|
US4360673A
(en)
|
1980-03-31 |
1982-11-23 |
Schering Corporation |
5 Phenyl-1,3-alkano-1,2,3,4,4a,9b-hexahydropyrido [4,3-b]indoles
|
|
US5273977A
(en)
|
1990-11-05 |
1993-12-28 |
Warner-Lambert Company |
Substituted tetrahydropyridines and hydroxypiperidines as central nervous system agents
|
|
ATE152718T1
(de)
*
|
1991-08-15 |
1997-05-15 |
Ciba Geigy Ag |
N-acyl-n-heterocyclyl- oder naphthylalkyl- aminosäuren als angiotensin ii antagonisten
|
|
US5250537A
(en)
|
1992-03-13 |
1993-10-05 |
Scios Nova Inc. |
5,6,7,8,9,10-hexahydro-7,10-iminocyclohept[b]indole,-6,7,8,9,10-hexahydro-7,11-imino-5H-cyclooct[b]indole and substituted derivatives
|
|
RU2106864C1
(ru)
|
1995-10-23 |
1998-03-20 |
Николай Серафимович Зефиров |
Средство для лечения болезни альцгеймера
|
|
US6251893B1
(en)
|
1998-06-15 |
2001-06-26 |
Nps Allelix Corp. |
Bicyclic piperidine and piperazine compounds having 5-HT6 receptor affinity
|
|
US20070179174A1
(en)
|
2003-12-08 |
2007-08-02 |
Bachurin Sergei O |
Methods and compositions for slowing aging
|
|
RU2283108C2
(ru)
|
2003-12-08 |
2006-09-10 |
Сергей Олегович Бачурин |
ГЕРОПРОТЕКТОР НА ОСНОВЕ ГИДРИРОВАННЫХ ПИРИДО(4,3-b) ИНДОЛОВ (ВАРИАНТЫ), ФАРМАКОЛОГИЧЕСКОЕ СРЕДСТВО НА ЕГО ОСНОВЕ И СПОСОБ ЕГО ПРИМЕНЕНИЯ
|
|
BRPI0614944A2
(pt)
|
2005-08-19 |
2011-04-26 |
Elan Pharm Inc |
inibidores sulfonamido n-bicìclicos ponte de gama-secretase
|
|
WO2007041697A2
(en)
|
2005-10-04 |
2007-04-12 |
Medivation, Inc. |
Hydrogenated pyrido-indole compounds for the treatment of huntington ' s disease
|
|
RU2338537C2
(ru)
|
2006-01-25 |
2008-11-20 |
Сергей Олегович Бачурин |
СРЕДСТВО ДЛЯ ЛЕЧЕНИЯ ШИЗОФРЕНИИ НА ОСНОВЕ ГИДРИРОВАННЫХ ПИРИДО(4,3-b)ИНДОЛОВ (ВАРИАНТЫ), ФАРМАКОЛОГИЧЕСКОЕ СРЕДСТВО НА ЕГО ОСНОВЕ И СПОСОБ ЕГО ПРИМЕНЕНИЯ
|
|
WO2008036400A2
(en)
|
2006-09-20 |
2008-03-27 |
Medivation Neurology, Inc. |
Hydrogenated pyrido [4,3-b] indoles such as dimebon for treating canine cognitive dysfunction syndrome
|
|
WO2008036410A2
(en)
|
2006-09-20 |
2008-03-27 |
Medivation Neurology, Inc. |
Methods and compositions for treating amyotrophic lateral sclerosis (als)
|
|
AU2007309390A1
(en)
|
2006-10-27 |
2008-05-02 |
Medivation Neurology, Inc. |
Methods and combination therapies for treating Alzheimer's disease
|
|
RU2329044C1
(ru)
|
2006-11-16 |
2008-07-20 |
Андрей Александрович Иващенко |
Лиганды 5-ht6 рецепторов, фармацевтическая композиция, способ ее получения и лекарственное средство
|
|
RU2334514C1
(ru)
|
2006-12-01 |
2008-09-27 |
Институт физиологически активных веществ Российской Академии наук |
СРЕДСТВО ДЛЯ УЛУЧШЕНИЯ КОГНИТИВНЫХ ФУНКЦИЙ И ПАМЯТИ НА ОСНОВЕ ГИДРИРОВАННЫХ ПИРИДО (4,3-b) ИНДОЛОВ (ВАРИАНТЫ), ФАРМАКОЛОГИЧЕСКОЕ СРЕДСТВО НА ЕГО ОСНОВЕ И СПОСОБ ЕГО ПРИМЕНЕНИЯ
|
|
RU2340342C2
(ru)
|
2006-12-07 |
2008-12-10 |
Сергей Олегович Бачурин |
СРЕДСТВО ДЛЯ ЛЕЧЕНИЯ ОСТРЫХ И ХРОНИЧЕСКИХ НАРУШЕНИЙ МОЗГОВОГО КРОВООБРАЩЕНИЯ, В ТОМ ЧИСЛЕ ИНСУЛЬТА, НА ОСНОВЕ ГИДРИРОВАННЫХ ПИРИДО[4,3-b]ИНДОЛОВ (ВАРИАНТЫ), ФАРМАКОЛОГИЧЕСКОЕ СРЕДСТВО НА ЕГО ОСНОВЕ И СПОСОБ ЕГО ПРИМЕНЕНИЯ
|
|
RU2338745C1
(ru)
|
2007-03-21 |
2008-11-20 |
Андрей Александрович Иващенко |
ЗАМЕЩЕННЫЕ 2,3,4,5-ТЕТРАГИДРО-1Н-ПИРИДО[4,3-b]ИНДОЛЫ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
|
|
RU2339637C1
(ru)
*
|
2007-04-05 |
2008-11-27 |
Андрей Александрович Иващенко |
Блокаторы гистаминного рецептора для фармацевтических композиций, обладающих противоаллергическим и аутоиммунным действием
|
|
AU2008236872B2
(en)
|
2007-04-05 |
2013-01-17 |
Alla Chem, Llc |
Substituted 2,3,4,5-tetrahydro-1h-pyrido[4,3-b]indoles, methods for the production and use thereof
|
|
JP2010528016A
(ja)
|
2007-05-25 |
2010-08-19 |
メディベーション ニューロロジー, インコーポレイテッド |
細胞を刺激するための方法および組成物
|
|
RU2338533C1
(ru)
|
2007-06-28 |
2008-11-20 |
Сергей Олегович Бачурин |
СРЕДСТВО, ОБЛАДАЮЩЕЕ АНКСИОЛИТИЧЕСКИМ ДЕЙСТВИЕМ, НА ОСНОВЕ ГИДРИРОВАННЫХ ПИРИДО(4,3-b)ИНДОЛОВ (ВАРИАНТЫ), ФАРМАКОЛОГИЧЕСКОЕ СРЕДСТВО НА ЕГО ОСНОВЕ И СПОСОБ ЕГО ПРИМЕНЕНИЯ
|
|
WO2009017836A1
(en)
|
2007-08-01 |
2009-02-05 |
Medivation Neurology, Inc. |
Methods and compositions for treating schizophrenia using antipsychotic combination therapy
|
|
WO2009039420A1
(en)
|
2007-09-21 |
2009-03-26 |
Medivation Neurology, Inc. |
Methods and compositions for treating neuronal death mediated ocular diseases
|
|
RU2007139634A
(ru)
|
2007-10-25 |
2009-04-27 |
Сергей Олегович Бачурин (RU) |
Новые тиазол-, триазол- или оксадиазол-содержащие тетрациклические соединения
|
|
WO2009082268A2
(ru)
|
2007-12-21 |
2009-07-02 |
Alla Chem, Llc |
ЛИГАНДЫ α-АДРЕНОЦЕПТОРОВ, ДОПАМИНОВЫХ, ГИСТАМИНОВЫХ, ИМИДАЗОЛИНОВЫХ И СЕРОТОНИНОВЫХ РЕЦЕПТОРОВ И ИХ ПРИМЕНЕНИЕ
|
|
RU2544856C2
(ru)
|
2008-01-25 |
2015-03-20 |
Сергей Олегович Бачурин |
НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ
|
|
WO2009111540A1
(en)
|
2008-03-04 |
2009-09-11 |
Medivation Neurology, Inc. |
Methods for preparing pyridylethyl-substituted carbolines
|
|
CN102046625B
(zh)
|
2008-03-24 |
2015-04-08 |
梅迪维新技术公司 |
桥连杂环化合物及其使用方法
|
|
TWI443098B
(zh)
|
2008-03-24 |
2014-07-01 |
Medivation Technologies Inc |
吡啶并〔3,4-b〕吲哚及使用方法
|
|
AU2009228647B2
(en)
|
2008-03-27 |
2013-07-04 |
Grunenthal Gmbh |
Substituted spirocyclic cyclohexane derivatives
|
|
WO2009135091A1
(en)
|
2008-04-30 |
2009-11-05 |
Medivation Technologies, Inc. |
Use of asenapine and related compounds for the treatment of neuronal or non-neuronal diseases or conditions
|
|
WO2010014758A1
(en)
|
2008-07-30 |
2010-02-04 |
Edison Pharmaceuticals, Inc. |
Use of hydrogenated pyrido[4,3-b] indoles for the treatment of oxidative stress
|
|
CN102227431A
(zh)
|
2008-09-29 |
2011-10-26 |
雅培制药有限公司 |
吲哚和二氢吲哚衍生物及其应用方法
|
|
US9625475B2
(en)
|
2008-09-29 |
2017-04-18 |
Abbvie Inc. |
Indole and indoline derivatives and methods of use thereof
|
|
AU2009308706C1
(en)
|
2008-10-31 |
2016-01-21 |
Medivation Technologies, Inc. |
Pyrido (4,3-b) indoles containing rigid moieties
|
|
WO2010051503A1
(en)
|
2008-10-31 |
2010-05-06 |
Medivation Technologies, Inc. |
Azepino [4, 5-b] indoles and methods of use
|
|
EP2385829B1
(en)
|
2009-01-09 |
2018-08-01 |
Board of Regents of the University of Texas System |
Pro-neurogenic compounds
|
|
US8362277B2
(en)
|
2009-01-09 |
2013-01-29 |
Board Of Regents Of The University Of Texas System |
Pro-neurogenic compounds
|
|
US9095572B2
(en)
|
2009-01-09 |
2015-08-04 |
Board Of Regents Of The University Of Texas System |
Pro-neurogenic compounds
|
|
US9962368B2
(en)
|
2009-01-09 |
2018-05-08 |
Board Of Regents Of The University Of Texas System |
Pro-neurogenic compounds
|
|
JP5827943B2
(ja)
|
2009-04-29 |
2015-12-02 |
メディベイション テクノロジーズ, インコーポレイテッド |
ピリド[4,3−b]インドールおよびその使用方法
|
|
CA2760541A1
(en)
|
2009-04-29 |
2010-11-04 |
Medivation Technologies, Inc. |
Pyrido[4,3-b] indoles and methods of use
|
|
WO2011008312A2
(en)
*
|
2009-07-14 |
2011-01-20 |
Abbott Laboratories |
Indole and indoline derivatives and methods of use thereof
|
|
RU2009128817A
(ru)
|
2009-07-28 |
2011-02-10 |
Общество с ограниченной ответственностью "Инномед" (RU) |
Производные гидрированных пиридо[4,3-b]индолов, фармацевтическая композиция, способы получения и применения
|
|
WO2011014695A1
(en)
|
2009-07-29 |
2011-02-03 |
Medivation Technologies, Inc. |
New 2,3,4,5-tetrahydro-1h-pyrido[4,3-b] indoles and methods of use
|
|
EP2480079A4
(en)
|
2009-09-23 |
2015-04-08 |
Medivation Technologies Inc |
PYRIDO- (3,4-B-) INDOLE AND USE METHOD THEREFOR
|
|
WO2011038163A1
(en)
|
2009-09-23 |
2011-03-31 |
Medivation Technologies, Inc. |
Pyrido[3,4-b]indoles and methods of use
|
|
AU2010298169B2
(en)
|
2009-09-23 |
2015-10-29 |
Medivation Technologies, Inc. |
Bridged heterocyclic compounds and methods of use
|
|
EP2480078A4
(en)
|
2009-09-23 |
2013-03-06 |
Medivation Technologies Inc |
PYRIDO- [4,3-B] INDOLE AND USE METHOD THEREFOR
|
|
US9034865B2
(en)
|
2010-02-18 |
2015-05-19 |
Medivation Technologies, Inc. |
Pyrido [4,3-B] indole and pyrido [3,4-B] indole derivatives and methods of use
|
|
WO2011103487A1
(en)
|
2010-02-18 |
2011-08-25 |
Medivation Technologies, Inc. |
Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use
|
|
US9193728B2
(en)
|
2010-02-18 |
2015-11-24 |
Medivation Technologies, Inc. |
Fused tetracyclic pyrido [4,3-B] indole and pyrido [3,4-B] indole derivatives and methods of use
|
|
WO2011103485A1
(en)
|
2010-02-18 |
2011-08-25 |
Medivation Technologies, Inc. |
Fused tetracyclic pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use
|
|
WO2011103430A1
(en)
|
2010-02-19 |
2011-08-25 |
Medivation Technologies, Inc. |
Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use
|
|
WO2011103448A1
(en)
|
2010-02-19 |
2011-08-25 |
Medivation Technologies, Inc. |
Methods and compositions for treating psychotic disorders using antipsychotic combination therapy
|
|
US20140155384A1
(en)
|
2011-02-18 |
2014-06-05 |
Medivation Technologies, Inc. |
Compounds and methods of treating diabetes
|
|
CN103476417A
(zh)
|
2011-02-18 |
2013-12-25 |
梅迪维新技术公司 |
治疗糖尿病的化合物和方法
|
|
US9434747B2
(en)
|
2011-02-18 |
2016-09-06 |
Medivation Technologies, Inc. |
Methods of treating diabetes
|
|
US9035056B2
(en)
|
2011-02-18 |
2015-05-19 |
Medivation Technologies, Inc. |
Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use
|
|
EP2887805A4
(en)
|
2012-08-22 |
2016-08-17 |
Medivation Technologies Inc |
COMPOUNDS AND METHOD FOR TREATING BLOOD HIGH PRESSURE
|
|
WO2014031170A1
(en)
|
2012-08-22 |
2014-02-27 |
Medivation Technologies, Inc. |
Pyrido[4,3-b]indole and pyrido[3,4-b]indole derivatives and methods of use
|
|
CA2882923A1
(en)
|
2012-08-24 |
2014-02-27 |
Board Of Regents Of The University Of Texas System |
Pro-neurogenic compounds
|
|
US9422267B2
(en)
|
2012-12-26 |
2016-08-23 |
Medivation Technologies, Inc. |
Fused pyrimidine compounds and use thereof
|