JP6535022B2 - ヘテロアリールｓｙｋ阻害剤 - Google Patents

ヘテロアリールｓｙｋ阻害剤 Download PDF

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JP6535022B2
JP6535022B2 JP2016557602A JP2016557602A JP6535022B2 JP 6535022 B2 JP6535022 B2 JP 6535022B2 JP 2016557602 A JP2016557602 A JP 2016557602A JP 2016557602 A JP2016557602 A JP 2016557602A JP 6535022 B2 JP6535022 B2 JP 6535022B2
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amino
acid
methyl
phenyl
ethyl
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JP2017512779A5 (enExample
JP2017512779A (ja
Inventor
ダーマン，ゲオルク
ホフマン，マティアス
クリシク，ヤスナ
ラム，デイビッド・ジェームズ
マッカーシー，クライブ
ネイピア，スペンサー
パリッシュ，カレン
スコット，ジョン
フィッツジェラルド，ジェニファー・エル・スワンテック
ウォーカー，エドワード
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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KR20160132999A (ko) 2016-11-21
CA2942997A1 (en) 2015-09-24
PL3119772T3 (pl) 2019-11-29
IL247057A0 (en) 2016-09-29
RS59110B1 (sr) 2019-09-30
CN110183440B (zh) 2022-04-22
WO2015140055A1 (en) 2015-09-24
CN110183440A (zh) 2019-08-30
EP3119772A1 (en) 2017-01-25
JP6599884B2 (ja) 2019-10-30
CN106255689A (zh) 2016-12-21
AP2016009373A0 (en) 2016-08-31
AR099785A1 (es) 2016-08-17
WO2015140054A1 (en) 2015-09-24
EP3119772B1 (en) 2019-05-22
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JP2017511805A (ja) 2017-04-27
LT3119772T (lt) 2019-08-26
WO2015140051A1 (en) 2015-09-24
IL247057B (en) 2019-10-31
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SI3119772T1 (sl) 2019-08-30
ES2738416T3 (es) 2020-01-22
CN110713489B (zh) 2022-05-31
TW201623285A (zh) 2016-07-01
CL2016001963A1 (es) 2016-12-23
WO2015140051A8 (en) 2015-12-30
UY36037A (es) 2015-09-30
JP2017512779A (ja) 2017-05-25
JP6416275B2 (ja) 2018-10-31
UA119667C2 (uk) 2019-07-25
US20190359620A1 (en) 2019-11-28
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EP3119772B8 (en) 2019-08-21
US20180072744A1 (en) 2018-03-15
DK3119772T3 (da) 2019-08-26
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EP3119765A1 (en) 2017-01-25
EP3119766B1 (en) 2019-05-22
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AU2015233654A1 (en) 2016-08-11
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MX2016011784A (es) 2016-12-02

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