JPS59227888A - ７−フルオロプロスタグランジン類の製造方法 - Google Patents

７−フルオロプロスタグランジン類の製造方法

Info

Publication number
JPS59227888A
JPS59227888A JP58102885A JP10288583A JPS59227888A JP S59227888 A JPS59227888 A JP S59227888A JP 58102885 A JP58102885 A JP 58102885A JP 10288583 A JP10288583 A JP 10288583A JP S59227888 A JPS59227888 A JP S59227888A
Authority
JP
Japan
Prior art keywords
group
formula
compound
compound represented
protecting group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP58102885A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6343385B2 (enrdf_load_stackoverflow
Inventor
Arata Yasuda
新 安田
Masao Kato
正雄 加藤
Masaaki Yamabe
山辺　正顕
Keiichi Uchida
内田　啓一
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AGC Inc
Original Assignee
Asahi Glass Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asahi Glass Co Ltd filed Critical Asahi Glass Co Ltd
Priority to JP58102885A priority Critical patent/JPS59227888A/ja
Priority to PCT/JP1984/000294 priority patent/WO1984004917A1/ja
Priority to EP84902214A priority patent/EP0148953B1/en
Priority to DE8484902214T priority patent/DE3483314D1/de
Priority to US06/702,790 priority patent/US4699989A/en
Publication of JPS59227888A publication Critical patent/JPS59227888A/ja
Priority to US07/060,088 priority patent/US4822909A/en
Publication of JPS6343385B2 publication Critical patent/JPS6343385B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
    • C07D307/935—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
    • C07D307/937—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans with hydrocarbon or substituted hydrocarbon radicals directly attached in position 2, e.g. prostacyclins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP58102885A 1983-06-10 1983-06-10 ７−フルオロプロスタグランジン類の製造方法 Granted JPS59227888A (ja)

Priority Applications (6)

Application Number Priority Date Filing Date Title
JP58102885A JPS59227888A (ja) 1983-06-10 1983-06-10 ７−フルオロプロスタグランジン類の製造方法
PCT/JP1984/000294 WO1984004917A1 (en) 1983-06-10 1984-06-07 7-fluoroprostaglandins and process for their preparation
EP84902214A EP0148953B1 (en) 1983-06-10 1984-06-07 7-fluoroprostaglandins and process for their preparation
DE8484902214T DE3483314D1 (de) 1983-06-10 1984-06-07 7-fluorprostaglandine und deren herstellungsverfahren.
US06/702,790 US4699989A (en) 1983-06-10 1984-06-07 7-fluoroprostaglandins and process for their production
US07/060,088 US4822909A (en) 1983-06-10 1987-06-09 7-fluoroprostaglandins and process for their production

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP58102885A JPS59227888A (ja) 1983-06-10 1983-06-10 ７−フルオロプロスタグランジン類の製造方法

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP62323719A Division JPS63211292A (ja) 1987-12-23 1987-12-23 プロスタグランジン類

Publications (2)

Publication Number Publication Date
JPS59227888A true JPS59227888A (ja) 1984-12-21
JPS6343385B2 JPS6343385B2 (enrdf_load_stackoverflow) 1988-08-30

Family

ID=14339318

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58102885A Granted JPS59227888A (ja) 1983-06-10 1983-06-10 ７−フルオロプロスタグランジン類の製造方法

Country Status (5)

Country Link
US (1) US4699989A (enrdf_load_stackoverflow)
EP (1) EP0148953B1 (enrdf_load_stackoverflow)
JP (1) JPS59227888A (enrdf_load_stackoverflow)
DE (1) DE3483314D1 (enrdf_load_stackoverflow)
WO (1) WO1984004917A1 (enrdf_load_stackoverflow)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4634782A (en) * 1985-06-24 1987-01-06 Hoffmann-La Roche Inc. 7-fluoro-dihydro PGI compounds
US4680415A (en) * 1985-06-24 1987-07-14 Hoffmann-La Roche Inc. Intermediates for 7-fluoro dihydro PGI compounds
CH674363A5 (enrdf_load_stackoverflow) * 1986-12-01 1990-05-31 Hoffmann La Roche
US4808734A (en) * 1986-12-01 1989-02-28 Hoffmann-La Roche Inc. 16-cycloalkyl-7-fluoro-prostacyclins
JPH01102059A (ja) * 1987-10-16 1989-04-19 Asahi Glass Co Ltd ６−フルオロプロスタグランジン誘導体
US20110293549A1 (en) 2009-02-03 2011-12-01 Athena Cosmetics, Inc. Composition, method and kit for enhancing hair

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3997587A (en) * 1975-06-26 1976-12-14 Syntex (U.S.A.) Inc. D1- and 8R-9-fluoro-prostadienoic acid derivatives
JPS57165382A (en) * 1981-04-06 1982-10-12 Teijin Ltd Fluoro-pgi2 compound and its preparation
ZA821449B (en) * 1981-03-11 1983-01-26 Hoffmann La Roche Novel fluoro prostacyclins
US4634782A (en) * 1985-06-24 1987-01-06 Hoffmann-La Roche Inc. 7-fluoro-dihydro PGI compounds

Also Published As

Publication number Publication date
WO1984004917A1 (en) 1984-12-20
DE3483314D1 (de) 1990-10-31
EP0148953B1 (en) 1990-09-26
EP0148953A1 (en) 1985-07-24
US4699989A (en) 1987-10-13
EP0148953A4 (en) 1985-09-26
JPS6343385B2 (enrdf_load_stackoverflow) 1988-08-30

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