JPS54128599A - Pyrrolobenzazepin derivative - Google Patents
Pyrrolobenzazepin derivativeInfo
- Publication number
- JPS54128599A JPS54128599A JP3482978A JP3482978A JPS54128599A JP S54128599 A JPS54128599 A JP S54128599A JP 3482978 A JP3482978 A JP 3482978A JP 3482978 A JP3482978 A JP 3482978A JP S54128599 A JPS54128599 A JP S54128599A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- pyrrolobenzazepin
- derivative
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Abstract
NEW MATERIAL:A pyrrolobenzazepin derivative of formula I: (R1 is 1W6C alkyl, 1W6C alkoxy, OH, or carboxylate of COR1; R2 is H or 1W6C alkyl; R3 is 1W6C alkyl, 1W6C alkoxy, 1W6C alkyl-thio, H, F, Cl, Br, or trifluoromethyl group; n is 0 or 1).
EXAMPLE: 2-(1,1-Oxo-6,11-dihydro-5H-pyrrolo[2,1-b][3]benzazebin-2-yl)-propionic acid.
USE: Medicines, e.g. antiphlogistics, analogesics, and antithrombotics.
PROCESS: A substituted pyrrole-carboxylic acid chlride of formula II is converted into the compound of formula I via cyclization and exchange reaction of side chains.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3482978A JPS54128599A (en) | 1978-03-28 | 1978-03-28 | Pyrrolobenzazepin derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3482978A JPS54128599A (en) | 1978-03-28 | 1978-03-28 | Pyrrolobenzazepin derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS54128599A true JPS54128599A (en) | 1979-10-05 |
Family
ID=12425077
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP3482978A Pending JPS54128599A (en) | 1978-03-28 | 1978-03-28 | Pyrrolobenzazepin derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS54128599A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110357894A (en) * | 2019-08-22 | 2019-10-22 | 云南省烟草农业科学研究院 | A kind of tricyclic alkaloid compound and the preparation method and application thereof |
CN110372707A (en) * | 2019-08-22 | 2019-10-25 | 云南省烟草农业科学研究院 | Miscellaneous tall and erect alkaloid compound of a kind of benzo and the preparation method and application thereof |
-
1978
- 1978-03-28 JP JP3482978A patent/JPS54128599A/en active Pending
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110357894A (en) * | 2019-08-22 | 2019-10-22 | 云南省烟草农业科学研究院 | A kind of tricyclic alkaloid compound and the preparation method and application thereof |
CN110372707A (en) * | 2019-08-22 | 2019-10-25 | 云南省烟草农业科学研究院 | Miscellaneous tall and erect alkaloid compound of a kind of benzo and the preparation method and application thereof |
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