JP6023082B2 - 精神神経性の疾病を処置するためのプロスタグランジンを含む組成物 - Google Patents

精神神経性の疾病を処置するためのプロスタグランジンを含む組成物 Download PDF

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JP6023082B2
JP6023082B2 JP2013549683A JP2013549683A JP6023082B2 JP 6023082 B2 JP6023082 B2 JP 6023082B2 JP 2013549683 A JP2013549683 A JP 2013549683A JP 2013549683 A JP2013549683 A JP 2013549683A JP 6023082 B2 JP6023082 B2 JP 6023082B2
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ジー. マストロナルディ,ファブリツィオ
ジー. マストロナルディ,ファブリツィオ
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インセプタム リサーチ アンド セラピューティクス,インク.
インセプタム リサーチ アンド セラピューティクス,インク.
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4706—4-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
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    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • C—CHEMISTRY; METALLURGY
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    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof

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  • Health & Medical Sciences (AREA)
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2013549683A 2011-01-24 2012-01-24 精神神経性の疾病を処置するためのプロスタグランジンを含む組成物 Expired - Fee Related JP6023082B2 (ja)

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US201161435546P 2011-01-24 2011-01-24
US61/435,546 2011-01-24
PCT/CA2012/050037 WO2012100347A1 (en) 2011-01-24 2012-01-24 Compositions comprising a prostaglandin for treating neuropsychiatric conditions

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JP2014502974A JP2014502974A (ja) 2014-02-06
JP2014502974A5 JP2014502974A5 (enExample) 2015-02-05
JP6023082B2 true JP6023082B2 (ja) 2016-11-09

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US (2) US9259409B2 (enExample)
EP (1) EP2667875A4 (enExample)
JP (1) JP6023082B2 (enExample)
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WO (1) WO2012100347A1 (enExample)

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US20130309330A1 (en) 2013-11-21
EP2667875A1 (en) 2013-12-04
WO2012100347A1 (en) 2012-08-02
CA2860453A1 (en) 2012-08-02
US9259409B2 (en) 2016-02-16
JP2014502974A (ja) 2014-02-06
CA2860453C (en) 2020-04-28
US20160113942A1 (en) 2016-04-28

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