JP5710268B2 - ８−アニリノイミダゾピリジン及びその抗ガン及び／又は抗炎症剤としての使用 - Google Patents

８−アニリノイミダゾピリジン及びその抗ガン及び／又は抗炎症剤としての使用 Download PDF

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JP5710268B2
JP5710268B2 JP2010539814A JP2010539814A JP5710268B2 JP 5710268 B2 JP5710268 B2 JP 5710268B2 JP 2010539814 A JP2010539814 A JP 2010539814A JP 2010539814 A JP2010539814 A JP 2010539814A JP 5710268 B2 JP5710268 B2 JP 5710268B2
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alkyl
compound
formula
imidazo
pyridine
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JP2011507888A5 (https=
JP2011507888A (ja
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スティーヴン プライス，
スティーヴン プライス，
ロバート ヒールド，
ロバート ヒールド，
パスカル ピエール アレクサンドル サヴィ，
パスカル ピエール アレクサンドル サヴィ，
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Genentech Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
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    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
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    • A61P17/00—Drugs for dermatological disorders
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    • A61P19/00—Drugs for skeletal disorders
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    • A61P19/00—Drugs for skeletal disorders
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P35/00—Antineoplastic agents
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    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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JP2010539814A 2007-12-19 2008-12-18 ８−アニリノイミダゾピリジン及びその抗ガン及び／又は抗炎症剤としての使用 Expired - Fee Related JP5710268B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US1515507P 2007-12-19 2007-12-19
US61/015,155 2007-12-19
US5402408P 2008-05-16 2008-05-16
US61/054,024 2008-05-16
PCT/US2008/087476 WO2009085980A1 (en) 2007-12-19 2008-12-18 8-anilin0imidaz0pyridines and their use as anti-cancer and/or anti-inflammatory agents

Publications (3)

Publication Number Publication Date
JP2011507888A JP2011507888A (ja) 2011-03-10
JP2011507888A5 JP2011507888A5 (https=) 2012-02-23
JP5710268B2 true JP5710268B2 (ja) 2015-04-30

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JP2010539814A Expired - Fee Related JP5710268B2 (ja) 2007-12-19 2008-12-18 ８−アニリノイミダゾピリジン及びその抗ガン及び／又は抗炎症剤としての使用

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Country Link
US (1) US8293763B2 (https=)
EP (1) EP2231662B1 (https=)
JP (1) JP5710268B2 (https=)
KR (1) KR20100101666A (https=)
CN (1) CN101903387B (https=)
AT (1) ATE513832T1 (https=)
AU (1) AU2008343062B2 (https=)
CA (1) CA2704125A1 (https=)
DK (1) DK2231662T3 (https=)
IL (1) IL205490A (https=)
NZ (1) NZ585306A (https=)
PL (1) PL2231662T3 (https=)
PT (1) PT2231662E (https=)
RU (1) RU2498985C2 (https=)
WO (1) WO2009085980A1 (https=)
ZA (1) ZA201003046B (https=)

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DK2231662T3 (da) 2011-08-29
RU2498985C2 (ru) 2013-11-20
PT2231662E (pt) 2011-09-12
KR20100101666A (ko) 2010-09-17
ATE513832T1 (de) 2011-07-15
IL205490A0 (en) 2010-12-30
EP2231662A1 (en) 2010-09-29
NZ585306A (en) 2012-05-25
JP2011507888A (ja) 2011-03-10
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US20100280063A1 (en) 2010-11-04
EP2231662B1 (en) 2011-06-22
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US8293763B2 (en) 2012-10-23
AU2008343062B2 (en) 2013-03-07
CN101903387A (zh) 2010-12-01
AU2008343062A1 (en) 2009-07-09

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