JPS59137470A - トリアゾ−ル系抗真菌剤 - Google Patents
トリアゾ−ル系抗真菌剤Info
- Publication number
- JPS59137470A JPS59137470A JP59008381A JP838184A JPS59137470A JP S59137470 A JPS59137470 A JP S59137470A JP 59008381 A JP59008381 A JP 59008381A JP 838184 A JP838184 A JP 838184A JP S59137470 A JPS59137470 A JP S59137470A
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- compound
- methyl
- represented
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/22—Tin compounds
- C07F7/2284—Compounds with one or more Sn-N linkages
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838301699A GB8301699D0 (en) | 1983-01-21 | 1983-01-21 | Antifungal agents |
| GB8301699 | 1983-01-21 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS59137470A true JPS59137470A (ja) | 1984-08-07 |
| JPS6346072B2 JPS6346072B2 (https=) | 1988-09-13 |
Family
ID=10536722
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP59008381A Granted JPS59137470A (ja) | 1983-01-21 | 1984-01-20 | トリアゾ−ル系抗真菌剤 |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0115400B1 (https=) |
| JP (1) | JPS59137470A (https=) |
| KR (1) | KR840007226A (https=) |
| AT (1) | ATE18766T1 (https=) |
| AU (1) | AU546388B2 (https=) |
| CA (1) | CA1226578A (https=) |
| DE (1) | DE3460055D1 (https=) |
| DK (1) | DK160091C (https=) |
| ES (1) | ES528984A0 (https=) |
| FI (1) | FI75811C (https=) |
| GB (1) | GB8301699D0 (https=) |
| GR (1) | GR79767B (https=) |
| IE (1) | IE56590B1 (https=) |
| IL (1) | IL70718A (https=) |
| PH (1) | PH19282A (https=) |
| PT (1) | PT77975B (https=) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6172767A (ja) * | 1984-09-05 | 1986-04-14 | インペリアル・ケミカル・インダストリーズ・ピーエルシー | 新規１，３―ジアゾリル―２―プロパノール誘導体、その製造法及び製薬学的又は獣医学的抗菌剤組成物 |
| JPS61215390A (ja) * | 1985-03-14 | 1986-09-25 | フアイザー・コーポレーシヨン | トリアゾール抗真菌剤 |
| JP2014517044A (ja) * | 2011-06-19 | 2014-07-17 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素阻害化合物 |
| JP2014523880A (ja) * | 2011-06-23 | 2014-09-18 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素化合物 |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU1313347A3 (ru) * | 1982-09-30 | 1987-05-23 | Пфайзер Корпорейшн (Фирма) | Способ получени производных триазола |
| EP0106515B1 (en) * | 1982-09-30 | 1988-12-28 | Pfizer Limited | Triazole anti-fungal agents |
| GB9002375D0 (en) * | 1990-02-02 | 1990-04-04 | Pfizer Ltd | Triazole antifungal agents |
| GB9107055D0 (en) * | 1991-04-04 | 1991-05-22 | Pfizer Ltd | Triazole antifungal agents |
| NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
| JP2005298333A (ja) * | 2001-11-15 | 2005-10-27 | Meiji Seika Kaisha Ltd | 新規トリアゾール誘導体及びこれを有効成分とする抗真菌剤 |
| CN111217795B (zh) * | 2020-02-14 | 2023-07-18 | 华侨大学 | 一种抗菌药物及其制备方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2078719B (en) * | 1980-06-02 | 1984-04-26 | Ici Ltd | Heterocyclic compounds |
-
1983
- 1983-01-21 GB GB838301699A patent/GB8301699D0/en active Pending
-
1984
- 1984-01-16 GR GR73516A patent/GR79767B/el unknown
- 1984-01-18 DE DE8484300285T patent/DE3460055D1/de not_active Expired
- 1984-01-18 EP EP84300285A patent/EP0115400B1/en not_active Expired
- 1984-01-18 AT AT84300285T patent/ATE18766T1/de not_active IP Right Cessation
- 1984-01-19 IL IL70718A patent/IL70718A/xx not_active IP Right Cessation
- 1984-01-19 CA CA000445636A patent/CA1226578A/en not_active Expired
- 1984-01-19 AU AU23592/84A patent/AU546388B2/en not_active Ceased
- 1984-01-19 PT PT77975A patent/PT77975B/pt not_active IP Right Cessation
- 1984-01-19 ES ES528984A patent/ES528984A0/es active Granted
- 1984-01-20 KR KR1019840000242A patent/KR840007226A/ko not_active Ceased
- 1984-01-20 JP JP59008381A patent/JPS59137470A/ja active Granted
- 1984-01-20 IE IE134/84A patent/IE56590B1/en not_active IP Right Cessation
- 1984-01-20 FI FI840237A patent/FI75811C/fi not_active IP Right Cessation
- 1984-01-20 DK DK024884A patent/DK160091C/da active
- 1984-01-23 PH PH30146A patent/PH19282A/en unknown
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6172767A (ja) * | 1984-09-05 | 1986-04-14 | インペリアル・ケミカル・インダストリーズ・ピーエルシー | 新規１，３―ジアゾリル―２―プロパノール誘導体、その製造法及び製薬学的又は獣医学的抗菌剤組成物 |
| JPS61215390A (ja) * | 1985-03-14 | 1986-09-25 | フアイザー・コーポレーシヨン | トリアゾール抗真菌剤 |
| JP2014517044A (ja) * | 2011-06-19 | 2014-07-17 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素阻害化合物 |
| JP2014518219A (ja) * | 2011-06-19 | 2014-07-28 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素阻害剤化合物 |
| US9556143B2 (en) | 2011-06-19 | 2017-01-31 | Viamet Pharmaceuticals, Inc. | Metalloenzyme inhibitor compounds |
| JP2014523880A (ja) * | 2011-06-23 | 2014-09-18 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素化合物 |
| JP2017101027A (ja) * | 2011-06-23 | 2017-06-08 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| IL70718A (en) | 1986-09-30 |
| KR840007226A (ko) | 1984-12-06 |
| FI840237A0 (fi) | 1984-01-20 |
| GB8301699D0 (en) | 1983-02-23 |
| IE56590B1 (en) | 1991-10-09 |
| DK160091C (da) | 1991-06-24 |
| PT77975B (en) | 1986-06-18 |
| GR79767B (https=) | 1984-10-31 |
| IL70718A0 (en) | 1984-04-30 |
| FI840237L (fi) | 1984-07-22 |
| AU546388B2 (en) | 1985-08-29 |
| ES8506000A1 (es) | 1985-06-16 |
| DK160091B (da) | 1991-01-28 |
| ATE18766T1 (de) | 1986-04-15 |
| DK24884D0 (da) | 1984-01-20 |
| CA1226578A (en) | 1987-09-08 |
| DE3460055D1 (en) | 1986-04-30 |
| EP0115400A1 (en) | 1984-08-08 |
| EP0115400B1 (en) | 1986-03-26 |
| AU2359284A (en) | 1984-07-26 |
| PT77975A (en) | 1984-02-01 |
| PH19282A (en) | 1986-03-04 |
| DK24884A (da) | 1984-07-22 |
| FI75811B (fi) | 1988-04-29 |
| IE840134L (en) | 1984-07-21 |
| JPS6346072B2 (https=) | 1988-09-13 |
| FI75811C (fi) | 1988-08-08 |
| ES528984A0 (es) | 1985-06-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU602638B2 (en) | Triazole antifungal agents | |
| AU688455B2 (en) | Watersoluble azole antifungals | |
| US4482558A (en) | Antifungal amide and urea derivatives of (3-amino-2-aryl-2-hydroxyprop-1-yl)-1H-1,2,4-triazoles | |
| CA1056380A (en) | Process for preparation of novel imidazole derivatives | |
| JPS59137470A (ja) | トリアゾ−ル系抗真菌剤 | |
| US4483863A (en) | Triazole antifungal agents | |
| IE55233B1 (en) | Triazole antifungal agents | |
| IE56055B1 (en) | Triazole antifungal agents | |
| JPH01190672A (ja) | トリアゾール抗真菌剤 | |
| US4678789A (en) | Triazole antifungal agents | |
| DK159205B (da) | Bis(triazol)alkanol-forbindelser, anvendelse af disse, farmaceutiske praeparater og landbrugsfungicider indeholdende disse og fremgangsmaade til behandling af planter eller froe, som har en svampeinfektion | |
| US5047548A (en) | 3-aryl-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butyramide and derivatives as antifungal agents | |
| US4737508A (en) | 1-aryl-1-(1H-azol-1-ylalkyl)-1,3-dihydroisobenzofurans, related derivatives and pharmaceutical compositions thereof useful as antifungals | |
| JPS59176266A (ja) | トリアゾ−ル系抗真菌薬 | |
| DK157998B (da) | 1-(1,2,4-triazol-1-yl)-3-(5-trifluormethylimidazol-1-yl)propan-2-ol-forbindelser og farmaceutisk og landbrugsmaessigt acceptable salte deraf samt farmaceutisk praeparat og landbrugsfungicid indeholdende disse | |
| FI83777B (fi) | Foerfarande foer framstaellning av terapeutiskt anvaendbara 1-aryl-1-(fluorhydroxialkyl eller perfluoralkanoyl)-2-(1h-1,2,4-triazol-1-yl) etanoler. | |
| EP0102727B1 (en) | Chloropyridyl antifungal agents | |
| US5206364A (en) | Triazole antifungal agents | |
| US4877801A (en) | 1-Aryl-1-(1H-azol-1-ylalkyl)-1,3-dihydroisobenzofurans, related derivatives and pharmaceutical compositions thereof useful as antifungals | |
| JPS6345676B2 (https=) | ||
| IL106262A (en) | Intermediates to triazole antifungal agents |