (en) | 2004-10-20 | 2010-12-29 | NeuroSearch A/S | Novel diazabicyclic aryl derivatives and their medical use |
| JP2009184924A (ja) | 2006-05-31 | 2009-08-20 | Eisai R & D Management Co Ltd | 生物学的試薬用化合物 |
| TW201444849A (zh) | 2013-03-13 | 2014-12-01 | Janssen Pharmaceutica Nv | 經取代的7-氮雜雙環類及其作為食慾激素受體調節劑之用途 |
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2021
- 2021-07-15 TW TW110126031A patent/TWI888599B/zh active
- 2021-07-15 DK DK21842047.9T patent/DK4151277T3/da active
- 2021-07-15 PE PE2022003006A patent/PE20231103A1/es unknown
- 2021-07-15 PH PH1/2022/553488A patent/PH12022553488A1/en unknown
- 2021-07-15 CN CN202411459551.4A patent/CN119235864A/zh active Pending
- 2021-07-15 AR ARP210101982A patent/AR122973A1/es unknown
- 2021-07-15 UA UAA202204882A patent/UA129636C2/uk unknown
- 2021-07-15 EP EP21842047.9A patent/EP4151277B1/en active Active
- 2021-07-15 WO PCT/JP2021/026649 patent/WO2022014680A1/ja not_active Ceased
- 2021-07-15 IL IL299125A patent/IL299125B2/en unknown
- 2021-07-15 AU AU2021308053A patent/AU2021308053A1/en active Pending
- 2021-07-15 CN CN202180044081.3A patent/CN115884971B/zh active Active
- 2021-07-15 US US17/376,452 patent/US11479552B2/en active Active
- 2021-07-15 CN CN202411462171.6A patent/CN119258067A/zh active Pending
- 2021-07-15 CA CA3187835A patent/CA3187835A1/en active Pending
- 2021-07-15 FI FIEP21842047.9T patent/FI4151277T3/fi active
- 2021-07-15 LT LTEPPCT/JP2021/026649T patent/LT4151277T/lt unknown
- 2021-07-15 KR KR1020227044679A patent/KR20230040953A/ko active Pending
- 2021-07-15 JP JP2022536446A patent/JP7190612B2/ja active Active
- 2021-07-15 BR BR112022026161A patent/BR112022026161A2/pt unknown
- 2021-07-15 MX MX2022016388A patent/MX2022016388A/es unknown
-
2022
- 2022-12-14 ZA ZA2022/13562A patent/ZA202213562B/en unknown
- 2022-12-20 CL CL2022003666A patent/CL2022003666A1/es unknown
- 2022-12-20 CO CONC2022/0018446A patent/CO2022018446A2/es unknown
- 2022-12-21 JO JOJO/P/2022/0345A patent/JOP20220345A1/ar unknown