JPWO2021072198A5 - - Google Patents
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- Publication number
- JPWO2021072198A5 JPWO2021072198A5 JP2022520897A JP2022520897A JPWO2021072198A5 JP WO2021072198 A5 JPWO2021072198 A5 JP WO2021072198A5 JP 2022520897 A JP2022520897 A JP 2022520897A JP 2022520897 A JP2022520897 A JP 2022520897A JP WO2021072198 A5 JPWO2021072198 A5 JP WO2021072198A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- optionally substituted
- cycloalkyl
- compound according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962912929P | 2019-10-09 | 2019-10-09 | |
US62/912,929 | 2019-10-09 | ||
PCT/US2020/054992 WO2021072198A1 (fr) | 2019-10-09 | 2020-10-09 | Inhibiteurs oraux du facteur d du complément |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2022552185A JP2022552185A (ja) | 2022-12-15 |
JPWO2021072198A5 true JPWO2021072198A5 (fr) | 2023-10-12 |
Family
ID=75436778
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2022520897A Pending JP2022552185A (ja) | 2019-10-09 | 2020-10-09 | 経口補体因子d阻害剤 |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP4041238A4 (fr) |
JP (1) | JP2022552185A (fr) |
KR (1) | KR20220100585A (fr) |
CN (1) | CN114502168A (fr) |
AR (1) | AR120173A1 (fr) |
AU (1) | AU2020361600A1 (fr) |
BR (1) | BR112022006572A2 (fr) |
CA (1) | CA3156287A1 (fr) |
CL (1) | CL2022000875A1 (fr) |
CO (1) | CO2022005999A2 (fr) |
CR (1) | CR20220199A (fr) |
CU (1) | CU20220024A7 (fr) |
EC (1) | ECSP22036502A (fr) |
IL (1) | IL291942A (fr) |
JO (1) | JOP20220075A1 (fr) |
MX (1) | MX2022004197A (fr) |
PE (1) | PE20221270A1 (fr) |
TW (1) | TW202128637A (fr) |
UY (1) | UY38912A (fr) |
WO (1) | WO2021072198A1 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2021021909A1 (fr) * | 2019-07-31 | 2021-02-04 | Biocryst Pharmaceuticals, Inc. | Schémas posologiques pour inhibiteurs oraux du facteur d du complément |
TW202304890A (zh) * | 2021-04-14 | 2023-02-01 | 美商百歐克斯製藥公司 | Klk5雙環雜芳香族抑制劑 |
TW202330489A (zh) * | 2021-10-21 | 2023-08-01 | 大陸商江蘇恆瑞醫藥股份有限公司 | 稠合環類化合物、其製備方法及其在醫藥上的應用 |
WO2023227696A1 (fr) * | 2022-05-25 | 2023-11-30 | Katholieke Universiteit Leuven | Nouveaux dérivés pour le traitement de troubles médiés par trpm3 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3900261A1 (de) * | 1988-05-31 | 1989-12-07 | Bayer Ag | Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate |
US6277877B1 (en) * | 2000-08-15 | 2001-08-21 | Pfizer, Inc. | Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors |
US7919519B2 (en) * | 2005-11-23 | 2011-04-05 | Epix Pharmaceuticals Inc. | S1P receptor modulating compounds and use thereof |
AU2012203083A1 (en) * | 2006-02-03 | 2012-06-14 | Bionomics Limited | Substituted benzofurans, benzothiophenes, benzoselenophenes and indoles and their use as tubulin polymerisation inhibitors |
AR076126A1 (es) * | 2009-03-18 | 2011-05-18 | Schering Corp | Compuestos biciclicos como inhibidores de diacilglicerol aciltransferasa |
WO2016088082A1 (fr) * | 2014-12-05 | 2016-06-09 | Novartis Ag | Dérivés d'aminométhyl-biaryle en tant qu'inhibiteurs du facteur d du complément et leurs utilisations |
TWI747873B (zh) * | 2016-02-01 | 2021-12-01 | 美商百歐克斯製藥公司 | 苯并吡唑化合物及其類似物 |
WO2019057946A1 (fr) * | 2017-09-25 | 2019-03-28 | F. Hoffmann-La Roche Ag | Composés aromatiques multi-cycliques utilisés en tant qu'inhibiteurs du facteur d |
TW202010742A (zh) * | 2018-04-06 | 2020-03-16 | 美商百歐克斯製藥公司 | 取代的苯并呋喃、苯并吡咯、苯并噻吩及結構相關的補體抑制劑 |
-
2020
- 2020-10-08 UY UY0001038912A patent/UY38912A/es unknown
- 2020-10-08 TW TW109135076A patent/TW202128637A/zh unknown
- 2020-10-08 AR ARP200102782A patent/AR120173A1/es unknown
- 2020-10-09 EP EP20874925.9A patent/EP4041238A4/fr active Pending
- 2020-10-09 WO PCT/US2020/054992 patent/WO2021072198A1/fr unknown
- 2020-10-09 MX MX2022004197A patent/MX2022004197A/es unknown
- 2020-10-09 CU CU2022000024A patent/CU20220024A7/es unknown
- 2020-10-09 CR CR20220199A patent/CR20220199A/es unknown
- 2020-10-09 JP JP2022520897A patent/JP2022552185A/ja active Pending
- 2020-10-09 CA CA3156287A patent/CA3156287A1/fr active Pending
- 2020-10-09 KR KR1020227015220A patent/KR20220100585A/ko unknown
- 2020-10-09 JO JOP/2022/0075A patent/JOP20220075A1/ar unknown
- 2020-10-09 AU AU2020361600A patent/AU2020361600A1/en active Pending
- 2020-10-09 PE PE2022000576A patent/PE20221270A1/es unknown
- 2020-10-09 BR BR112022006572A patent/BR112022006572A2/pt unknown
- 2020-10-09 CN CN202080070572.0A patent/CN114502168A/zh active Pending
-
2022
- 2022-04-04 IL IL291942A patent/IL291942A/en unknown
- 2022-04-06 CL CL2022000875A patent/CL2022000875A1/es unknown
- 2022-05-06 EC ECSENADI202236502A patent/ECSP22036502A/es unknown
- 2022-05-09 CO CONC2022/0005999A patent/CO2022005999A2/es unknown
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