JPS5791998A - Novel 5'-o-acylnucleoside derivative and its preparation - Google Patents

Novel 5'-o-acylnucleoside derivative and its preparation

Info

Publication number
JPS5791998A
JPS5791998A JP56080231A JP8023181A JPS5791998A JP S5791998 A JPS5791998 A JP S5791998A JP 56080231 A JP56080231 A JP 56080231A JP 8023181 A JP8023181 A JP 8023181A JP S5791998 A JPS5791998 A JP S5791998A
Authority
JP
Japan
Prior art keywords
derivative
expressed
acyl group
formula
aminocarboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP56080231A
Other languages
English (en)
Inventor
Takeshi Endo
Katsumi Sakai
Kiyoaki Cho
Yoshitaka Inamoto
Haruhiko Teshigahara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fuji Chemical Industries Co Ltd
Original Assignee
Fuji Chemical Industries Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/210,796 external-priority patent/US4340728A/en
Application filed by Fuji Chemical Industries Co Ltd filed Critical Fuji Chemical Industries Co Ltd
Publication of JPS5791998A publication Critical patent/JPS5791998A/ja
Pending legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP56080231A 1980-11-26 1981-05-28 Novel 5'-o-acylnucleoside derivative and its preparation Pending JPS5791998A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/210,796 US4340728A (en) 1979-11-28 1980-11-26 Nucleoside derivatives and process for preparing same

Publications (1)

Publication Number Publication Date
JPS5791998A true JPS5791998A (en) 1982-06-08

Family

ID=22784293

Family Applications (5)

Application Number Title Priority Date Filing Date
JP56079434A Pending JPS5791994A (en) 1980-11-26 1981-05-27 5'-o-(n-alkylcarbamoylalanyl)-5-fluorouridine and its preparation
JP56080231A Pending JPS5791998A (en) 1980-11-26 1981-05-28 Novel 5'-o-acylnucleoside derivative and its preparation
JP56080228A Pending JPS5791995A (en) 1980-11-26 1981-05-28 Nucleoside-5'-o-morpholinoacyl ester and its preparation
JP56080229A Granted JPS5791996A (en) 1980-11-26 1981-05-28 Novel nucleoside derivative and its preparation
JP56080230A Granted JPS5791997A (en) 1980-11-26 1981-05-28 5'-o-acylnucleoside and its preparation

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP56079434A Pending JPS5791994A (en) 1980-11-26 1981-05-27 5'-o-(n-alkylcarbamoylalanyl)-5-fluorouridine and its preparation

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP56080228A Pending JPS5791995A (en) 1980-11-26 1981-05-28 Nucleoside-5'-o-morpholinoacyl ester and its preparation
JP56080229A Granted JPS5791996A (en) 1980-11-26 1981-05-28 Novel nucleoside derivative and its preparation
JP56080230A Granted JPS5791997A (en) 1980-11-26 1981-05-28 5'-o-acylnucleoside and its preparation

Country Status (1)

Country Link
JP (5) JPS5791994A (ja)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0301873A2 (en) * 1987-07-31 1989-02-01 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US4892939A (en) * 1986-05-30 1990-01-09 Fuji Kagaku Kogyo Kabushiki Kaisha Oligopeptidyl-5-fluorouridine compounds and process for preparing the same
US5783689A (en) * 1996-11-12 1998-07-21 University Of Notre Dame Antibacterial and antifungal nucleosides
US5808049A (en) * 1994-05-20 1998-09-15 Director-General Of Agency Of Industrial Science And Technology Stereospecific 5-fu esters and methods for preparing same

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5925327A (ja) * 1982-07-31 1984-02-09 Hidematsu Hirai 抗腫瘍性複合体の製造方法
JPS61134397A (ja) * 1984-12-01 1986-06-21 Fuji Kagaku Kogyo Kk ５’−０−オリゴペプチジル−５−フルオロウリジン及びその製造方法
JP2575372B2 (ja) * 1987-02-12 1997-01-22 三井東圧化学株式会社 制ガン剤
US6020322A (en) 1993-11-09 2000-02-01 Pro-Neuron, Inc. Acyl deoxyribonucleoside derivatives and uses thereof
DE3855513T2 (de) * 1987-10-28 1997-01-09 Pro Neuron Inc Acyl deoxyribonukleosid-derivate und deren verwendungen
US5470838A (en) 1987-10-28 1995-11-28 Pro-Neuron, Inc. Method of delivering exogenous uridine or cytidine using acylated uridine or cytidine
JP2894610B2 (ja) * 1987-10-28 1999-05-24 プロ−ニューロン，インコーポレーテッド アシル化ウリジンおよびシチジンならびにその使用
JP2631227B2 (ja) * 1988-07-11 1997-07-16 大鵬薬品工業株式会社 ５´−ベンジル−５−フルオロウリジン誘導体及びその中間体
US7169765B1 (en) 1988-10-27 2007-01-30 Wellstat Therapeutics Corporation Acyl deoxyribonucleoside derivatives and uses thereof
WO1991012259A1 (en) * 1990-02-08 1991-08-22 Sankyo Company, Limited 5-fu derivative

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4892939A (en) * 1986-05-30 1990-01-09 Fuji Kagaku Kogyo Kabushiki Kaisha Oligopeptidyl-5-fluorouridine compounds and process for preparing the same
EP0301873A2 (en) * 1987-07-31 1989-02-01 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US4946951A (en) * 1987-07-31 1990-08-07 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US5808049A (en) * 1994-05-20 1998-09-15 Director-General Of Agency Of Industrial Science And Technology Stereospecific 5-fu esters and methods for preparing same
US5783689A (en) * 1996-11-12 1998-07-21 University Of Notre Dame Antibacterial and antifungal nucleosides

Also Published As

Publication number Publication date
JPS5791996A (en) 1982-06-08
JPS6247196B2 (ja) 1987-10-06
JPS6247198B2 (ja) 1987-10-06
JPS5791997A (en) 1982-06-08
JPS5791995A (en) 1982-06-08
JPS5791994A (en) 1982-06-08

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