JP5771524B2 - アリール−フェニル−スルホンアミド−シクロアルキル化合物とその使用 - Google Patents

アリール−フェニル−スルホンアミド−シクロアルキル化合物とその使用 Download PDF

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JP5771524B2
JP5771524B2 JP2011527394A JP2011527394A JP5771524B2 JP 5771524 B2 JP5771524 B2 JP 5771524B2 JP 2011527394 A JP2011527394 A JP 2011527394A JP 2011527394 A JP2011527394 A JP 2011527394A JP 5771524 B2 JP5771524 B2 JP 5771524B2
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JP2012502964A5 (enExample
JP2012502964A (ja
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ロバート グレイグ，イアン
ロバート グレイグ，イアン
メアリー シェリダン，ローズ
メアリー シェリダン，ローズ
フィッシャー，レイモンド
トーザー，マシュー，ジョン
クラセ，ユハ，アンドリュー
スミス，アンドリュー
タフネル，アンドリュー，ロバート
ホフ，ロベルト，ユルゲン ヴァント
ホフ，ロベルト，ユルゲン ヴァント
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ピムコ ２６６４ リミテッド
ピムコ ２６６４ リミテッド
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • A—HUMAN NECESSITIES
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07C311/20—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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JP2011527394A 2008-09-19 2009-09-18 アリール−フェニル−スルホンアミド−シクロアルキル化合物とその使用 Active JP5771524B2 (ja)

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Application Number Priority Date Filing Date Title
US9827108P 2008-09-19 2008-09-19
GB0817207.4 2008-09-19
GBGB0817207.4A GB0817207D0 (en) 2008-09-19 2008-09-19 therapeutic apsac compounds and their use
US61/098,271 2008-09-19
PCT/GB2009/002221 WO2010032009A1 (en) 2008-09-19 2009-09-18 Aryl-phenyl-sulfonamido-cycloalkyl compounds and their use

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JP2012502964A5 JP2012502964A5 (enExample) 2012-10-25
JP5771524B2 true JP5771524B2 (ja) 2015-09-02

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CA (1) CA2736971C (enExample)
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GB0817207D0 (en) 2008-09-19 2008-10-29 Pimco 2664 Ltd therapeutic apsac compounds and their use
US8394858B2 (en) * 2009-12-03 2013-03-12 Novartis Ag Cyclohexane derivatives and uses thereof
BR112014025201A2 (pt) 2012-04-10 2017-07-11 Sumitomo Dainippon Pharma Co Ltd derivado de indazol 1-substituído
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TWI745652B (zh) 2018-02-16 2021-11-11 美商基利科學股份有限公司 用於製備有療效化合物之方法及中間物
US11944611B2 (en) 2018-07-16 2024-04-02 Gilead Sciences, Inc. Capsid inhibitors for the treatment of HIV
GB201813312D0 (en) 2018-08-15 2018-09-26 Modern Biosciences Ltd Compounds and their therapeutic use
GB201905520D0 (en) * 2019-04-18 2019-06-05 Modern Biosciences Ltd Compounds and their therapeutic use
EP4643882A3 (en) 2019-11-26 2026-01-14 Gilead Sciences, Inc. Capsid inhibitors for the prevention of hiv
PT4440702T (pt) 2021-12-03 2025-08-13 Gilead Sciences Inc Compostos terapêuticos para a infecção pelo vírus do hiv
JP7765637B2 (ja) 2021-12-03 2025-11-06 ギリアード サイエンシーズ， インコーポレイテッド Ｈｉｖウイルス感染症のための治療化合物
WO2023102523A1 (en) 2021-12-03 2023-06-08 Gilead Sciences, Inc. Therapeutic compounds for hiv virus infection
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US9616037B2 (en) 2017-04-11
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US8822507B2 (en) 2014-09-02
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US20150266815A1 (en) 2015-09-24
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US20150141472A1 (en) 2015-05-21
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