JPS5721387A - Preparation of oxazolidinone derivative - Google Patents
Preparation of oxazolidinone derivativeInfo
- Publication number
- JPS5721387A JPS5721387A JP9383980A JP9383980A JPS5721387A JP S5721387 A JPS5721387 A JP S5721387A JP 9383980 A JP9383980 A JP 9383980A JP 9383980 A JP9383980 A JP 9383980A JP S5721387 A JPS5721387 A JP S5721387A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- alkyl
- reaction product
- oxazolidinone derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
Abstract
PURPOSE: To obtain an oxazolidinone derivative useful as a synthetic intermediate for medicines in high yield, by reacting specific compounds, and reducing the reaction product.
CONSTITUTION: A compound of formula I (R is alkyl) is reacted with a compound of formula II (R1 is alkyl, aryl or aralkyl; X is halogen) in the presence of a solvent, e.g. a hydrocarbon, at a temperature of the boiling point of the reaction mixture or below for several hours to 24hr, and the reaction product is then reduced catalytically or with a reducing agent by the conventional method to give the aimed compound of formula III.
USE: 4-(2-Hydroxy-3-alkylaminopropoxy)indole obtained by hydrolyzing the aimed compound has β-adrenergic neuroplegic action and is useful for the prevention and the remedy of arrhythmia, etc.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9383980A JPS5721387A (en) | 1980-07-11 | 1980-07-11 | Preparation of oxazolidinone derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9383980A JPS5721387A (en) | 1980-07-11 | 1980-07-11 | Preparation of oxazolidinone derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5721387A true JPS5721387A (en) | 1982-02-04 |
Family
ID=14093554
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP9383980A Pending JPS5721387A (en) | 1980-07-11 | 1980-07-11 | Preparation of oxazolidinone derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5721387A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59158691A (en) * | 1983-03-01 | 1984-09-08 | Canon Inc | Image pickup device |
-
1980
- 1980-07-11 JP JP9383980A patent/JPS5721387A/en active Pending
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59158691A (en) * | 1983-03-01 | 1984-09-08 | Canon Inc | Image pickup device |
JPH05914B2 (en) * | 1983-03-01 | 1993-01-07 | Canon Kk |
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