JP6419347B2 - 胃腸疾患治療用医薬組成物 - Google Patents
胃腸疾患治療用医薬組成物 Download PDFInfo
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- JP6419347B2 JP6419347B2 JP2017540683A JP2017540683A JP6419347B2 JP 6419347 B2 JP6419347 B2 JP 6419347B2 JP 2017540683 A JP2017540683 A JP 2017540683A JP 2017540683 A JP2017540683 A JP 2017540683A JP 6419347 B2 JP6419347 B2 JP 6419347B2
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- AXZKOIWUVFPNLO-UHFFFAOYSA-N magnesium;oxygen(2-) Chemical compound [O-2].[Mg+2] AXZKOIWUVFPNLO-UHFFFAOYSA-N 0.000 description 1
- 239000000594 mannitol Substances 0.000 description 1
- 235000010355 mannitol Nutrition 0.000 description 1
- 238000000691 measurement method Methods 0.000 description 1
- 239000012528 membrane Substances 0.000 description 1
- 229940016286 microcrystalline cellulose Drugs 0.000 description 1
- 235000019813 microcrystalline cellulose Nutrition 0.000 description 1
- 239000008108 microcrystalline cellulose Substances 0.000 description 1
- 239000002480 mineral oil Substances 0.000 description 1
- 235000010446 mineral oil Nutrition 0.000 description 1
- 239000001788 mono and diglycerides of fatty acids Substances 0.000 description 1
- 239000000041 non-steroidal anti-inflammatory agent Substances 0.000 description 1
- 229940021182 non-steroidal anti-inflammatory drug Drugs 0.000 description 1
- 150000007530 organic bases Chemical class 0.000 description 1
- 210000004798 organs belonging to the digestive system Anatomy 0.000 description 1
- 239000012071 phase Substances 0.000 description 1
- 229960000540 polacrilin potassium Drugs 0.000 description 1
- 229920001223 polyethylene glycol Polymers 0.000 description 1
- 235000013809 polyvinylpolypyrrolidone Nutrition 0.000 description 1
- 229920000523 polyvinylpolypyrrolidone Polymers 0.000 description 1
- 239000001267 polyvinylpyrrolidone Substances 0.000 description 1
- 230000002980 postoperative effect Effects 0.000 description 1
- 239000001103 potassium chloride Substances 0.000 description 1
- 235000011164 potassium chloride Nutrition 0.000 description 1
- WVWZXTJUCNEUAE-UHFFFAOYSA-M potassium;1,2-bis(ethenyl)benzene;2-methylprop-2-enoate Chemical compound [K+].CC(=C)C([O-])=O.C=CC1=CC=CC=C1C=C WVWZXTJUCNEUAE-UHFFFAOYSA-M 0.000 description 1
- 229940069328 povidone Drugs 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
- 230000002265 prevention Effects 0.000 description 1
- 230000008569 process Effects 0.000 description 1
- -1 pyridine Chemical class 0.000 description 1
- UMJSCPRVCHMLSP-UHFFFAOYSA-N pyridine Natural products COC1=CC=CN=C1 UMJSCPRVCHMLSP-UHFFFAOYSA-N 0.000 description 1
- 238000011160 research Methods 0.000 description 1
- 230000004044 response Effects 0.000 description 1
- 238000000790 scattering method Methods 0.000 description 1
- 230000028327 secretion Effects 0.000 description 1
- 230000035945 sensitivity Effects 0.000 description 1
- 238000007873 sieving Methods 0.000 description 1
- 235000010413 sodium alginate Nutrition 0.000 description 1
- 239000000661 sodium alginate Substances 0.000 description 1
- 229940005550 sodium alginate Drugs 0.000 description 1
- WXMKPNITSTVMEF-UHFFFAOYSA-M sodium benzoate Chemical compound [Na+].[O-]C(=O)C1=CC=CC=C1 WXMKPNITSTVMEF-UHFFFAOYSA-M 0.000 description 1
- 235000010234 sodium benzoate Nutrition 0.000 description 1
- 239000004299 sodium benzoate Substances 0.000 description 1
- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- 235000019333 sodium laurylsulphate Nutrition 0.000 description 1
- 229940080313 sodium starch Drugs 0.000 description 1
- 229920003109 sodium starch glycolate Polymers 0.000 description 1
- 239000008109 sodium starch glycolate Substances 0.000 description 1
- 229940079832 sodium starch glycolate Drugs 0.000 description 1
- 229940045902 sodium stearyl fumarate Drugs 0.000 description 1
- YFGAFXCSLUUJRG-WCCKRBBISA-M sodium;(2s)-2-amino-5-(diaminomethylideneamino)pentanoate Chemical compound [Na+].[O-]C(=O)[C@@H](N)CCCN=C(N)N YFGAFXCSLUUJRG-WCCKRBBISA-M 0.000 description 1
- 239000008279 sol Substances 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
- 208000011580 syndromic disease Diseases 0.000 description 1
- 230000002194 synthesizing effect Effects 0.000 description 1
- 230000001225 therapeutic effect Effects 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- 235000019731 tricalcium phosphate Nutrition 0.000 description 1
- 239000003643 water by type Substances 0.000 description 1
- XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical compound [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
- 229940057977 zinc stearate Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7024—Esters of saccharides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/245—Bismuth; Compounds thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Inorganic Chemistry (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR10-2015-0015339 | 2015-01-30 | ||
| KR20150015339 | 2015-01-30 | ||
| KR1020150147513A KR101583452B1 (ko) | 2015-01-30 | 2015-10-22 | 위장질환 치료용 의약 조성물 |
| KR10-2015-0147513 | 2015-10-22 | ||
| PCT/KR2016/000935 WO2016122226A2 (en) | 2015-01-30 | 2016-01-28 | A pharmaceutical composition for treating gastrointestinal diseases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018503672A JP2018503672A (ja) | 2018-02-08 |
| JP6419347B2 true JP6419347B2 (ja) | 2018-11-07 |
Family
ID=55169799
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017540683A Active JP6419347B2 (ja) | 2015-01-30 | 2016-01-28 | 胃腸疾患治療用医薬組成物 |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP3250199A4 (zh) |
| JP (1) | JP6419347B2 (zh) |
| KR (2) | KR101583452B1 (zh) |
| CN (1) | CN107205947B (zh) |
| AR (1) | AR105413A1 (zh) |
| CL (1) | CL2017001680A1 (zh) |
| CO (1) | CO2017006222A2 (zh) |
| EA (1) | EA032385B9 (zh) |
| EC (1) | ECSP17038599A (zh) |
| GE (1) | GEP20196941B (zh) |
| MA (1) | MA41432A (zh) |
| MX (1) | MX2017007567A (zh) |
| MY (1) | MY195824A (zh) |
| PE (1) | PE20171340A1 (zh) |
| PH (1) | PH12017550051A1 (zh) |
| SA (1) | SA517382016B1 (zh) |
| TW (1) | TWI635859B (zh) |
| UA (1) | UA116517C2 (zh) |
| WO (1) | WO2016122226A2 (zh) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101988479B1 (ko) | 2017-10-11 | 2019-09-24 | (주)휴럼 | 리트세노라이드를 유효성분으로 하는 헬리코박터 파이로리 균주로부터 유래되는 위장질환 예방 및 치료용 약학 조성물 |
| WO2019199134A1 (ko) * | 2018-04-13 | 2019-10-17 | 주식회사 삼양바이오팜 | 레날리도마이드를 포함하는 약제학적 조성물 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE81011T1 (de) * | 1987-03-09 | 1992-10-15 | Procter & Gamble | Zusammensetzungen und ihre verwendung zur behandlung von magen-darmstoerungen. |
| US4990610A (en) * | 1988-08-25 | 1991-02-05 | Applied Analytical Industries, Inc. | Method for preparing high potency sucralfate |
| EP0403048A3 (en) * | 1989-06-14 | 1991-01-30 | Warner-Lambert Company | Medicated compositions containing sucralfate and processes for their production |
| KR970006083B1 (ko) * | 1992-01-22 | 1997-04-23 | 주식회사 대웅제약 | 위장질환 치료용 의약 조성물 |
| ES2173183T3 (es) * | 1994-04-26 | 2002-10-16 | Chugai Pharmaceutical Co Ltd | Procedimiento de preparacion de sucralfato granulado y fundido. |
| JPH0879097A (ja) * | 1994-09-01 | 1996-03-22 | Matsushita Electric Ind Co Ltd | 携帯無線機 |
| KR970006083A (ko) | 1995-07-06 | 1997-02-19 | 한승준 | 자동차용 카울부의 와이어 고정장치 취부구조 |
| AU8354498A (en) * | 1997-08-25 | 1999-03-16 | Procter & Gamble Company, The | Combined preparations for treating upper gastrointestinal tract distress |
| CN1173698C (zh) | 1999-06-21 | 2004-11-03 | 株式会社大熊制药 | 包含包衣的雷尼替丁、碱式柠檬酸铋和硫糖铝的对胃肠障碍具有治疗作用的可口服给药的药物制剂 |
| JP2006076956A (ja) * | 2004-09-10 | 2006-03-23 | Taiyo Yakuhin Kogyo Kk | 胃炎の治療・予防用配合剤 |
| KR101617054B1 (ko) * | 2008-07-01 | 2016-04-29 | 라이온 가부시키가이샤 | 고형내복제제 |
| KR20110105223A (ko) * | 2010-03-18 | 2011-09-26 | 일양약품주식회사 | 일라프라졸 및 수크랄페이트와 비스무스 제제의 혼합물을 함유하는 위장질환을 예방 또는 치료하기 위한 경구용 약제 조성물 |
| KR20140072673A (ko) | 2012-12-05 | 2014-06-13 | (주)한국파비스제약 | 경구용 위장질환 치료를 위한 정제 |
-
2015
- 2015-10-22 KR KR1020150147513A patent/KR101583452B1/ko active IP Right Review Request
- 2015-12-31 KR KR1020150190850A patent/KR20160094268A/ko active Application Filing
-
2016
- 2016-01-27 MA MA041432A patent/MA41432A/fr unknown
- 2016-01-27 TW TW105102582A patent/TWI635859B/zh active
- 2016-01-28 CN CN201680007680.7A patent/CN107205947B/zh active Active
- 2016-01-28 UA UAA201707833A patent/UA116517C2/uk unknown
- 2016-01-28 MY MYPI2017702737A patent/MY195824A/en unknown
- 2016-01-28 EP EP16743704.5A patent/EP3250199A4/en not_active Withdrawn
- 2016-01-28 JP JP2017540683A patent/JP6419347B2/ja active Active
- 2016-01-28 EA EA201791458A patent/EA032385B9/ru not_active IP Right Cessation
- 2016-01-28 WO PCT/KR2016/000935 patent/WO2016122226A2/en active Application Filing
- 2016-01-28 PE PE2017001147A patent/PE20171340A1/es unknown
- 2016-01-28 MX MX2017007567A patent/MX2017007567A/es active IP Right Grant
- 2016-01-28 GE GEAP201614551A patent/GEP20196941B/en unknown
- 2016-01-29 AR ARP160100272A patent/AR105413A1/es unknown
-
2017
- 2017-06-20 EC ECIEPI201738599A patent/ECSP17038599A/es unknown
- 2017-06-23 CO CONC2017/0006222A patent/CO2017006222A2/es unknown
- 2017-06-23 CL CL2017001680A patent/CL2017001680A1/es unknown
- 2017-07-25 PH PH12017550051A patent/PH12017550051A1/en unknown
- 2017-07-29 SA SA517382016A patent/SA517382016B1/ar unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TWI635859B (zh) | 2018-09-21 |
| ECSP17038599A (es) | 2017-09-29 |
| KR20160094268A (ko) | 2016-08-09 |
| EP3250199A2 (en) | 2017-12-06 |
| MY195824A (en) | 2023-02-22 |
| SA517382016B1 (ar) | 2021-03-18 |
| AR105413A1 (es) | 2017-10-04 |
| CN107205947B (zh) | 2020-05-22 |
| KR101583452B1 (ko) | 2016-01-11 |
| EP3250199A4 (en) | 2018-08-08 |
| WO2016122226A2 (en) | 2016-08-04 |
| JP2018503672A (ja) | 2018-02-08 |
| MX2017007567A (es) | 2017-10-19 |
| CN107205947A (zh) | 2017-09-26 |
| TW201639559A (zh) | 2016-11-16 |
| UA116517C2 (uk) | 2018-03-26 |
| PH12017550051A1 (en) | 2018-01-29 |
| EA032385B9 (ru) | 2019-07-31 |
| CL2017001680A1 (es) | 2018-01-12 |
| PE20171340A1 (es) | 2017-09-13 |
| CO2017006222A2 (es) | 2017-09-20 |
| EA201791458A1 (ru) | 2017-11-30 |
| EA032385B1 (ru) | 2019-05-31 |
| KR101583452B9 (ko) | 2022-05-02 |
| WO2016122226A3 (en) | 2016-09-15 |
| GEP20196941B (en) | 2019-01-10 |
| BR112017013857A2 (pt) | 2018-02-27 |
| MA41432A (fr) | 2017-12-05 |
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