JP5711725B2 - ピリド［４，３−ｂ］インドールおよびその使用方法 - Google Patents

ピリド［４，３−ｂ］インドールおよびその使用方法 Download PDF

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JP5711725B2
JP5711725B2 JP2012508751A JP2012508751A JP5711725B2 JP 5711725 B2 JP5711725 B2 JP 5711725B2 JP 2012508751 A JP2012508751 A JP 2012508751A JP 2012508751 A JP2012508751 A JP 2012508751A JP 5711725 B2 JP5711725 B2 JP 5711725B2
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pyrido
indol
dihydro
methyl
compound
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JP2012525430A (ja
JP2012525430A5 (enExample
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ラジェンドラ パラスマル ジェイン，
ラジェンドラ パラスマル ジェイン，
サルバジット チャクラバルティ，
サルバジット チャクラバルティ，
Original Assignee
メディベイション テクノロジーズ， インコーポレイテッド
メディベイション テクノロジーズ， インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP2012508751A 2009-04-29 2010-04-29 ピリド［４，３−ｂ］インドールおよびその使用方法 Expired - Fee Related JP5711725B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN1136MU2009 2009-04-29
IN1136/MUM/2009 2009-04-29
US18126209P 2009-05-26 2009-05-26
US61/181,262 2009-05-26
PCT/US2010/033053 WO2010127177A1 (en) 2009-04-29 2010-04-29 Pyrido [4,3-b] indoles and methods of use

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Publication Number Publication Date
JP2012525430A JP2012525430A (ja) 2012-10-22
JP2012525430A5 JP2012525430A5 (enExample) 2013-06-27
JP5711725B2 true JP5711725B2 (ja) 2015-05-07

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US (2) US9255094B2 (enExample)
EP (1) EP2424364A4 (enExample)
JP (1) JP5711725B2 (enExample)
CN (1) CN102480955B (enExample)
AU (1) AU2010242910B2 (enExample)
BR (1) BRPI1006602A2 (enExample)
CA (1) CA2760541A1 (enExample)
WO (1) WO2010127177A1 (enExample)

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AU2010242910A1 (en) 2011-11-17
HK1170380A1 (en) 2013-03-01
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US20120136008A1 (en) 2012-05-31
WO2010127177A1 (en) 2010-11-04
EP2424364A4 (en) 2012-12-19
WO2010127177A8 (en) 2011-12-15
BRPI1006602A2 (pt) 2019-01-15
US9255094B2 (en) 2016-02-09
CA2760541A1 (en) 2010-11-04
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