JP6300207B2 - 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤 - Google Patents

新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤 Download PDF

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Publication number
JP6300207B2
JP6300207B2 JP2014521405A JP2014521405A JP6300207B2 JP 6300207 B2 JP6300207 B2 JP 6300207B2 JP 2014521405 A JP2014521405 A JP 2014521405A JP 2014521405 A JP2014521405 A JP 2014521405A JP 6300207 B2 JP6300207 B2 JP 6300207B2
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formula
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JP2014521405A
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Japanese (ja)
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JPWO2013187480A1 (ja
Inventor
正明 三冨
正明 三冨
政世 坂井
政世 坂井
亮 堀越
亮 堀越
保道 小野崎
保道 小野崎
中村　哲
哲 中村
大村　智
智 大村
砂塚　敏明
敏明 砂塚
友靖 廣瀬
友靖 廣瀬
塩見　和朗
和朗 塩見
碌郎 増間
碌郎 増間
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Meiji Seika Kaisha Ltd
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Meiji Seika Kaisha Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B51/00—Introduction of protecting groups or activating groups, not provided for in the preceding groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C235/12—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C07D273/08—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00 having two nitrogen atoms and more than one oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2014521405A 2012-06-13 2013-06-13 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤 Expired - Fee Related JP6300207B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2014521405A JP6300207B2 (ja) 2012-06-13 2013-06-13 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2012134304 2012-06-13
JP2012134304 2012-06-13
JP2014521405A JP6300207B2 (ja) 2012-06-13 2013-06-13 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤
PCT/JP2013/066360 WO2013187480A1 (ja) 2012-06-13 2013-06-13 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤

Publications (2)

Publication Number Publication Date
JPWO2013187480A1 JPWO2013187480A1 (ja) 2016-02-08
JP6300207B2 true JP6300207B2 (ja) 2018-03-28

Family

ID=49758298

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JP2014521405A Expired - Fee Related JP6300207B2 (ja) 2012-06-13 2013-06-13 新規環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤

Country Status (19)

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US (2) US20150166608A1 (enExample)
EP (2) EP2862872B1 (enExample)
JP (1) JP6300207B2 (enExample)
KR (1) KR20150037766A (enExample)
CN (1) CN104540845B (enExample)
AU (2) AU2013275223A1 (enExample)
BR (1) BR112014031334A2 (enExample)
CA (1) CA2876387A1 (enExample)
ES (1) ES2702598T3 (enExample)
HU (1) HUE042661T2 (enExample)
IN (1) IN2014DN10617A (enExample)
MX (1) MX2014014838A (enExample)
NZ (1) NZ703217A (enExample)
PH (1) PH12014502752A1 (enExample)
PL (1) PL2862872T3 (enExample)
PT (1) PT2862872T (enExample)
RU (1) RU2015100521A (enExample)
TW (1) TWI609860B (enExample)
WO (1) WO2013187480A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3038640B1 (en) 2013-08-30 2019-01-02 St. Jude Children's Research Hospital Substituted urea depsipeptide analogs as activators of the clpp endopeptidase
WO2015093558A1 (ja) * 2013-12-18 2015-06-25 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤
US10100090B2 (en) 2015-03-04 2018-10-16 St. Jude Children's Research Hospital Substituted urea depsipeptide analogs as activators of the CLPP endopeptidase
US10308729B2 (en) 2015-05-08 2019-06-04 Exxonmobil Chemical Patents Inc. Reactor systems and processes related thereto
CN107835818B (zh) 2015-05-20 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
KR20220003663A (ko) 2015-12-28 2022-01-10 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 뎁시펩티드 화합물
EP3506922B1 (en) 2016-09-02 2024-05-08 St. Jude Children's Research Hospital Substituted urea depsipeptide analogs as activators of the clpp endopeptidase
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
EP3480195A1 (en) * 2017-11-07 2019-05-08 Bayer Animal Health GmbH Method for the synthesis of cyclic depsipeptides
CN111757880A (zh) * 2017-11-07 2020-10-09 拜耳动物保健有限责任公司 用于合成环状缩肽的方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
JP3132167B2 (ja) 1991-08-23 2001-02-05 藤沢薬品工業株式会社 デプシペプチド誘導体の製造法
CA2132199C (en) 1992-03-17 2000-01-18 Hitoshi Nishiyama Depsipeptide derivative, production thereof and use thereof
JPH05271013A (ja) 1992-03-27 1993-10-19 Meiji Seika Kaisha Ltd 環状デプシペプチド物質を有効成分とする害虫防除剤
CN1073560C (zh) * 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317432A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
AU6229898A (en) * 1997-02-19 1998-09-09 Bayer Aktiengesellschaft Derivatives of cyclodepsipeptide, pf1022 substance
DE19828043A1 (de) * 1998-06-24 1999-12-30 Bayer Ag Ektoparasitizide Mittel
DE19840320A1 (de) * 1998-09-04 2000-03-09 Bayer Ag Aza-Cyclodepsipeptide
DE19962145A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel/Depsipeptide
EP1561820B1 (en) * 2002-11-12 2008-12-31 The Kitasato Institute Anthelmintic substance fki-1033 and process for producing the same
JP4734656B2 (ja) * 2007-03-30 2011-07-27 国立大学法人群馬大学 Ｐｆ１０２２類の製造法
EP2509967B1 (en) 2009-12-11 2016-02-17 Bayer Intellectual Property GmbH Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides
JP2014037351A (ja) * 2010-12-10 2014-02-27 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 新規デプシペプチドｐｆ１４４２物質およびその製造法

Also Published As

Publication number Publication date
PL2862872T3 (pl) 2019-03-29
US20170215422A1 (en) 2017-08-03
TW201410659A (zh) 2014-03-16
BR112014031334A2 (pt) 2017-06-27
ES2702598T3 (es) 2019-03-04
WO2013187480A1 (ja) 2013-12-19
JPWO2013187480A1 (ja) 2016-02-08
EP2862872A4 (en) 2015-10-28
CN104540845A (zh) 2015-04-22
MX2014014838A (es) 2015-02-12
PH12014502752A1 (en) 2015-02-23
RU2015100521A (ru) 2016-08-10
CA2876387A1 (en) 2013-12-19
EP2862872B1 (en) 2018-09-19
AU2018201101A1 (en) 2018-03-08
IN2014DN10617A (enExample) 2015-09-11
KR20150037766A (ko) 2015-04-08
EP2862872A1 (en) 2015-04-22
HUE042661T2 (hu) 2019-07-29
US20150166608A1 (en) 2015-06-18
NZ703217A (en) 2016-11-25
EP3441399A1 (en) 2019-02-13
CN104540845B (zh) 2018-01-26
TWI609860B (zh) 2018-01-01
AU2013275223A1 (en) 2015-01-22
PT2862872T (pt) 2018-12-17

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