KR20160135283A - 5-치환된 인다졸-3-카르복스아미드 및 이의 제조 및 용도 - Google Patents

5-치환된 인다졸-3-카르복스아미드 및 이의 제조 및 용도 Download PDF

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KR20160135283A
KR20160135283A KR1020167028641A KR20167028641A KR20160135283A KR 20160135283 A KR20160135283 A KR 20160135283A KR 1020167028641 A KR1020167028641 A KR 1020167028641A KR 20167028641 A KR20167028641 A KR 20167028641A KR 20160135283 A KR20160135283 A KR 20160135283A
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carboxamide
indazole
pyridin
alkyl
ylmethyl
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존 후드
써닐 쿠마르 케이씨
데이비드 마크 월레이스
고피 쿠마르 미타팔리
브리안 죠셉 호필레나
치 칭 막
벤카타이아 볼루
브라이언 이스트맨
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사뮤메드, 엘엘씨
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KR1020167028641A 2014-03-20 2015-03-20 5-치환된 인다졸-3-카르복스아미드 및 이의 제조 및 용도 Withdrawn KR20160135283A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461968350P 2014-03-20 2014-03-20
US61/968,350 2014-03-20
PCT/US2015/021847 WO2015143380A1 (en) 2014-03-20 2015-03-20 5-substituted indazole-3-carboxamides and preparation and use thereof

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KR20160135283A true KR20160135283A (ko) 2016-11-25

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US (2) US9745271B2 (enExample)
EP (1) EP3119393A4 (enExample)
JP (1) JP6586104B2 (enExample)
KR (1) KR20160135283A (enExample)
CN (1) CN106535890A (enExample)
BR (1) BR112016021626A2 (enExample)
CA (1) CA2942687A1 (enExample)
CL (1) CL2016002364A1 (enExample)
IL (1) IL247713A0 (enExample)
MA (1) MA39763A (enExample)
MX (1) MX2016012208A (enExample)
PE (1) PE20170127A1 (enExample)
PH (1) PH12016501835A1 (enExample)
RU (1) RU2016141088A (enExample)
SG (2) SG10201914111XA (enExample)
WO (1) WO2015143380A1 (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20190043013A (ko) * 2017-10-17 2019-04-25 한국화학연구원 신규한 인다졸 유도체 및 이의 용도
KR20210005863A (ko) * 2018-05-07 2021-01-15 아지엔드 키미쉐 리유나이트 안젤리니 프란체스코 에이.씨.알.에이.에프. 에스.피.에이 글리코겐 합성효소 키나아제 3 베타 억제제로서 1h-인다졸-3-카복사마이드 화합물
WO2021125802A1 (ko) * 2019-12-16 2021-06-24 한국화학연구원 신규한 인다졸 유도체 및 이의 용도

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HUE041576T2 (hu) 2011-09-14 2019-05-28 Samumed Llc Indazol-3-karboxamid-származékok és alkalmazásuk Wnt/b-katenin szignalizáló útvonal inhibitorokként
PH12017500997A1 (en) 2012-04-04 2018-02-19 Samumed Llc Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof
US9908867B2 (en) 2013-01-08 2018-03-06 Samumed, Llc 3-(benzoimidazol-2-yl)-indazole inhibitors of the Wnt signaling pathway and therapeutic uses thereof
BR112016021626A2 (pt) 2014-03-20 2018-05-15 Samumed, Llc indazol-3-carboxamidas 5-substituídas e preparação e uso das mesmas
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
WO2016040190A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
WO2016040185A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 2-(1h-indazol-3-yl)-3h-imidazo[4,5-b]pyridine and therapeutic uses thereof
WO2016040184A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
WO2016040181A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
WO2016040180A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
US10195185B2 (en) 2015-08-03 2019-02-05 Samumed, Llc 3-(1H-imidazo[4,5-C]pyridin-2-yl)-1H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
US10350199B2 (en) 2015-08-03 2019-07-16 Samumed, Llc 3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indazoles and therapeutic uses thereof
WO2017024025A1 (en) 2015-08-03 2017-02-09 Sunil Kumar Kc 3-(1h-pyrrolo[2,3-c]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
WO2017023987A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(1h-pyrrolo[3,2-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
WO2017023989A1 (en) 2015-08-03 2017-02-09 Samumed, Llc. 3-(1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
US10231956B2 (en) 2015-08-03 2019-03-19 Samumed, Llc 3-(1H-pyrrolo[3,2-C]pyridin-2-YL)-1 H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
US10206909B2 (en) 2015-08-03 2019-02-19 Samumed, Llc 3-(1H-pyrrolo[2,3-B]pyridin-2-yl)-1H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
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