JP5717752B2 - ピリピロペン誘導体の製造法 - Google Patents
ピリピロペン誘導体の製造法 Download PDFInfo
- Publication number
- JP5717752B2 JP5717752B2 JP2012540182A JP2012540182A JP5717752B2 JP 5717752 B2 JP5717752 B2 JP 5717752B2 JP 2012540182 A JP2012540182 A JP 2012540182A JP 2012540182 A JP2012540182 A JP 2012540182A JP 5717752 B2 JP5717752 B2 JP 5717752B2
- Authority
- JP
- Japan
- Prior art keywords
- compound
- acylating
- producing
- hydroxyl group
- cyclopropanecarbonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- 0 C[C@@]([C@](CC[C@]1(C)[C@@]([C@]2O)[C@@](C)([C@](C3)O)OC(C=C(c4cccnc4)O4)=C2C4=O)O*)[C@@]13NC Chemical compound C[C@@]([C@](CC[C@]1(C)[C@@]([C@]2O)[C@@](C)([C@](C3)O)OC(C=C(c4cccnc4)O4)=C2C4=O)O*)[C@@]13NC 0.000 description 2
Images
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2012540182A JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010044416 | 2010-03-01 | ||
| JP2010044416 | 2010-03-01 | ||
| JP2012540182A JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
| PCT/JP2010/070414 WO2011108155A1 (en) | 2010-03-01 | 2010-11-10 | Process for producing pyripyropene derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013521224A JP2013521224A (ja) | 2013-06-10 |
| JP2013521224A5 JP2013521224A5 (https=) | 2014-01-09 |
| JP5717752B2 true JP5717752B2 (ja) | 2015-05-13 |
Family
ID=43528310
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012540182A Active JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US8853414B2 (https=) |
| EP (1) | EP2542555B1 (https=) |
| JP (1) | JP5717752B2 (https=) |
| KR (1) | KR101787789B1 (https=) |
| CN (1) | CN102947312B (https=) |
| AR (1) | AR078975A1 (https=) |
| BR (1) | BR112012021911B8 (https=) |
| CA (1) | CA2791660C (https=) |
| CR (1) | CR20120487A (https=) |
| DK (1) | DK2542555T3 (https=) |
| EC (1) | ECSP12012203A (https=) |
| ES (1) | ES2607191T3 (https=) |
| IL (1) | IL221651A (https=) |
| MX (1) | MX2012010173A (https=) |
| NZ (1) | NZ602719A (https=) |
| RU (1) | RU2578605C2 (https=) |
| TW (1) | TWI504602B (https=) |
| UA (1) | UA111151C2 (https=) |
| WO (1) | WO2011108155A1 (https=) |
| ZA (1) | ZA201207335B (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2426124B1 (en) * | 2009-05-13 | 2013-08-07 | Meiji Seika Pharma Co., Ltd. | Process for producing pyripyropene derivative |
| UA111151C2 (uk) | 2010-03-01 | 2016-04-11 | Мейдзі Сейка Фарма Ко., Лтд. | Спосіб одержання похідних пірипіропену |
| ES2534745T3 (es) * | 2010-09-14 | 2015-04-28 | Basf Se | Composición que contiene un insecticida de piripiropeno y un adyuvante |
| JP6174057B2 (ja) * | 2012-03-12 | 2017-08-02 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | ピリピロペン殺虫剤の水性懸濁濃厚製剤の調製方法 |
| AU2014206958B2 (en) * | 2013-01-16 | 2017-08-10 | Basf Se | Method for preparing a pyripyropene compound |
| JP6215355B2 (ja) * | 2013-01-25 | 2017-10-18 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | 水性懸濁製剤の調製方法 |
| ES2705537T3 (es) | 2013-03-28 | 2019-03-25 | Basf Se | Producción de piripiropenos a partir de biomasa seca |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5192887A (en) * | 1991-09-23 | 1993-03-09 | Emerson Electric Co. | Starting multi-speed motors at a low speed connection |
| JP3233476B2 (ja) | 1992-10-22 | 2001-11-26 | 社団法人北里研究所 | Fo−1289物質およびその製造法 |
| JPH08239385A (ja) | 1995-03-03 | 1996-09-17 | Kitasato Inst:The | Fo−1289物質およびその製造法 |
| JP3725198B2 (ja) * | 1995-03-27 | 2005-12-07 | 社団法人北里研究所 | ピリピロペン誘導体 |
| JPH08269065A (ja) | 1995-04-03 | 1996-10-15 | Kitasato Inst:The | ピリピロペン誘導体 |
| KR100522446B1 (ko) | 2003-01-07 | 2005-10-18 | 한국생명공학연구원 | 아실 코에이:콜레스테롤 아실 트란스퍼라제의 저해활성을갖는 화합물 또는 그 염을 유효성분으로 하는 살충제 |
| JP5179174B2 (ja) | 2004-05-28 | 2013-04-10 | ノバルティス ファーマ アーゲー | アルドステロンシンターゼ阻害剤としてのテトラヒドロ−イミダゾ[1,5−a]ピリジン誘導体 |
| US7491738B2 (en) | 2005-06-01 | 2009-02-17 | Meiji Seika Kaisha, Ltd. | Pest control agents |
| TWI388282B (zh) | 2005-06-01 | 2013-03-11 | Meiji Seika Pharma Co Ltd | 害蟲控制劑 |
| JP2008050997A (ja) | 2006-08-24 | 2008-03-06 | Matsushita Electric Ind Co Ltd | 密閉型電動圧縮機 |
| US8202890B2 (en) | 2006-11-30 | 2012-06-19 | Meiji Seika Pharma Co., Ltd. | Pest control agent |
| JP4488033B2 (ja) | 2007-02-06 | 2010-06-23 | ソニー株式会社 | 偏光素子及び液晶プロジェクター |
| EP2186815A4 (en) | 2007-08-13 | 2012-01-25 | Meiji Seika Kaisha | PROCESS FOR PREPARING A PYRIPYROPEN DERIVATIVE AND INTERMEDIATE PRODUCT |
| TW200936047A (en) | 2007-12-21 | 2009-09-01 | Meiji Seika Kaisha | Novel systemic pesticide |
| EP2426124B1 (en) | 2009-05-13 | 2013-08-07 | Meiji Seika Pharma Co., Ltd. | Process for producing pyripyropene derivative |
| UA111151C2 (uk) | 2010-03-01 | 2016-04-11 | Мейдзі Сейка Фарма Ко., Лтд. | Спосіб одержання похідних пірипіропену |
-
2010
- 2010-10-11 UA UAA201211289A patent/UA111151C2/uk unknown
- 2010-11-10 WO PCT/JP2010/070414 patent/WO2011108155A1/en not_active Ceased
- 2010-11-10 MX MX2012010173A patent/MX2012010173A/es active IP Right Grant
- 2010-11-10 DK DK10788151.8T patent/DK2542555T3/da active
- 2010-11-10 KR KR1020127025488A patent/KR101787789B1/ko active Active
- 2010-11-10 JP JP2012540182A patent/JP5717752B2/ja active Active
- 2010-11-10 CA CA2791660A patent/CA2791660C/en active Active
- 2010-11-10 RU RU2012141555/04A patent/RU2578605C2/ru active
- 2010-11-10 EP EP10788151.8A patent/EP2542555B1/en active Active
- 2010-11-10 CN CN201080065119.7A patent/CN102947312B/zh active Active
- 2010-11-10 ES ES10788151.8T patent/ES2607191T3/es active Active
- 2010-11-10 US US13/581,857 patent/US8853414B2/en active Active
- 2010-11-10 NZ NZ602719A patent/NZ602719A/en unknown
- 2010-11-10 BR BR112012021911A patent/BR112012021911B8/pt active IP Right Grant
- 2010-11-11 TW TW099139126A patent/TWI504602B/zh active
- 2010-11-11 AR ARP100104185A patent/AR078975A1/es active IP Right Grant
-
2012
- 2012-08-27 IL IL221651A patent/IL221651A/en active IP Right Grant
- 2012-09-26 CR CR20120487A patent/CR20120487A/es unknown
- 2012-10-01 ZA ZA2012/07335A patent/ZA201207335B/en unknown
- 2012-10-01 EC ECSP12012203 patent/ECSP12012203A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20130040180A (ko) | 2013-04-23 |
| US20130060042A1 (en) | 2013-03-07 |
| UA111151C2 (uk) | 2016-04-11 |
| CA2791660A1 (en) | 2011-09-09 |
| ES2607191T3 (es) | 2017-03-29 |
| WO2011108155A1 (en) | 2011-09-09 |
| RU2012141555A (ru) | 2014-04-10 |
| AU2010347354B2 (en) | 2016-09-01 |
| CA2791660C (en) | 2020-09-22 |
| JP2013521224A (ja) | 2013-06-10 |
| ZA201207335B (en) | 2014-01-29 |
| EP2542555A1 (en) | 2013-01-09 |
| KR101787789B1 (ko) | 2017-10-18 |
| CN102947312B (zh) | 2015-05-27 |
| AR078975A1 (es) | 2011-12-14 |
| ECSP12012203A (es) | 2013-06-28 |
| BR112012021911B1 (pt) | 2021-06-08 |
| TW201139447A (en) | 2011-11-16 |
| TWI504602B (zh) | 2015-10-21 |
| DK2542555T3 (da) | 2017-01-02 |
| US8853414B2 (en) | 2014-10-07 |
| RU2578605C2 (ru) | 2016-03-27 |
| BR112012021911A2 (pt) | 2015-09-29 |
| MX2012010173A (es) | 2012-10-03 |
| NZ602719A (en) | 2015-01-30 |
| CR20120487A (es) | 2013-01-11 |
| BR112012021911B8 (pt) | 2022-08-02 |
| AU2010347354A1 (en) | 2012-10-25 |
| IL221651A (en) | 2017-05-29 |
| EP2542555B1 (en) | 2016-09-21 |
| CN102947312A (zh) | 2013-02-27 |
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