JPWO2021021717A5 - - Google Patents

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Publication number
JPWO2021021717A5
JPWO2021021717A5 JP2022505447A JP2022505447A JPWO2021021717A5 JP WO2021021717 A5 JPWO2021021717 A5 JP WO2021021717A5 JP 2022505447 A JP2022505447 A JP 2022505447A JP 2022505447 A JP2022505447 A JP 2022505447A JP WO2021021717 A5 JPWO2021021717 A5 JP WO2021021717A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
pharmaceutical composition
adenosine derivative
acceptable salt
tautomer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022505447A
Other languages
English (en)
Japanese (ja)
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JP2022541667A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/043713 external-priority patent/WO2021021717A1/en
Publication of JP2022541667A publication Critical patent/JP2022541667A/ja
Publication of JPWO2021021717A5 publication Critical patent/JPWO2021021717A5/ja
Pending legal-status Critical Current

Links

JP2022505447A 2019-07-27 2020-07-27 アデノシン誘導体及びそれを含む薬学的組成物 Pending JP2022541667A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962879414P 2019-07-27 2019-07-27
US62/879,414 2019-07-27
PCT/US2020/043713 WO2021021717A1 (en) 2019-07-27 2020-07-27 Adenosine derivative and pharmaceutical composition comprising the same

Publications (2)

Publication Number Publication Date
JP2022541667A JP2022541667A (ja) 2022-09-26
JPWO2021021717A5 true JPWO2021021717A5 (es) 2023-08-07

Family

ID=74229552

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022505447A Pending JP2022541667A (ja) 2019-07-27 2020-07-27 アデノシン誘導体及びそれを含む薬学的組成物

Country Status (12)

Country Link
US (2) US20220288098A1 (es)
EP (1) EP4003369A4 (es)
JP (1) JP2022541667A (es)
KR (1) KR20220068987A (es)
CN (1) CN114502175A (es)
AU (1) AU2020320876A1 (es)
BR (1) BR112022000965A2 (es)
CA (1) CA3146679A1 (es)
IL (1) IL289925A (es)
MX (1) MX2022000563A (es)
TW (1) TW202118496A (es)
WO (1) WO2021021717A1 (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117982682A (zh) 2017-07-11 2024-05-07 吉利德科学公司 用于治疗病毒感染的包含rna聚合酶抑制剂和环糊精的组合物
CN114929236B (zh) * 2019-09-11 2024-06-07 斯克里普斯研究所 抗病毒前药及其制剂
KR20220132608A (ko) 2020-01-27 2022-09-30 길리애드 사이언시즈, 인코포레이티드 SARS CoV-2 감염증을 치료하기 위한 방법
KR20220153619A (ko) 2020-03-12 2022-11-18 길리애드 사이언시즈, 인코포레이티드 1'-시아노 뉴클레오사이드의 제조 방법
WO2021188959A1 (en) 2020-03-20 2021-09-23 Gilead Sciences, Inc. Prodrugs of 4'-c-substituted-2-halo-2'-deoxyadenosine nucleosides and methods of making and using the same
US11701372B2 (en) 2020-04-06 2023-07-18 Gilead Sciences, Inc. Inhalation formulations of 1'-cyano substituted carba-nucleoside analogs
TW202203941A (zh) 2020-05-29 2022-02-01 美商基利科學股份有限公司 瑞德西韋之治療方法
MX2022016405A (es) 2020-06-24 2023-01-30 Gilead Sciences Inc Análogos de nucleósido de 1¿-ciano y usos de estos.
CR20230104A (es) 2020-08-27 2023-04-28 Gilead Sciences Inc Compuestos y métodos para el tratamiento de infecciones virales
MX2023008004A (es) 2021-01-25 2023-07-13 Brii Biosciences Inc Derivado de adenosina y composicion farmaceutica que lo comprende.
CA3204255A1 (en) * 2021-01-25 2022-07-28 Lianhong Xu Combination therapy for hiv with adenosine derivative and capsid inhibitors
IL307967A (en) * 2021-04-28 2023-12-01 Astrocyte Pharmaceuticals Inc Purine nucleosides, their intermediates and methods for their preparation
IL315102A (en) 2022-03-02 2024-10-01 Gilead Sciences Inc COMPOSITIONS AND METHODS FOR THE TREATMENT OF VIRAL INFECTIONS
WO2023196832A2 (en) * 2022-04-06 2023-10-12 Brii Biosciences, Inc. Pharmaceutical composition and method for treatment of human immunodeficiency virus infections
WO2024163262A2 (en) * 2023-01-30 2024-08-08 Merck Sharp & Dohme Llc Prodrugs of 4'-substituted nucleoside reverse transcriptase inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004271972B2 (en) * 2003-09-05 2010-06-03 Anadys Pharmaceuticals, Inc. TLR7 ligands for the treatment of hepatitis C
CA2502109C (en) * 2004-03-24 2010-02-23 Yamasa Corporation 4'-c-substituted-2-haloadenosine derivative
JP2009504677A (ja) * 2005-08-12 2009-02-05 メルク・エンド・カムパニー・インコーポレーテツド 新規2’−c−メチル及び4’−c−メチルヌクレオシド誘導体
WO2017053216A2 (en) * 2015-09-23 2017-03-30 Merck Sharp & Dohme Corp. 4'-substituted nucleoside reverse transcriptase inhibitors and preparations thereof
EP3844164A1 (en) * 2018-08-30 2021-07-07 GlaxoSmithKline Intellectual Property (No.2) Limited Compounds useful in hiv therapy

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