JPH09169730A - エチルアミノカルバゾールメラトニン作動性薬 - Google Patents

エチルアミノカルバゾールメラトニン作動性薬

Info

Publication number
JPH09169730A
JPH09169730A JP8289439A JP28943996A JPH09169730A JP H09169730 A JPH09169730 A JP H09169730A JP 8289439 A JP8289439 A JP 8289439A JP 28943996 A JP28943996 A JP 28943996A JP H09169730 A JPH09169730 A JP H09169730A
Authority
JP
Japan
Prior art keywords
dimethoxy
carbazol
ethyl
nmr
dmso
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP8289439A
Other languages
English (en)
Japanese (ja)
Other versions
JPH09169730A5 (https=
Inventor
Katherine S Takaki
エス タカキ カサリーン
Marc A Bruce
エイ ブルース マーク
Graham S Poindexter
エス ポインデクスター グレイアム
Brett T Watson
ティー ワトソン ブレット
Joseph P Yevich
ピー イェーヴィック ジョセフ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of JPH09169730A publication Critical patent/JPH09169730A/ja
Publication of JPH09169730A5 publication Critical patent/JPH09169730A5/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
JP8289439A 1995-10-31 1996-10-31 エチルアミノカルバゾールメラトニン作動性薬 Pending JPH09169730A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US815495P 1995-10-31 1995-10-31
US60/008154 1995-10-31

Publications (2)

Publication Number Publication Date
JPH09169730A true JPH09169730A (ja) 1997-06-30
JPH09169730A5 JPH09169730A5 (https=) 2004-10-21

Family

ID=21730073

Family Applications (1)

Application Number Title Priority Date Filing Date
JP8289439A Pending JPH09169730A (ja) 1995-10-31 1996-10-31 エチルアミノカルバゾールメラトニン作動性薬

Country Status (4)

Country Link
US (1) US5677328A (https=)
EP (1) EP0771791A1 (https=)
JP (1) JPH09169730A (https=)
CA (1) CA2186412A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100130579A1 (en) * 2006-10-23 2010-05-27 Georgetown University Cancer therapy
ES2331274B1 (es) * 2007-10-25 2010-10-21 Ferrer Internacional, S.A. Compuesto de indolina.
CN102186820B (zh) * 2008-08-15 2013-08-28 乔治城大学 Rassf1a表达和人癌细胞增殖的荧光调节剂
WO2015003146A1 (en) 2013-07-03 2015-01-08 Georgetown University Boronic acid derivatives of resveratrol for activating deacetylase enzymes
US11053255B2 (en) 2015-06-22 2021-07-06 Georgetown University Synthesis of mahanine and related compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3975398A (en) * 1973-08-01 1976-08-17 Boehringer Mannheim G.M.B.H. 9-Substituted 3-aminocarbazole compounds
US5206377A (en) 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
US5449683A (en) 1992-10-01 1995-09-12 Massachussetts Institute Of Technology Methods of inducing sleep using melatonin

Also Published As

Publication number Publication date
US5677328A (en) 1997-10-14
CA2186412A1 (en) 1997-05-01
AU7049796A (en) 1997-05-08
AU701113B2 (en) 1999-01-21
EP0771791A1 (en) 1997-05-07

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