JP5885832B2 - ネプリライシン阻害剤 - Google Patents

ネプリライシン阻害剤 Download PDF

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JP5885832B2
JP5885832B2 JP2014513549A JP2014513549A JP5885832B2 JP 5885832 B2 JP5885832 B2 JP 5885832B2 JP 2014513549 A JP2014513549 A JP 2014513549A JP 2014513549 A JP2014513549 A JP 2014513549A JP 5885832 B2 JP5885832 B2 JP 5885832B2
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alkyl
alkylene
compound
coor
phenyl
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JP2014528903A5 (enExample
JP2014528903A (ja
Inventor
メリッサ フルーリー，
メリッサ フルーリー，
ローランド ジェンドロン，
ローランド ジェンドロン，
アダム ディー． ヒューズ，
アダム ディー． ヒューズ，
ジェーン シュミット，
ジェーン シュミット，
Original Assignee
セラヴァンス バイオファーマ アール＆ディー アイピー， エルエルシー
セラヴァンス バイオファーマ アール＆ディー アイピー， エルエルシー
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    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
    • C07D231/26—1-Phenyl-3-methyl-5- pyrazolones, unsubstituted or substituted on the phenyl ring
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