JP6586104B2 - ５−置換インダゾール−３−カルボキサミドならびにその調製および使用の方法 - Google Patents

５−置換インダゾール−３−カルボキサミドならびにその調製および使用の方法 Download PDF

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JP6586104B2
JP6586104B2 JP2016558073A JP2016558073A JP6586104B2 JP 6586104 B2 JP6586104 B2 JP 6586104B2 JP 2016558073 A JP2016558073 A JP 2016558073A JP 2016558073 A JP2016558073 A JP 2016558073A JP 6586104 B2 JP6586104 B2 JP 6586104B2
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pyridin
carboxamide
indazole
alkyl
ylmethyl
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JP2017508763A (ja
JP2017508763A5 (enExample
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ジョン フード
ジョン フード
スニル クマー ケーシー
スニル クマー ケーシー
デービッド マーク ウォーレンス
デービッド マーク ウォーレンス
ゴピ クマー ミッタパリ
ゴピ クマー ミッタパリ
ブライアン ジョゼフ ホフィレナ
ブライアン ジョゼフ ホフィレナ
チ チン マック
チ チン マック
ベンカタイア ボル
ベンカタイア ボル
ブライアン イーストマン
ブライアン イーストマン
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サミュメッド リミテッド ライアビリティ カンパニー
サミュメッド リミテッド ライアビリティ カンパニー
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    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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JP2016558073A 2014-03-20 2015-03-20 ５−置換インダゾール−３−カルボキサミドならびにその調製および使用の方法 Active JP6586104B2 (ja)

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US201461968350P 2014-03-20 2014-03-20
US61/968,350 2014-03-20
PCT/US2015/021847 WO2015143380A1 (en) 2014-03-20 2015-03-20 5-substituted indazole-3-carboxamides and preparation and use thereof

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JP2017508763A JP2017508763A (ja) 2017-03-30
JP2017508763A5 JP2017508763A5 (enExample) 2018-05-10
JP6586104B2 true JP6586104B2 (ja) 2019-10-02

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US (2) US9745271B2 (enExample)
EP (1) EP3119393A4 (enExample)
JP (1) JP6586104B2 (enExample)
KR (1) KR20160135283A (enExample)
CN (1) CN106535890A (enExample)
BR (1) BR112016021626A2 (enExample)
CA (1) CA2942687A1 (enExample)
CL (1) CL2016002364A1 (enExample)
IL (1) IL247713A0 (enExample)
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RU (1) RU2016141088A (enExample)
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PH12017500997A1 (en) 2012-04-04 2018-02-19 Samumed Llc Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof
WO2014110086A2 (en) 2013-01-08 2014-07-17 Samumed, Llc 3-(benzoimidazol-2-yl)-indazole inhibitors of the wnt signaling pathway and therapeutic uses thereof
EP3119393A4 (en) 2014-03-20 2018-02-28 Samumed, LLC 5-substituted indazole-3-carboxamides and preparation and use thereof
WO2016040180A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
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WO2016040185A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 2-(1h-indazol-3-yl)-3h-imidazo[4,5-b]pyridine and therapeutic uses thereof
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