JP6804297B2 - ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 - Google Patents

５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 Download PDF

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JP6804297B2
JP6804297B2 JP2016543746A JP2016543746A JP6804297B2 JP 6804297 B2 JP6804297 B2 JP 6804297B2 JP 2016543746 A JP2016543746 A JP 2016543746A JP 2016543746 A JP2016543746 A JP 2016543746A JP 6804297 B2 JP6804297 B2 JP 6804297B2
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formula
molar ratio
plant
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JP2017502963A5 (https=
JP2017502963A (ja
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チョイ，ナキェン
ロス，ジュニア．，ロナルド
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アダマ・マクテシム・リミテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
    • C07D333/10—Thiophene
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Detergent Compositions (AREA)
  • Cosmetics (AREA)
JP2016543746A 2013-12-31 2014-12-29 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 Active JP6804297B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361922582P 2013-12-31 2013-12-31
US201361922572P 2013-12-31 2013-12-31
US61/922,582 2013-12-31
US61/922,572 2013-12-31
PCT/US2014/072566 WO2015103142A1 (en) 2013-12-31 2014-12-29 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation

Publications (3)

Publication Number Publication Date
JP2017502963A JP2017502963A (ja) 2017-01-26
JP2017502963A5 JP2017502963A5 (https=) 2018-02-15
JP6804297B2 true JP6804297B2 (ja) 2020-12-23

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JP2016543746A Active JP6804297B2 (ja) 2013-12-31 2014-12-29 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
JP2016543735A Active JP6585057B2 (ja) 2013-12-31 2014-12-29 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
JP2019160781A Withdrawn JP2019218396A (ja) 2013-12-31 2019-09-04 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法

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JP2016543735A Active JP6585057B2 (ja) 2013-12-31 2014-12-29 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
JP2019160781A Withdrawn JP2019218396A (ja) 2013-12-31 2019-09-04 ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法

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US (8) US20150183750A1 (https=)
EP (4) EP3862347A1 (https=)
JP (3) JP6804297B2 (https=)
CN (4) CN111217759A (https=)
AP (1) AP2016009342A0 (https=)
AU (2) AU2014373959B2 (https=)
BR (2) BR102014033010B1 (https=)
CA (2) CA2935594C (https=)
CL (1) CL2016001677A1 (https=)
CR (2) CR20160343A (https=)
DO (1) DOP2016000163A (https=)
EA (2) EA036389B1 (https=)
EC (1) ECSP16064249A (https=)
IL (3) IL246512B (https=)
MX (2) MX392211B (https=)
NI (1) NI201600094A (https=)
NZ (2) NZ722438A (https=)
PE (1) PE20161174A1 (https=)
PH (1) PH12016501284A1 (https=)
SG (2) SG11201605372QA (https=)
TW (2) TWI667229B (https=)
UA (2) UA129860C2 (https=)
UY (2) UY35942A (https=)
WO (2) WO2015103144A1 (https=)

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CN118139845A (zh) 2021-09-15 2024-06-04 安道麦马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
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AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
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NZ722438A (en) 2018-01-26
JP2019218396A (ja) 2019-12-26
SG11201605377VA (en) 2016-08-30
MX375727B (es) 2025-03-06
UY35942A (es) 2015-07-31
EA036389B1 (ru) 2020-11-03
MX2016008758A (es) 2017-05-09
US20150183750A1 (en) 2015-07-02
IL269694B (en) 2021-09-30
TWI667229B (zh) 2019-08-01
CN111362881A (zh) 2020-07-03
US20180072686A1 (en) 2018-03-15
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BR102014033037A2 (pt) 2015-11-17
IL246512B (en) 2019-09-26
EP3097096A1 (en) 2016-11-30
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DOP2016000163A (es) 2016-09-30
EA201691351A1 (ru) 2016-12-30
CN106068268A (zh) 2016-11-02
AP2016009342A0 (en) 2016-07-31
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US20160280663A1 (en) 2016-09-29
US20200148649A1 (en) 2020-05-14
CL2016001677A1 (es) 2016-12-09
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IL269694A (en) 2019-11-28
IL246511B (en) 2019-10-31
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AU2014373959A1 (en) 2016-08-11
UY35943A (es) 2015-07-31
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US20150183749A1 (en) 2015-07-02
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