JP5797655B2 - 消化管障害のためのオピオイド受容体アンタゴニストの使用 - Google Patents

消化管障害のためのオピオイド受容体アンタゴニストの使用 Download PDF

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Publication number
JP5797655B2
JP5797655B2 JP2012529934A JP2012529934A JP5797655B2 JP 5797655 B2 JP5797655 B2 JP 5797655B2 JP 2012529934 A JP2012529934 A JP 2012529934A JP 2012529934 A JP2012529934 A JP 2012529934A JP 5797655 B2 JP5797655 B2 JP 5797655B2
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compound
dose
opioid
day
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JP2013505260A (ja
JP2013505260A5 (enExample
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ウツドワード，リチヤード・エム
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アドラー・コーポレーション
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2012529934A 2009-09-18 2010-09-17 消化管障害のためのオピオイド受容体アンタゴニストの使用 Expired - Fee Related JP5797655B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24361609P 2009-09-18 2009-09-18
US61/243,616 2009-09-18
PCT/US2010/049311 WO2011035142A1 (en) 2009-09-18 2010-09-17 Use of opioid receptor antagonist for gastrointestinal tract disorders

Publications (3)

Publication Number Publication Date
JP2013505260A JP2013505260A (ja) 2013-02-14
JP2013505260A5 JP2013505260A5 (enExample) 2013-11-07
JP5797655B2 true JP5797655B2 (ja) 2015-10-21

Family

ID=43216894

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012529934A Expired - Fee Related JP5797655B2 (ja) 2009-09-18 2010-09-17 消化管障害のためのオピオイド受容体アンタゴニストの使用

Country Status (19)

Country Link
US (1) US20110071163A1 (enExample)
EP (1) EP2477627B1 (enExample)
JP (1) JP5797655B2 (enExample)
KR (1) KR20120092592A (enExample)
CN (2) CN102695508A (enExample)
AU (1) AU2010295464B2 (enExample)
BR (1) BR112012006069A8 (enExample)
CA (1) CA2774021A1 (enExample)
CL (1) CL2012000676A1 (enExample)
CO (1) CO6531453A2 (enExample)
HK (1) HK1210959A1 (enExample)
IL (1) IL218679A0 (enExample)
MX (1) MX342548B (enExample)
NZ (1) NZ598783A (enExample)
PE (1) PE20120991A1 (enExample)
RU (1) RU2561873C2 (enExample)
TW (1) TW201118084A (enExample)
WO (1) WO2011035142A1 (enExample)
ZA (1) ZA201201954B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE027856T2 (en) * 2012-12-28 2016-11-28 Inst Medycyny Doswiadczalnej I Klinicznej Im Miroslawa Mossakowskiego Polskiej Akademii Nauk Peptidomimetics and their use
TW201808937A (zh) 2016-05-20 2018-03-16 艾斯提夫博士實驗股份有限公司 針對疼痛具有多模態活性的四氫哌喃和噻喃衍生物
CN106117190B (zh) * 2016-06-21 2019-03-29 山东川成医药股份有限公司 一种倍福普兰的合成方法

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MXPA01003197A (es) 1998-09-28 2004-04-21 Warner Lambert Co Suministro enterico y colonico utilizando capsulas de chpm.
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PT1220849E (pt) * 1999-10-15 2004-10-29 Sucampo Ag Composicao de compostos biciclicos e metodo para a sua estabilizacao
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Also Published As

Publication number Publication date
CN104958298A (zh) 2015-10-07
BR112012006069A8 (pt) 2017-10-10
NZ598783A (en) 2013-07-26
AU2010295464B2 (en) 2015-11-26
IL218679A0 (en) 2012-05-31
KR20120092592A (ko) 2012-08-21
PE20120991A1 (es) 2012-08-01
CN102695508A (zh) 2012-09-26
ZA201201954B (en) 2012-11-28
WO2011035142A1 (en) 2011-03-24
HK1210959A1 (en) 2016-05-13
US20110071163A1 (en) 2011-03-24
BR112012006069A2 (pt) 2016-03-29
MX2012003310A (es) 2012-07-17
RU2561873C2 (ru) 2015-09-10
MX342548B (es) 2016-10-04
AU2010295464A1 (en) 2012-04-12
EP2477627A1 (en) 2012-07-25
EP2477627B1 (en) 2018-08-15
JP2013505260A (ja) 2013-02-14
TW201118084A (en) 2011-06-01
RU2012115450A (ru) 2013-10-27
CO6531453A2 (es) 2012-09-28
CA2774021A1 (en) 2011-03-24
CL2012000676A1 (es) 2012-10-19

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