JPWO2021072198A5 - - Google Patents

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Publication number
JPWO2021072198A5
JPWO2021072198A5 JP2022520897A JP2022520897A JPWO2021072198A5 JP WO2021072198 A5 JPWO2021072198 A5 JP WO2021072198A5 JP 2022520897 A JP2022520897 A JP 2022520897A JP 2022520897 A JP2022520897 A JP 2022520897A JP WO2021072198 A5 JPWO2021072198 A5 JP WO2021072198A5
Authority
JP
Japan
Prior art keywords
alkyl
formula
optionally substituted
cycloalkyl
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022520897A
Other languages
English (en)
Japanese (ja)
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JP2022552185A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/054992 external-priority patent/WO2021072198A1/fr
Publication of JP2022552185A publication Critical patent/JP2022552185A/ja
Publication of JPWO2021072198A5 publication Critical patent/JPWO2021072198A5/ja
Pending legal-status Critical Current

Links

JP2022520897A 2019-10-09 2020-10-09 経口補体因子d阻害剤 Pending JP2022552185A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962912929P 2019-10-09 2019-10-09
US62/912,929 2019-10-09
PCT/US2020/054992 WO2021072198A1 (fr) 2019-10-09 2020-10-09 Inhibiteurs oraux du facteur d du complément

Publications (2)

Publication Number Publication Date
JP2022552185A JP2022552185A (ja) 2022-12-15
JPWO2021072198A5 true JPWO2021072198A5 (fr) 2023-10-12

Family

ID=75436778

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022520897A Pending JP2022552185A (ja) 2019-10-09 2020-10-09 経口補体因子d阻害剤

Country Status (20)

Country Link
EP (1) EP4041238A4 (fr)
JP (1) JP2022552185A (fr)
KR (1) KR20220100585A (fr)
CN (1) CN114502168A (fr)
AR (1) AR120173A1 (fr)
AU (1) AU2020361600A1 (fr)
BR (1) BR112022006572A2 (fr)
CA (1) CA3156287A1 (fr)
CL (1) CL2022000875A1 (fr)
CO (1) CO2022005999A2 (fr)
CR (1) CR20220199A (fr)
CU (1) CU20220024A7 (fr)
EC (1) ECSP22036502A (fr)
IL (1) IL291942A (fr)
JO (1) JOP20220075A1 (fr)
MX (1) MX2022004197A (fr)
PE (1) PE20221270A1 (fr)
TW (1) TW202128637A (fr)
UY (1) UY38912A (fr)
WO (1) WO2021072198A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021021909A1 (fr) * 2019-07-31 2021-02-04 Biocryst Pharmaceuticals, Inc. Schémas posologiques pour inhibiteurs oraux du facteur d du complément
TW202304890A (zh) * 2021-04-14 2023-02-01 美商百歐克斯製藥公司 Klk5雙環雜芳香族抑制劑
TW202330489A (zh) * 2021-10-21 2023-08-01 大陸商江蘇恆瑞醫藥股份有限公司 稠合環類化合物、其製備方法及其在醫藥上的應用
WO2023227696A1 (fr) * 2022-05-25 2023-11-30 Katholieke Universiteit Leuven Nouveaux dérivés pour le traitement de troubles médiés par trpm3

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3900261A1 (de) * 1988-05-31 1989-12-07 Bayer Ag Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
US6277877B1 (en) * 2000-08-15 2001-08-21 Pfizer, Inc. Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors
US7919519B2 (en) * 2005-11-23 2011-04-05 Epix Pharmaceuticals Inc. S1P receptor modulating compounds and use thereof
AU2012203083A1 (en) * 2006-02-03 2012-06-14 Bionomics Limited Substituted benzofurans, benzothiophenes, benzoselenophenes and indoles and their use as tubulin polymerisation inhibitors
AR076126A1 (es) * 2009-03-18 2011-05-18 Schering Corp Compuestos biciclicos como inhibidores de diacilglicerol aciltransferasa
WO2016088082A1 (fr) * 2014-12-05 2016-06-09 Novartis Ag Dérivés d'aminométhyl-biaryle en tant qu'inhibiteurs du facteur d du complément et leurs utilisations
TWI747873B (zh) * 2016-02-01 2021-12-01 美商百歐克斯製藥公司 苯并吡唑化合物及其類似物
WO2019057946A1 (fr) * 2017-09-25 2019-03-28 F. Hoffmann-La Roche Ag Composés aromatiques multi-cycliques utilisés en tant qu'inhibiteurs du facteur d
TW202010742A (zh) * 2018-04-06 2020-03-16 美商百歐克斯製藥公司 取代的苯并呋喃、苯并吡咯、苯并噻吩及結構相關的補體抑制劑

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