JPS54103890A - Novel antibacteral compound - Google Patents

Novel antibacteral compound

Info

Publication number
JPS54103890A
JPS54103890A JP1077278A JP1077278A JPS54103890A JP S54103890 A JPS54103890 A JP S54103890A JP 1077278 A JP1077278 A JP 1077278A JP 1077278 A JP1077278 A JP 1077278A JP S54103890 A JPS54103890 A JP S54103890A
Authority
JP
Japan
Prior art keywords
formula
compound
group
carboxyl
iii
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1077278A
Other languages
English (en)
Other versions
JPS6052714B2 (ja
Inventor
Masaru Iwanami
Kensho Nagano
Yoshinobu Nagano
Masaharu Fujiki
Tetsuya Maeda
Atsuki Yamazaki
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yamanouchi Pharmaceutical Co Ltd
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Priority to JP53010772A priority Critical patent/JPS6052714B2/ja
Priority to GB25353/78A priority patent/GB1604739A/en
Priority to GB25352/78A priority patent/GB1604738A/en
Priority to DE2824575A priority patent/DE2824575C2/de
Priority to CH610878A priority patent/CH636098A5/de
Priority to CH6107/78A priority patent/CH648317A5/de
Priority to DE2824559A priority patent/DE2824559C2/de
Priority to US05/913,500 priority patent/US4263432A/en
Priority to NLAANVRAGE7806208,A priority patent/NL185622C/xx
Priority to US05/913,501 priority patent/US4198339A/en
Priority to CA305,045A priority patent/CA1103659A/en
Priority to HU78JA822A priority patent/HU178584B/hu
Priority to SU782627106A priority patent/SU818486A3/ru
Priority to DK258078A priority patent/DK164224C/da
Priority to FR7817304A priority patent/FR2398745A1/fr
Priority to AT421978A priority patent/AT360650B/de
Priority to SE7806711A priority patent/SE438338B/sv
Priority to ES470689A priority patent/ES470689A1/es
Priority to FR7817303A priority patent/FR2405952A1/fr
Priority to UA2627106A priority patent/UA5923A1/uk
Priority to IT68369/78A priority patent/IT1159721B/it
Priority to MX1051378U priority patent/MX7170E/es
Priority to MX787141U priority patent/MX5137E/es
Priority to MX1051478U priority patent/MX7171E/es
Priority to IT68370/78A priority patent/IT1109095B/it
Priority to ES479166A priority patent/ES479166A1/es
Priority to ES479168A priority patent/ES479168A1/es
Priority to ES479167A priority patent/ES479167A1/es
Publication of JPS54103890A publication Critical patent/JPS54103890A/ja
Priority to SU792805308A priority patent/SU1024010A3/ru
Priority to AT685879A priority patent/AT361626B/de
Priority to US06/208,298 priority patent/US4404373A/en
Priority to US06/304,986 priority patent/US4414153A/en
Priority to KE3489A priority patent/KE3489A/xx
Priority to US06/727,233 priority patent/USRE32491E/en
Publication of JPS6052714B2 publication Critical patent/JPS6052714B2/ja
Priority to NL8901120A priority patent/NL8901120A/nl
Priority to US07/449,114 priority patent/USRE33778E/en
Expired legal-status Critical Current

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP53010772A 1977-06-10 1978-02-02 新規抗菌化合物 Expired JPS6052714B2 (ja)

Priority Applications (36)

Application Number Priority Date Filing Date Title
JP53010772A JPS6052714B2 (ja) 1978-02-02 1978-02-02 新規抗菌化合物
GB25353/78A GB1604739A (en) 1977-07-28 1978-05-31 7-methoxy-7-(1,3-dithietane-2-carboxamide) cephalosporanic acid derivatives
GB25352/78A GB1604738A (en) 1977-07-28 1978-05-31 1,3-dithietane-2-carboxylic acid derivatives and the preparation thereof
DE2824575A DE2824575C2 (de) 1977-07-28 1978-06-05 4-substituierte Methylen-1,3-dithietan-2-carbonsäure oder ihre niederen Alkylester, Verfahren zu ihrer Herstellung und ihre Verwendung als Acylierungsmittel
CH610878A CH636098A5 (de) 1977-07-28 1978-06-05 1,3-dithietan-2-carbonsaeuren sowie verfahren zu ihrer herstellung.
CH6107/78A CH648317A5 (de) 1977-06-10 1978-06-05 7alpha-methoxy-7betha-(1,3-dithietan-2- carboxamido)cephalosporansaeurederivate und verfahren zu ihrer herstellung.
DE2824559A DE2824559C2 (de) 1977-06-10 1978-06-05 7α-Methoxy-7β-(4-substituierte-methylen-1,3-dithietan-2-yl)-carboxamido-3-Δ↑3↑-cephem-4-carbonsäuren, Verfahren zu deren Herstellung sowie ihre Verwendung
US05/913,500 US4263432A (en) 1977-06-10 1978-06-07 7α-Methoxy-7β-(1,3-dithietane-2-carboxamido)cephalosporanic acid derivatives
NLAANVRAGE7806208,A NL185622C (nl) 1977-06-10 1978-06-07 Farmaceutisch preparaat met antibacteriele werking, alsmede 7beta-acylamino-7alfa-methoxy-3-heterocyclylthiomethyl-3-cefem-4-carbonzuur.
US05/913,501 US4198339A (en) 1977-07-28 1978-06-07 1,3-Dithietane-2-carboxylic acids and the preparation thereof
CA305,045A CA1103659A (en) 1977-06-10 1978-06-08 PROCESS FOR THE PREPARATION OF 7.alpha.-METHOXY-7.beta.-(1,3- DITHIETANE-2-CARBOXAMIDO)CEPHALOSPORANIC ACID DERIVATIVES
HU78JA822A HU178584B (en) 1977-07-28 1978-06-08 Process for preparing 7alpha-metoxy-7beta-/4-substituted methylene-1,3-dithiethan-2-yl-carboxamido/-ceph-3-em-4-carboxylic acid derivatives
UA2627106A UA5923A1 (uk) 1977-07-28 1978-06-09 СПОСІБ ОДЕРЖАННЯ 7alРha-МЕТОКСІ-7beta-(4-ЗАМІЩЕНИЙ МЕТІЛЕН-1,3-ДІТІЕТАН-2-ІЛКАРБОКСАМІДО)-3-(1-МЕТІЛТЕТРАЛ-5-ІЛТІОМЕТІЛ)-3-ЦЕФЕМ-4-КАРБОНОВИХ КИСЛОТ
DK258078A DK164224C (da) 1977-06-10 1978-06-09 Analogifremgangsmaade til fremstilling af 7alfa-methoxy-7beta-(4-methylen-1,3-dithietan-2-yl)carboxamido-3-heterocyclylthiomethyl-delta3-cephem-4-carboxylsyre-forbindelser eller salte deraf og mellemprodukter til anvendelse herved
FR7817304A FR2398745A1 (fr) 1977-07-28 1978-06-09 Acides dithietane-1,3-carboxylique-2 et leur procede de preparation
AT421978A AT360650B (de) 1977-07-28 1978-06-09 Verfahren zur herstellung von neuen 7alpha- methoxy-7beta-(1,3-dithiaethan-2-carboxamido) cephalosporansaeurederivaten
SE7806711A SE438338B (sv) 1977-06-10 1978-06-09 7alfa-metoxi-7beta-(1,3-ditietan-2-karboxamido)-cefalosporansyraderivat med antibakteriell verkan
ES470689A ES470689A1 (es) 1977-06-10 1978-06-09 Un procedimiento para la preparacion de acido 7-metoxi-7- (4-metilen sustituido-1,3-ditietan-2-il-carboxamido)-3-hete-rociclotiometil-3-cefem-4-carboxilico
FR7817303A FR2405952A1 (fr) 1977-06-10 1978-06-09 Derives de l'acide methoxy-7a-(dithietane-1,3-carboxamido-2)-cephalosporanique, presentant une activite anti-bacterienne et leurs procedes de preparation
SU782627106A SU818486A3 (ru) 1977-07-28 1978-06-09 Спосоь получени 7 -метокси - 7 -(4-зАМЕщЕННый МЕТилЕН-1,3-диТи-эТАН-2-илКАРбОКСАМидО)-3-(1-МЕТил-ТЕТРАзОл-5-илТиОМЕТил)-3-цЕфЕМ-4- КАРбОНОВыХ КиСлОТ
IT68369/78A IT1159721B (it) 1977-06-10 1978-06-12 Derivati dell'acido 7 alfa metossi-7 beta-(1,3-ditietane-2-carbossiamido)-cefalosporanico e procedimento per la loro preparazione
MX1051378U MX7170E (es) 1977-06-10 1978-06-12 Procedimiento para la preparacion del acido tiometil-delta3-cefem-4-carboxilico,7 alfa-metoxi-7beta-(metilen-1,3-ditietan-2-il 4-substituido)-carboxamido-3-heterociclico
MX787141U MX5137E (es) 1977-06-10 1978-06-12 Procedimiento para la preparacion del acido tio-metil-delta3-cefem-carboxilico,7 alfa metoxi-7 beta(metilen-1,3-ditietan-2-il-carboxamido-4-substituido)-3-heterociclico
MX1051478U MX7171E (es) 1977-06-10 1978-06-12 Procedimiento para la preparacion del acido tio-metil-delta3-cefem-4-carboxilico,7alfa-metoxi-7beta-(metilen-1,3-ditietan-2-il,4-substituido)carboxamido-3-heterociclico
IT68370/78A IT1109095B (it) 1977-07-28 1978-06-12 Acidi 1.3 ditietan 2 carbossilici e procedimento per la loro preparazione
ES479166A ES479166A1 (es) 1977-06-10 1979-03-31 Un procedimiento para la preparacion de acido 7&-metoxi-7b-(4-metilen sustituido 1,3-ditietan-2il) carboxamido-3-hetero-ciclotiometil-3-cefem-4-carboxilico.
ES479167A ES479167A1 (es) 1977-06-10 1979-03-31 Un procedimiento para la preparacion de acido 7&-metoxi-7b( 4-metilen sustituido-1,3-ditietan-2-il)carboxamido-3-hete- ro-ciclotiometil-3-cefem-4-carboxilico.
ES479168A ES479168A1 (es) 1977-06-10 1979-03-31 Un procedimiento para la preparacion de derivados de acido 7&-metoxicefalosporanico.
SU792805308A SU1024010A3 (ru) 1977-07-28 1979-08-31 Способ получени 7 @ -метокси-7 @ -(4-замещенный метилен-1,3-дитиэтан-2-илкарбоксамидо)-3-гетероциклический тиометил-3-цефем-4-карбоновых кислот
AT685879A AT361626B (de) 1977-07-28 1979-10-22 Verfahren zur herstellung von neuen 7alpha- -methoxy-7beta-(4-substituiert-methylen-1,3- -dithiaethan-2-yl)carboxamido-3-heterocyclisch- thiomethyl-delta3-cehpem-4-carbonsaeuren
US06/208,298 US4404373A (en) 1977-06-10 1980-11-19 Process for the preparation of 7α-methoxy-7β-(1,3-diethietane-2-carboxamido)cephalosporanic acid derivatives
US06/304,986 US4414153A (en) 1977-07-28 1981-09-23 1,3-Dithietane-2-carboxylic acid penicillin and cephalosporin derivatives
KE3489A KE3489A (en) 1977-07-28 1984-12-07 7alpha-methoxy-7beta-(1,3-dithietane-2-carboxamido)cephalosporanic acid derivatives
US06/727,233 USRE32491E (en) 1977-06-10 1985-04-25 Process for the preparation of 7α-methoxy-7β-(1,3-diethietane-2-carboxyamido)cephalosporanic acid derivatives
NL8901120A NL8901120A (nl) 1977-06-10 1989-05-02 Farmaceutisch preparaat met anti-bacteriele werking alsmede 7beta-acylamino 7alfa-methoxy-3-heterocyclylthiomethyl-3-cefem-4-carbonzuur.
US07/449,114 USRE33778E (en) 1977-07-28 1989-12-08 1,3-dithietane-2-carboxylic acid penicillin and cephalosporin derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP53010772A JPS6052714B2 (ja) 1978-02-02 1978-02-02 新規抗菌化合物

Publications (2)

Publication Number Publication Date
JPS54103890A true JPS54103890A (en) 1979-08-15
JPS6052714B2 JPS6052714B2 (ja) 1985-11-20

Family

ID=11759614

Family Applications (1)

Application Number Title Priority Date Filing Date
JP53010772A Expired JPS6052714B2 (ja) 1977-06-10 1978-02-02 新規抗菌化合物

Country Status (1)

Country Link
JP (1) JPS6052714B2 (ja)

Also Published As

Publication number Publication date
JPS6052714B2 (ja) 1985-11-20

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