JP6011543B2 - 糖尿病、肥満および関連疾患の治療のためのｇｐｒ１１９モジュレーターとしての縮合ジヒドロフラン - Google Patents

糖尿病、肥満および関連疾患の治療のためのｇｐｒ１１９モジュレーターとしての縮合ジヒドロフラン Download PDF

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JP6011543B2
JP6011543B2 JP2013543816A JP2013543816A JP6011543B2 JP 6011543 B2 JP6011543 B2 JP 6011543B2 JP 2013543816 A JP2013543816 A JP 2013543816A JP 2013543816 A JP2013543816 A JP 2013543816A JP 6011543 B2 JP6011543 B2 JP 6011543B2
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piperidine
dihydro
carboxylic acid
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JP2013545791A (ja
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ヒンメルスバッハ　フランク
フランク ヒンメルスバッハ
マティアス エックハルト
マティアス エックハルト
ニクラス ハイネ
ニクラス ハイネ
エルケ ランクコープフ
エルケ ランクコープフ
ベルント ノッセ
ベルント ノッセ
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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JP2013543816A 2010-12-17 2011-12-16 糖尿病、肥満および関連疾患の治療のためのｇｐｒ１１９モジュレーターとしての縮合ジヒドロフラン Active JP6011543B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10195814.8 2010-12-17
EP10195814 2010-12-17
PCT/EP2011/073067 WO2012080476A1 (en) 2010-12-17 2011-12-16 Fused dihydropyrans as gpr119 modulators for the treatment of diabetes, obesity and related diseases

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JP2013545791A JP2013545791A (ja) 2013-12-26
JP2013545791A5 JP2013545791A5 (OSRAM) 2015-02-05
JP6011543B2 true JP6011543B2 (ja) 2016-10-19

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US (1) US8669271B2 (OSRAM)
EP (1) EP2651931B1 (OSRAM)
JP (1) JP6011543B2 (OSRAM)
AR (1) AR084349A1 (OSRAM)
UY (1) UY33805A (OSRAM)
WO (1) WO2012080476A1 (OSRAM)

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EP2686312B1 (en) 2011-03-14 2016-08-31 Boehringer Ingelheim International GmbH N-cyclopropyl-n-piperidinylbenzamides as gpr119 modulators
EP2718288B1 (en) 2011-06-09 2015-03-11 Boehringer Ingelheim International GmbH Substituted piperidines as gpr119 modulators for the treatment of metabolic disorders
EP2718279B1 (en) * 2011-06-09 2016-08-10 Rhizen Pharmaceuticals SA Novel compounds as modulators of gpr-119
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EP2651931A1 (en) 2013-10-23
AR084349A1 (es) 2013-05-08
US20120322784A1 (en) 2012-12-20
JP2013545791A (ja) 2013-12-26
US8669271B2 (en) 2014-03-11
EP2651931B1 (en) 2015-08-19
WO2012080476A1 (en) 2012-06-21
UY33805A (es) 2012-07-31

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