JPS57176988A - Penam-3-carboxylic acid derivative and its preparation - Google Patents
Penam-3-carboxylic acid derivative and its preparationInfo
- Publication number
- JPS57176988A JPS57176988A JP56053694A JP5369481A JPS57176988A JP S57176988 A JPS57176988 A JP S57176988A JP 56053694 A JP56053694 A JP 56053694A JP 5369481 A JP5369481 A JP 5369481A JP S57176988 A JPS57176988 A JP S57176988A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- amino
- protecting group
- compound shown
- penam
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP56053694A JPS57176988A (en) | 1981-04-09 | 1981-04-09 | Penam-3-carboxylic acid derivative and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP56053694A JPS57176988A (en) | 1981-04-09 | 1981-04-09 | Penam-3-carboxylic acid derivative and its preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS57176988A true JPS57176988A (en) | 1982-10-30 |
JPH03395B2 JPH03395B2 (ja) | 1991-01-07 |
Family
ID=12949912
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP56053694A Granted JPS57176988A (en) | 1981-04-09 | 1981-04-09 | Penam-3-carboxylic acid derivative and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS57176988A (ja) |
Cited By (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5813588A (ja) * | 1981-07-15 | 1983-01-26 | Sumitomo Chem Co Ltd | 新規なβ−ラクタム化合物及びその製造法 |
JPS59139386A (ja) * | 1983-01-25 | 1984-08-10 | メルク エンド カムパニー インコーポレーテツド | 2―置換アルケニルチオ―ペン―2―エム3―カルボキシル酸 |
JPS6016990A (ja) * | 1983-06-21 | 1985-01-28 | フアイザ−・インコ−ポレ−テツド | 2−アルキルチオペネム誘導体 |
US4504485A (en) * | 1983-04-04 | 1985-03-12 | Schering Corporation | 5R,6S,8R-6-(1-Hydroxyethyl)-2-(2-carbamoyloxyethylthio)-penem-3-carboxylic acid |
JPS60120881A (ja) * | 1983-10-14 | 1985-06-28 | フアイザ−・インコ−ポレ−テツド | 2−アザシクロアルキルチオペネム誘導体 |
US4595539A (en) * | 1983-06-10 | 1986-06-17 | Pfizer Inc. | Preparation of penem derivatives and azetidinone intermediates |
US4613595A (en) * | 1982-05-14 | 1986-09-23 | Sankyo Company Limited | Penem derivatives, and composition containing them |
US4614738A (en) * | 1983-03-25 | 1986-09-30 | Schering Corporation | 2-(N-heterocycloaliphaticthio)penems |
JPS61236785A (ja) * | 1985-04-15 | 1986-10-22 | Sankyo Co Ltd | アゼチジノン誘導体 |
US4619783A (en) * | 1983-06-10 | 1986-10-28 | Pfizer Inc. | Process and intermediates for the preparation of penem derivatives |
US4725678A (en) * | 1983-06-10 | 1988-02-16 | Pfizer Inc. | Azetidinone intermediates for the preparation of penem derivatives |
JPS6341481A (ja) * | 1986-07-29 | 1988-02-22 | フアイザ−・インコ−ポレ−テツド | ペネム類の合成方法 |
US4933333A (en) * | 1983-05-09 | 1990-06-12 | Sumitomo Pharmaceuticals Co., Ltd. | β-lactam compounds |
CN110062760A (zh) * | 2016-10-10 | 2019-07-26 | 约翰霍普金斯大学 | 抗d,d-转肽酶和l,d-转肽酶的抗细菌剂 |
-
1981
- 1981-04-09 JP JP56053694A patent/JPS57176988A/ja active Granted
Cited By (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5813588A (ja) * | 1981-07-15 | 1983-01-26 | Sumitomo Chem Co Ltd | 新規なβ−ラクタム化合物及びその製造法 |
US4613595A (en) * | 1982-05-14 | 1986-09-23 | Sankyo Company Limited | Penem derivatives, and composition containing them |
JPS59139386A (ja) * | 1983-01-25 | 1984-08-10 | メルク エンド カムパニー インコーポレーテツド | 2―置換アルケニルチオ―ペン―2―エム3―カルボキシル酸 |
JPH0516433B2 (ja) * | 1983-01-25 | 1993-03-04 | Merck & Co Inc | |
US4614738A (en) * | 1983-03-25 | 1986-09-30 | Schering Corporation | 2-(N-heterocycloaliphaticthio)penems |
US4504485A (en) * | 1983-04-04 | 1985-03-12 | Schering Corporation | 5R,6S,8R-6-(1-Hydroxyethyl)-2-(2-carbamoyloxyethylthio)-penem-3-carboxylic acid |
US4933333A (en) * | 1983-05-09 | 1990-06-12 | Sumitomo Pharmaceuticals Co., Ltd. | β-lactam compounds |
US4595539A (en) * | 1983-06-10 | 1986-06-17 | Pfizer Inc. | Preparation of penem derivatives and azetidinone intermediates |
US4619783A (en) * | 1983-06-10 | 1986-10-28 | Pfizer Inc. | Process and intermediates for the preparation of penem derivatives |
US4725678A (en) * | 1983-06-10 | 1988-02-16 | Pfizer Inc. | Azetidinone intermediates for the preparation of penem derivatives |
JPS6016990A (ja) * | 1983-06-21 | 1985-01-28 | フアイザ−・インコ−ポレ−テツド | 2−アルキルチオペネム誘導体 |
JPH0528237B2 (ja) * | 1983-06-21 | 1993-04-23 | Pfizer | |
JPS60120881A (ja) * | 1983-10-14 | 1985-06-28 | フアイザ−・インコ−ポレ−テツド | 2−アザシクロアルキルチオペネム誘導体 |
JPS61236785A (ja) * | 1985-04-15 | 1986-10-22 | Sankyo Co Ltd | アゼチジノン誘導体 |
JPH0572396B2 (ja) * | 1985-04-15 | 1993-10-12 | Sankyo Co | |
JPS6341481A (ja) * | 1986-07-29 | 1988-02-22 | フアイザ−・インコ−ポレ−テツド | ペネム類の合成方法 |
CN110062760A (zh) * | 2016-10-10 | 2019-07-26 | 约翰霍普金斯大学 | 抗d,d-转肽酶和l,d-转肽酶的抗细菌剂 |
EP3523309A4 (en) * | 2016-10-10 | 2020-07-22 | The Johns Hopkins University | ANTIBACTERIAL AGENTS AGAINST D, D- AND L, D-TRANSPEPTIDASES |
US11084833B2 (en) | 2016-10-10 | 2021-08-10 | The Johns Hopkins University | Antibacterial agents against D,D- and L,D-transpeptidases |
Also Published As
Publication number | Publication date |
---|---|
JPH03395B2 (ja) | 1991-01-07 |
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