JPS54112881A - Preparation of 2-mercaptopyrimidine hydrochloride - Google Patents
Preparation of 2-mercaptopyrimidine hydrochlorideInfo
- Publication number
- JPS54112881A JPS54112881A JP1919778A JP1919778A JPS54112881A JP S54112881 A JPS54112881 A JP S54112881A JP 1919778 A JP1919778 A JP 1919778A JP 1919778 A JP1919778 A JP 1919778A JP S54112881 A JPS54112881 A JP S54112881A
- Authority
- JP
- Japan
- Prior art keywords
- hcl gas
- mercaptopyrimidine
- hydrochloride
- pref
- thiourea
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PURPOSE: To prepare the title compound, useful as an amino acid protector, continuously, in high yield, by reacting a β-dicarbonyl compound and thiourea with HCl gas in water, crystallizing the reaction product, and recycling the filtrate as the solvent of the reaction system.
CONSTITUTION: 2-Mercaptopyrimidine hydrochloride of formula II (R1,2 are H, 1-4C lower alkyl) is prepared by (1) introducing HCl gas into an aqueous solvent containing 0.8W1.5 moles of a β-dicarbonyl compound of formula I and 1 mole of thiourea at ≥65°C, pref. 70W95°C for ≥15 min., (2) crystallizing the reaction product by cooling the solution, and (3) filtering the crystals. The reaction is pref. performed continuously, by introducing and absorbing the HCl gas into the filtrate.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1919778A JPS6058913B2 (en) | 1978-02-22 | 1978-02-22 | Method for producing 2-mercaptopyrimidine hydrochloride |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1919778A JPS6058913B2 (en) | 1978-02-22 | 1978-02-22 | Method for producing 2-mercaptopyrimidine hydrochloride |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS54112881A true JPS54112881A (en) | 1979-09-04 |
JPS6058913B2 JPS6058913B2 (en) | 1985-12-23 |
Family
ID=11992617
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP1919778A Expired JPS6058913B2 (en) | 1978-02-22 | 1978-02-22 | Method for producing 2-mercaptopyrimidine hydrochloride |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6058913B2 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS55157572A (en) * | 1979-05-25 | 1980-12-08 | Nitto Boseki Co Ltd | Preparation of 2-mercapto-4,6-dimethylpyrimidine hydrochloride |
-
1978
- 1978-02-22 JP JP1919778A patent/JPS6058913B2/en not_active Expired
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS55157572A (en) * | 1979-05-25 | 1980-12-08 | Nitto Boseki Co Ltd | Preparation of 2-mercapto-4,6-dimethylpyrimidine hydrochloride |
JPS6144870B2 (en) * | 1979-05-25 | 1986-10-04 | Nitto Boseki Co Ltd |
Also Published As
Publication number | Publication date |
---|---|
JPS6058913B2 (en) | 1985-12-23 |
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