JPS55115887A - 7beta-(4-lower alkylimino-1,3-dithietane-2-yl)carboxamide-3- (1-lower alkyltetrazol-5-yl)thiomethyl-delta3-cephem-4- carboxylic acid - Google Patents
7beta-(4-lower alkylimino-1,3-dithietane-2-yl)carboxamide-3- (1-lower alkyltetrazol-5-yl)thiomethyl-delta3-cephem-4- carboxylic acidInfo
- Publication number
- JPS55115887A JPS55115887A JP2396779A JP2396779A JPS55115887A JP S55115887 A JPS55115887 A JP S55115887A JP 2396779 A JP2396779 A JP 2396779A JP 2396779 A JP2396779 A JP 2396779A JP S55115887 A JPS55115887 A JP S55115887A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound shown
- cephem
- thiomethyl
- carboxamide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:The title compound shown by the formula I (R is lower alkyl; R1 is H or lower alkoxy; R2 is lower alkyl) and its salt.
EXAMPLE: 7β-( 4-Methylimino-1, 3-dithethane-2-yl )carboxamide-7α-methoxy-3-(1- methyltetrazol-5-yl) thiomethyl-Δ3-cephem-4-carboxylic acid.
USE: An antibacterial substance.
PROCESS: A compound shown by the formula II (X is halogen) is reacted with a compound shown by the formula III (Me is alkali metal) to give the desired compound shown by the formula I. A compound shown by the formula IV (R3 is H or carboxyl-protecting group) is reacted with a compound shown by the formula V or its reactive derivative to give the desired compound shown by the formula I. After the reaction, when R3 is the protecting group, it is removed to give the desired compound.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2396779A JPS55115887A (en) | 1979-02-28 | 1979-02-28 | 7beta-(4-lower alkylimino-1,3-dithietane-2-yl)carboxamide-3- (1-lower alkyltetrazol-5-yl)thiomethyl-delta3-cephem-4- carboxylic acid |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2396779A JPS55115887A (en) | 1979-02-28 | 1979-02-28 | 7beta-(4-lower alkylimino-1,3-dithietane-2-yl)carboxamide-3- (1-lower alkyltetrazol-5-yl)thiomethyl-delta3-cephem-4- carboxylic acid |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS55115887A true JPS55115887A (en) | 1980-09-06 |
Family
ID=12125313
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2396779A Pending JPS55115887A (en) | 1979-02-28 | 1979-02-28 | 7beta-(4-lower alkylimino-1,3-dithietane-2-yl)carboxamide-3- (1-lower alkyltetrazol-5-yl)thiomethyl-delta3-cephem-4- carboxylic acid |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55115887A (en) |
-
1979
- 1979-02-28 JP JP2396779A patent/JPS55115887A/en active Pending
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