JPS54138554A - Indole derivative - Google Patents

Indole derivative

Info

Publication number
JPS54138554A
JPS54138554A JP4420078A JP4420078A JPS54138554A JP S54138554 A JPS54138554 A JP S54138554A JP 4420078 A JP4420078 A JP 4420078A JP 4420078 A JP4420078 A JP 4420078A JP S54138554 A JPS54138554 A JP S54138554A
Authority
JP
Japan
Prior art keywords
formula
reacted
alkyl
compound
indole derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP4420078A
Other languages
Japanese (ja)
Inventor
Toshio Wakabayashi
Kenzo Watanabe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teijin Ltd
Original Assignee
Teijin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Ltd filed Critical Teijin Ltd
Priority to JP4420078A priority Critical patent/JPS54138554A/en
Publication of JPS54138554A publication Critical patent/JPS54138554A/en
Pending legal-status Critical Current

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  • Indole Compounds (AREA)

Abstract

NEW MATERIAL:A compound of formula I: (R1 is monofunctional substituent, halogen, alkoxy group, etc.; m is 0, 1, or 2; (R1)m is H when m is 0, and two R1's may form a ring when m is 2; R2 is H, CH3, or C2H5; R3 is H, alkyl, phenyl, benzyl group, etc,; R4 is H or alkyl group).
EXAMPLE: 2-Carbamoyl-3-indoleacetic acid.
USE: Intermediates for antiphlogistics, antithrombotics, psychotropic drugs, etc.
PROCESS: An acid anhydride of formula II is reacted with the corresponding sodium alkoxide or potassium alkoxide to form a reaction product, which is reacted with an amine of formula III in the presence of a condensing agent, e.g. dicyclohexylcarbodiimide, and, if necessary, hydrolyzed to form the objective compound of formula I.
COPYRIGHT: (C)1979,JPO&Japio
JP4420078A 1978-04-17 1978-04-17 Indole derivative Pending JPS54138554A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP4420078A JPS54138554A (en) 1978-04-17 1978-04-17 Indole derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP4420078A JPS54138554A (en) 1978-04-17 1978-04-17 Indole derivative

Publications (1)

Publication Number Publication Date
JPS54138554A true JPS54138554A (en) 1979-10-27

Family

ID=12684921

Family Applications (1)

Application Number Title Priority Date Filing Date
JP4420078A Pending JPS54138554A (en) 1978-04-17 1978-04-17 Indole derivative

Country Status (1)

Country Link
JP (1) JPS54138554A (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100466522B1 (en) * 2002-08-03 2005-01-15 대한민국(관리부서:농촌진흥청) Extracts of Paecilomyces sp. J300 having antitumor activity and pharmaceutical composition containing the same

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100466522B1 (en) * 2002-08-03 2005-01-15 대한민국(관리부서:농촌진흥청) Extracts of Paecilomyces sp. J300 having antitumor activity and pharmaceutical composition containing the same

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