JP5717752B2 - ピリピロペン誘導体の製造法 - Google Patents
ピリピロペン誘導体の製造法 Download PDFInfo
- Publication number
- JP5717752B2 JP5717752B2 JP2012540182A JP2012540182A JP5717752B2 JP 5717752 B2 JP5717752 B2 JP 5717752B2 JP 2012540182 A JP2012540182 A JP 2012540182A JP 2012540182 A JP2012540182 A JP 2012540182A JP 5717752 B2 JP5717752 B2 JP 5717752B2
- Authority
- JP
- Japan
- Prior art keywords
- compound
- acylating
- producing
- hydroxyl group
- cyclopropanecarbonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- 0 C[C@@]([C@](CC[C@]1(C)[C@@]([C@]2O)[C@@](C)([C@](C3)O)OC(C=C(c4cccnc4)O4)=C2C4=O)O*)[C@@]13NC Chemical compound C[C@@]([C@](CC[C@]1(C)[C@@]([C@]2O)[C@@](C)([C@](C3)O)OC(C=C(c4cccnc4)O4)=C2C4=O)O*)[C@@]13NC 0.000 description 2
Images
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2012540182A JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010044416 | 2010-03-01 | ||
| JP2010044416 | 2010-03-01 | ||
| PCT/JP2010/070414 WO2011108155A1 (en) | 2010-03-01 | 2010-11-10 | Process for producing pyripyropene derivatives |
| JP2012540182A JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013521224A JP2013521224A (ja) | 2013-06-10 |
| JP2013521224A5 JP2013521224A5 (https=) | 2014-01-09 |
| JP5717752B2 true JP5717752B2 (ja) | 2015-05-13 |
Family
ID=43528310
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012540182A Active JP5717752B2 (ja) | 2010-03-01 | 2010-11-10 | ピリピロペン誘導体の製造法 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US8853414B2 (https=) |
| EP (1) | EP2542555B1 (https=) |
| JP (1) | JP5717752B2 (https=) |
| KR (1) | KR101787789B1 (https=) |
| CN (1) | CN102947312B (https=) |
| AR (1) | AR078975A1 (https=) |
| BR (1) | BR112012021911B8 (https=) |
| CA (1) | CA2791660C (https=) |
| CR (1) | CR20120487A (https=) |
| DK (1) | DK2542555T3 (https=) |
| EC (1) | ECSP12012203A (https=) |
| ES (1) | ES2607191T3 (https=) |
| IL (1) | IL221651A (https=) |
| MX (1) | MX2012010173A (https=) |
| NZ (1) | NZ602719A (https=) |
| RU (1) | RU2578605C2 (https=) |
| TW (1) | TWI504602B (https=) |
| UA (1) | UA111151C2 (https=) |
| WO (1) | WO2011108155A1 (https=) |
| ZA (1) | ZA201207335B (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2426124T3 (da) | 2009-05-13 | 2013-09-30 | Meiji Seika Pharma Co Ltd | Fremgangsmåde til fremstilling af pyripyropene derivater |
| UA111151C2 (uk) | 2010-03-01 | 2016-04-11 | Мейдзі Сейка Фарма Ко., Лтд. | Спосіб одержання похідних пірипіропену |
| JP6425887B2 (ja) * | 2010-09-14 | 2018-11-21 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | ピリピロペン殺虫剤及び補助剤を含有する組成物 |
| EP2825043B1 (en) * | 2012-03-12 | 2018-09-05 | Basf Se | Method for producing an aqueous suspension concentrate formulation of a pyripyropene insecticide |
| KR102139923B1 (ko) * | 2013-01-16 | 2020-07-31 | 바스프 에스이 | 피리피로펜 화합물의 제조 방법 |
| EP2947989B1 (en) * | 2013-01-25 | 2016-12-07 | Basf Se | Method for producing aqueous suspension concentrate formulations |
| KR102139237B1 (ko) | 2013-03-28 | 2020-07-29 | 바스프 에스이 | 건조 바이오매스로부터의 피리피로펜의 제조 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5192887A (en) * | 1991-09-23 | 1993-03-09 | Emerson Electric Co. | Starting multi-speed motors at a low speed connection |
| JP3233476B2 (ja) | 1992-10-22 | 2001-11-26 | 社団法人北里研究所 | Fo−1289物質およびその製造法 |
| JPH08239385A (ja) | 1995-03-03 | 1996-09-17 | Kitasato Inst:The | Fo−1289物質およびその製造法 |
| JP3725198B2 (ja) | 1995-03-27 | 2005-12-07 | 社団法人北里研究所 | ピリピロペン誘導体 |
| JPH08269065A (ja) | 1995-04-03 | 1996-10-15 | Kitasato Inst:The | ピリピロペン誘導体 |
| KR100522446B1 (ko) | 2003-01-07 | 2005-10-18 | 한국생명공학연구원 | 아실 코에이:콜레스테롤 아실 트란스퍼라제의 저해활성을갖는 화합물 또는 그 염을 유효성분으로 하는 살충제 |
| CA2568159A1 (en) | 2004-05-28 | 2005-12-15 | Speedel Experimenta Ag | Tetrahydro-imidazo [1,5-a] pyridin derivatives as aldosterone synthase inhibitors |
| US7491738B2 (en) * | 2005-06-01 | 2009-02-17 | Meiji Seika Kaisha, Ltd. | Pest control agents |
| TWI388282B (zh) * | 2005-06-01 | 2013-03-11 | Meiji Seika Pharma Co Ltd | 害蟲控制劑 |
| JP2008050997A (ja) | 2006-08-24 | 2008-03-06 | Matsushita Electric Ind Co Ltd | 密閉型電動圧縮機 |
| ES2379928T3 (es) | 2006-11-30 | 2012-05-07 | Meiji Seika Kaisha Ltd. | Agente de control de plagas |
| JP4488033B2 (ja) | 2007-02-06 | 2010-06-23 | ソニー株式会社 | 偏光素子及び液晶プロジェクター |
| NZ583710A (en) | 2007-08-13 | 2012-03-30 | Meiji Seika Pharma Co Ltd | Method for producing pyripyropene derivative and production intermediate thereof |
| WO2009081851A1 (ja) | 2007-12-21 | 2009-07-02 | Meiji Seika Kaisha, Ltd. | 新規浸透移行性殺虫剤 |
| DK2426124T3 (da) | 2009-05-13 | 2013-09-30 | Meiji Seika Pharma Co Ltd | Fremgangsmåde til fremstilling af pyripyropene derivater |
| UA111151C2 (uk) | 2010-03-01 | 2016-04-11 | Мейдзі Сейка Фарма Ко., Лтд. | Спосіб одержання похідних пірипіропену |
-
2010
- 2010-10-11 UA UAA201211289A patent/UA111151C2/uk unknown
- 2010-11-10 NZ NZ602719A patent/NZ602719A/en unknown
- 2010-11-10 WO PCT/JP2010/070414 patent/WO2011108155A1/en not_active Ceased
- 2010-11-10 EP EP10788151.8A patent/EP2542555B1/en active Active
- 2010-11-10 JP JP2012540182A patent/JP5717752B2/ja active Active
- 2010-11-10 MX MX2012010173A patent/MX2012010173A/es active IP Right Grant
- 2010-11-10 ES ES10788151.8T patent/ES2607191T3/es active Active
- 2010-11-10 CA CA2791660A patent/CA2791660C/en active Active
- 2010-11-10 US US13/581,857 patent/US8853414B2/en active Active
- 2010-11-10 RU RU2012141555/04A patent/RU2578605C2/ru active
- 2010-11-10 DK DK10788151.8T patent/DK2542555T3/da active
- 2010-11-10 CN CN201080065119.7A patent/CN102947312B/zh active Active
- 2010-11-10 KR KR1020127025488A patent/KR101787789B1/ko active Active
- 2010-11-10 BR BR112012021911A patent/BR112012021911B8/pt active IP Right Grant
- 2010-11-11 TW TW099139126A patent/TWI504602B/zh active
- 2010-11-11 AR ARP100104185A patent/AR078975A1/es active IP Right Grant
-
2012
- 2012-08-27 IL IL221651A patent/IL221651A/en active IP Right Grant
- 2012-09-26 CR CR20120487A patent/CR20120487A/es unknown
- 2012-10-01 EC ECSP12012203 patent/ECSP12012203A/es unknown
- 2012-10-01 ZA ZA2012/07335A patent/ZA201207335B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2791660A1 (en) | 2011-09-09 |
| BR112012021911B8 (pt) | 2022-08-02 |
| US8853414B2 (en) | 2014-10-07 |
| EP2542555A1 (en) | 2013-01-09 |
| TW201139447A (en) | 2011-11-16 |
| US20130060042A1 (en) | 2013-03-07 |
| CA2791660C (en) | 2020-09-22 |
| KR20130040180A (ko) | 2013-04-23 |
| NZ602719A (en) | 2015-01-30 |
| CN102947312A (zh) | 2013-02-27 |
| AR078975A1 (es) | 2011-12-14 |
| CN102947312B (zh) | 2015-05-27 |
| DK2542555T3 (da) | 2017-01-02 |
| RU2012141555A (ru) | 2014-04-10 |
| TWI504602B (zh) | 2015-10-21 |
| AU2010347354B2 (en) | 2016-09-01 |
| BR112012021911B1 (pt) | 2021-06-08 |
| ECSP12012203A (es) | 2013-06-28 |
| BR112012021911A2 (pt) | 2015-09-29 |
| KR101787789B1 (ko) | 2017-10-18 |
| CR20120487A (es) | 2013-01-11 |
| JP2013521224A (ja) | 2013-06-10 |
| ES2607191T3 (es) | 2017-03-29 |
| ZA201207335B (en) | 2014-01-29 |
| RU2578605C2 (ru) | 2016-03-27 |
| MX2012010173A (es) | 2012-10-03 |
| UA111151C2 (uk) | 2016-04-11 |
| IL221651A (en) | 2017-05-29 |
| WO2011108155A1 (en) | 2011-09-09 |
| AU2010347354A1 (en) | 2012-10-25 |
| EP2542555B1 (en) | 2016-09-21 |
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