JP5779183B2 - ピリド［４，３−ｂ］インドールおよび使用方法 - Google Patents
ピリド［４，３−ｂ］インドールおよび使用方法 Download PDFInfo
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- JP5779183B2 JP5779183B2 JP2012531042A JP2012531042A JP5779183B2 JP 5779183 B2 JP5779183 B2 JP 5779183B2 JP 2012531042 A JP2012531042 A JP 2012531042A JP 2012531042 A JP2012531042 A JP 2012531042A JP 5779183 B2 JP5779183 B2 JP 5779183B2
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- alkoxy
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24525909P | 2009-09-23 | 2009-09-23 | |
| US24514009P | 2009-09-23 | 2009-09-23 | |
| US61/245,259 | 2009-09-23 | ||
| US61/245,140 | 2009-09-23 | ||
| PCT/US2010/050078 WO2011038161A1 (en) | 2009-09-23 | 2010-09-23 | Pyrido[4,3-b]indoles and methods of use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013505945A JP2013505945A (ja) | 2013-02-21 |
| JP2013505945A5 JP2013505945A5 (https=) | 2013-11-07 |
| JP5779183B2 true JP5779183B2 (ja) | 2015-09-16 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2012531042A Expired - Fee Related JP5779183B2 (ja) | 2009-09-23 | 2010-09-23 | ピリド［４，３−ｂ］インドールおよび使用方法 |
Country Status (8)
| Country | Link |
|---|---|
| US (5) | US8859561B2 (https=) |
| EP (1) | EP2480078A4 (https=) |
| JP (1) | JP5779183B2 (https=) |
| CN (1) | CN102711468B (https=) |
| AU (1) | AU2010298166B2 (https=) |
| BR (1) | BR112012006640A2 (https=) |
| CA (1) | CA2775328A1 (https=) |
| WO (1) | WO2011038161A1 (https=) |
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| RU2007139634A (ru) | 2007-10-25 | 2009-04-27 | Сергей Олегович Бачурин (RU) | Новые тиазол-, триазол- или оксадиазол-содержащие тетрациклические соединения |
| RU2544856C2 (ru) | 2008-01-25 | 2015-03-20 | Сергей Олегович Бачурин | НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ |
| CL2009000725A1 (es) | 2008-03-24 | 2009-05-29 | Medivation Technologies Inc | Compuestos derivados de heterociclos con uniones puente sustituidos, moduladores de receptores adrenergicos, de serotonina, de dopamina y de histaminas; composicion farmaceutica; kit farmaceutico; y su uso en el tratamiento del trastorno cognitivo y trastorno psicotico. |
| WO2009120717A2 (en) | 2008-03-24 | 2009-10-01 | Medivation Technologies, Inc. | Pyrido [3, 4-b] indoles and methods of use |
| TWI477503B (zh) * | 2008-10-31 | 2015-03-21 | Medivation Technologies Inc | 含有剛性部分之吡啶并〔４，３－ｂ〕吲哚 |
| AU2009308708B2 (en) | 2008-10-31 | 2015-11-19 | Medivation Technologies, Inc. | Azepino [4, 5-b] indoles and methods of use |
| EP2424366B1 (en) | 2009-04-29 | 2016-02-17 | Medivation Technologies, Inc. | Pyrido [4, 3-b]indoles and methods of use |
| CA2760541A1 (en) | 2009-04-29 | 2010-11-04 | Medivation Technologies, Inc. | Pyrido[4,3-b] indoles and methods of use |
| WO2011038164A1 (en) | 2009-09-23 | 2011-03-31 | Medivation Technologies, Inc. | Bridged heterocyclic compounds and methods of use |
| CA2775328A1 (en) | 2009-09-23 | 2011-03-31 | Medivation Technologies, Inc. | Pyrido[4,3-b]indoles and methods of use |
| US9079904B2 (en) | 2009-09-23 | 2015-07-14 | Medivation Technologies, Inc. | Pyrido[3,4-B]indoles and methods of use |
| WO2011103433A1 (en) | 2010-02-18 | 2011-08-25 | Medivation Technologies, Inc. | Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use |
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| WO2011103430A1 (en) | 2010-02-19 | 2011-08-25 | Medivation Technologies, Inc. | Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use |
| US8791132B2 (en) | 2011-02-18 | 2014-07-29 | Medivation Technologies, Inc. | Compounds and methods for treatment of hypertension |
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| US9434747B2 (en) | 2011-02-18 | 2016-09-06 | Medivation Technologies, Inc. | Methods of treating diabetes |
| WO2012112963A1 (en) | 2011-02-18 | 2012-08-23 | Medivation Technologies, Inc. | Compounds and methods for treatment of hypertension |
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| EP3704271B1 (en) * | 2017-11-02 | 2026-01-28 | California Institute of Technology | Neurokinin antagonists and uses thereof |
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| CA2748813C (en) | 2009-01-09 | 2018-07-10 | Board Of Regents Of The University Of Texas System | Pro-neurogenic compounds |
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| WO2011103430A1 (en) | 2010-02-19 | 2011-08-25 | Medivation Technologies, Inc. | Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use |
| CA2804161A1 (en) | 2010-07-07 | 2012-01-12 | Board Of Regents Of The University Of Texas System | Pro-neurogenic compounds |
| US9434747B2 (en) | 2011-02-18 | 2016-09-06 | Medivation Technologies, Inc. | Methods of treating diabetes |
| US8791132B2 (en) | 2011-02-18 | 2014-07-29 | Medivation Technologies, Inc. | Compounds and methods for treatment of hypertension |
| WO2012112964A2 (en) | 2011-02-18 | 2012-08-23 | Medivation Technologies, Inc. | PYRIDO[4,3-b]INDOLE AND PYRIDO[3,4-b]INDOLE DERIVATIVES AND METHODS OF USE |
| WO2012112963A1 (en) | 2011-02-18 | 2012-08-23 | Medivation Technologies, Inc. | Compounds and methods for treatment of hypertension |
| WO2014031170A1 (en) | 2012-08-22 | 2014-02-27 | Medivation Technologies, Inc. | Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use |
| WO2014031165A1 (en) | 2012-08-22 | 2014-02-27 | Medivation Technologies, Inc. | Compounds and methods of treating diabetes |
| CN108329253A (zh) | 2012-08-24 | 2018-07-27 | 得克萨斯州大学系统董事会 | 前神经原性化合物 |
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-
2010
- 2010-09-23 CA CA2775328A patent/CA2775328A1/en not_active Abandoned
- 2010-09-23 EP EP10819490A patent/EP2480078A4/en not_active Withdrawn
- 2010-09-23 BR BR112012006640A patent/BR112012006640A2/pt not_active IP Right Cessation
- 2010-09-23 AU AU2010298166A patent/AU2010298166B2/en not_active Ceased
- 2010-09-23 CN CN201080052847.4A patent/CN102711468B/zh not_active Expired - Fee Related
- 2010-09-23 WO PCT/US2010/050078 patent/WO2011038161A1/en not_active Ceased
- 2010-09-23 US US12/889,338 patent/US8859561B2/en not_active Expired - Fee Related
- 2010-09-23 JP JP2012531042A patent/JP5779183B2/ja not_active Expired - Fee Related
-
2013
- 2013-03-08 US US13/791,871 patent/US9045482B2/en not_active Expired - Fee Related
- 2013-03-08 US US13/791,570 patent/US20130184303A1/en not_active Abandoned
- 2013-03-08 US US13/791,874 patent/US9199996B2/en not_active Expired - Fee Related
-
2014
- 2014-09-12 US US14/485,238 patent/US9580425B2/en not_active Expired - Fee Related
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| US20110245272A1 (en) | 2011-10-06 |
| WO2011038161A1 (en) | 2011-03-31 |
| US8859561B2 (en) | 2014-10-14 |
| US20130184304A1 (en) | 2013-07-18 |
| AU2010298166A1 (en) | 2012-04-19 |
| US20130184303A1 (en) | 2013-07-18 |
| AU2010298166B2 (en) | 2015-09-17 |
| CN102711468B (zh) | 2014-07-09 |
| JP2013505945A (ja) | 2013-02-21 |
| US20150005322A1 (en) | 2015-01-01 |
| CN102711468A (zh) | 2012-10-03 |
| EP2480078A1 (en) | 2012-08-01 |
| US20130190344A1 (en) | 2013-07-25 |
| US9199996B2 (en) | 2015-12-01 |
| CA2775328A1 (en) | 2011-03-31 |
| HK1176811A1 (en) | 2013-08-09 |
| EP2480078A4 (en) | 2013-03-06 |
| BR112012006640A2 (pt) | 2019-09-24 |
| US9045482B2 (en) | 2015-06-02 |
| US9580425B2 (en) | 2017-02-28 |
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