JPS5587748A - Preparation of o-(2,6-dichloroanilino)phenylacetic acid - Google Patents
Preparation of o-(2,6-dichloroanilino)phenylacetic acidInfo
- Publication number
- JPS5587748A JPS5587748A JP16269878A JP16269878A JPS5587748A JP S5587748 A JPS5587748 A JP S5587748A JP 16269878 A JP16269878 A JP 16269878A JP 16269878 A JP16269878 A JP 16269878A JP S5587748 A JPS5587748 A JP S5587748A
- Authority
- JP
- Japan
- Prior art keywords
- dichloroanilino
- formula
- dialkyl
- base
- phenylacetic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PURPOSE: To prepare the title compound useful as an antiphlogistic agent, easily, with a few steps, by hydrolyzing an N,N-dialkyl-[o-(2,6-dichloroanilino)phenyl] acetamide derivative in the presence of a base.
CONSTITUTION: o-(2,6-Dichloroanilino)phenylacetic acid of formula II is prepared by hydrolyzing an N,N-dialkyl-[o-(2,6-dichloroanilino)-phenylacetamide derivative of formula I (R1,2 are lower alkyl) in a solvent such as ethanol, in the presence of a base such as KOH, at the refluxing temperature of the solvent. The amount of the base is pref. 10W20mol per 1mol of the acetamide derivative. The compound of formula I can be prepared by reacting an N,N-dialkyl-(o-halogenophenyl)acetamide derivative of formula III (X is Br or I) with 2,6-dichloroaniline of formula IV in the presence of a copper catalyst.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP16269878A JPS5587748A (en) | 1978-12-26 | 1978-12-26 | Preparation of o-(2,6-dichloroanilino)phenylacetic acid |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP16269878A JPS5587748A (en) | 1978-12-26 | 1978-12-26 | Preparation of o-(2,6-dichloroanilino)phenylacetic acid |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5587748A true JPS5587748A (en) | 1980-07-02 |
Family
ID=15759592
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP16269878A Pending JPS5587748A (en) | 1978-12-26 | 1978-12-26 | Preparation of o-(2,6-dichloroanilino)phenylacetic acid |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5587748A (en) |
-
1978
- 1978-12-26 JP JP16269878A patent/JPS5587748A/en active Pending
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