JPWO2021059136A5 - - Google Patents

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Publication number
JPWO2021059136A5
JPWO2021059136A5 JP2022518675A JP2022518675A JPWO2021059136A5 JP WO2021059136 A5 JPWO2021059136 A5 JP WO2021059136A5 JP 2022518675 A JP2022518675 A JP 2022518675A JP 2022518675 A JP2022518675 A JP 2022518675A JP WO2021059136 A5 JPWO2021059136 A5 JP WO2021059136A5
Authority
JP
Japan
Prior art keywords
cancer
pharmaceutically acceptable
acceptable salt
alkylene
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022518675A
Other languages
English (en)
Japanese (ja)
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JP2022550297A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2020/058854 external-priority patent/WO2021059136A1/fr
Publication of JP2022550297A publication Critical patent/JP2022550297A/ja
Publication of JPWO2021059136A5 publication Critical patent/JPWO2021059136A5/ja
Pending legal-status Critical Current

Links

JP2022518675A 2019-09-25 2020-09-22 Sting(インターフェロン遺伝子刺激因子)のヘテロ多環式モジュレーター Pending JP2022550297A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201962905532P 2019-09-25 2019-09-25
US62/905,532 2019-09-25
US202063021216P 2020-05-07 2020-05-07
US63/021,216 2020-05-07
US202063069831P 2020-08-25 2020-08-25
US63/069,831 2020-08-25
PCT/IB2020/058854 WO2021059136A1 (fr) 2019-09-25 2020-09-22 Modulateurs polyhétérocycliques de sting (stimulateur des gènes de l'interféron)

Publications (2)

Publication Number Publication Date
JP2022550297A JP2022550297A (ja) 2022-12-01
JPWO2021059136A5 true JPWO2021059136A5 (fr) 2023-09-25

Family

ID=72744805

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022518675A Pending JP2022550297A (ja) 2019-09-25 2020-09-22 Sting(インターフェロン遺伝子刺激因子)のヘテロ多環式モジュレーター

Country Status (19)

Country Link
US (1) US20210087180A1 (fr)
EP (1) EP4034534A1 (fr)
JP (1) JP2022550297A (fr)
KR (1) KR20220070254A (fr)
CN (1) CN114728946A (fr)
AU (1) AU2020355343B2 (fr)
BR (1) BR112022005463A2 (fr)
CA (1) CA3155569A1 (fr)
CL (1) CL2022000736A1 (fr)
CO (1) CO2022003321A2 (fr)
CR (1) CR20220126A (fr)
EC (1) ECSP22022958A (fr)
GE (1) GEP20237572B (fr)
IL (1) IL291650A (fr)
MX (1) MX2022003633A (fr)
PE (1) PE20221784A1 (fr)
TW (2) TW202244043A (fr)
UY (1) UY38892A (fr)
WO (1) WO2021059136A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022063205A1 (fr) * 2020-09-24 2022-03-31 中国医药研究开发中心有限公司 Composé aryl formamide, son procédé de préparation et ses utilisations médicales
US11964978B2 (en) 2021-03-18 2024-04-23 Pfizer Inc. Modulators of STING (stimulator of interferon genes)
US20220388986A1 (en) * 2021-04-29 2022-12-08 Boehringer Ingelheim International Gmbh Heterocyclic compounds capable of activating sting
WO2023222644A1 (fr) * 2022-05-18 2023-11-23 F. Hoffmann-La Roche Ag Dérivés de pyrazole utilisés en tant qu'agonistes de sting

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
US9040538B2 (en) 2009-05-21 2015-05-26 Universite Laval Pyrimidines as novel therapeutic agents
PL2614082T3 (pl) 2010-09-09 2019-02-28 Pfizer Inc. Cząsteczki wiążące 4-1BB
TWI595006B (zh) 2014-12-09 2017-08-11 禮納特神經系統科學公司 抗pd-1抗體類和使用彼等之方法
CN108473587A (zh) 2016-01-25 2018-08-31 辉瑞公司 用于治疗癌症的ox40激动剂和4-1bb激动剂单克隆抗体的组合
SG11201808708RA (en) * 2016-04-07 2018-11-29 Glaxosmithkline Ip Dev Ltd Heterocyclic amides useful as protein modulators
CA3067257A1 (fr) * 2017-06-22 2018-12-27 Curadev Pharma Limited Modulateurs a petites molecules de sting humain
US20200399268A1 (en) * 2018-02-16 2020-12-24 UCB Biopharma SRL Pharmaceutical 6,5 Heterobicyclic Ring Derivatives
US10538542B2 (en) * 2018-03-15 2020-01-21 Pfizer Inc. Cyclopentane-based modulators of STING (stimulator of interferon genes)

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